Novel low-molecular-weight hypromellose polymeric films for aqueous film coating applications

References

• Porter SC, Felton LA. (2010). Techniques to assess film coatings and evaluate film-coated products. Drug Dev Ind Pharm, 36:128–142.
   PubMed Web of Science ®Google Scholar
• Felton LA. (2007). Characterization of coating systems. AAPS Pharmscitech, 8:E112.
   PubMedGoogle Scholar
• Li SP, Martellucci SA, Bruce RD, Kinyon AC, Hay MB, Higgins JD 3rd. (2002). Evaluation of the film-coating properties of a hydroxyethyl cellulose/hydroxypropyl methylcellulose polymer system. Drug Dev Ind Pharm, 28:389–401.
   PubMed Web of Science ®Google Scholar
• Fell JT, Rowe RC, Newton JM. (1979). The mechanical strength of film-coated tablets. J Pharm Pharmacol, 31:69–72.
   PubMed Web of Science ®Google Scholar
• Dashevsky A, Ahmed AR, Mota J, Irfan M, Kolter K, Bodmeier RA. (2010). Effect of water-soluble polymers on the physical stability of aqueous polymeric dispersions and their implications on the drug release from coated pellets. Drug Dev Ind Pharm, 36:152–160.
   PubMed Web of Science ®Google Scholar
• Felton L, Haase M, Shah N, Zhang G, Infeld M, Malick A, McGinity JW. (1995). Physical and enteric properties of soft gelatin capsules coated with Eudragit L 30 D-55. Int J Pharm, 113:17–24.
   Web of Science ®Google Scholar
• Bussemer T, Bodmeier R. (2003). Formulation parameters affecting the performance of coated gelatin capsules with pulsatile release profiles. Int J Pharm, 267:59–68.
   PubMed Web of Science ®Google Scholar
• Mueller R, Kleinebudde P. (2007). Comparison of a laboratory and a production coating spray gun with respect to scale-up. AAPS Pharmscitech, 8:3.
   PubMedGoogle Scholar
• Siepmann F, Siepmann J, Walther M, MacRae R, Bodmeier R. (2006). Aqueous HPMCAS coatings: effects of formulation and processing parameters on drug release and mass transport mechanisms. Eur J Pharm Biopharm, 63:262–269.
   PubMed Web of Science ®Google Scholar
• Siepmann F, Siepmann J, Walther M, MacRae RJ, Bodmeier R. (2008). Polymer blends for controlled release coatings. J Control Release, 125:1–15.
   PubMed Web of Science ®Google Scholar
• Muschert S, Siepmann F, Leclercq B, Carlin B, Siepmann J. (2010). Simulated food effects on drug release from ethylcellulose: PVA-PEG graft copolymer-coated pellets. Drug Dev Ind Pharm, 36:173–179.
   PubMed Web of Science ®Google Scholar
• Dow Chemical Company. (2002). Technical Literature: METHOCEL™ Cellulose Ethers.
   Google Scholar
• American Society of Testing Materials (ASTM). (2002). ASTM D882-02: Standard Test Method for Properties of Thin Plastic Sheeting.
   Google Scholar
• American Society for Testing Materials (ASTM). (2005). ASTM E96/E 96 M-05: Standard Test Methods for Water Vapor Transmission of Materials.
   Google Scholar
• Bley O, Siepmann J, Bodmeier R. (2009). Characterization of moisture-protective polymer coatings using differential scanning calorimetry and dynamic vapor sorption. J Pharm Sci, 98:651–664.
   PubMed Web of Science ®Google Scholar
• Cunningham C. (2007). Reducing coated tablet defects from laboratory through production scale: performance of hypromellose or polyvinyl alcohol-based aqueous film coating systems. AAPS Annual Meeting, San Diego, CA.
   Google Scholar
• Rogers T, Sheskey P, Furukawa H, Mallon C, Trampe M, Holbrook D. (2008). Investigation of a novel hypromellose polymer for high-productivity tablet coating applications. AAPS Annual Meeting, Atlanta, GA.
   Google Scholar
• Porter S. (2010). The role of high-solids coating systems in reducing process costs. Tablets Capsules, 8:10–16.
   Google Scholar
• Cunningham C, Hansell J, Nuneviller F 3rd, Rajabi-Siahboomi AR. (2010). Evaluation of recent advances in continuous film coating processes. Drug Dev Ind Pharm, 36:227–233.
   PubMed Web of Science ®Google Scholar
• Hancock B, York P, Rowe R. (1997). The use of solubility parameters in pharmaceutical dosage form design. Int J Pharm, 148:1–21.
   Web of Science ®Google Scholar
• Guo J-H. (1993). Effects of plasticizers on water permeation and mechanical properties of cellulose acetate: antiplasticization in slightly plasticized polymer film. Drug Dev Ind Pharm, 19:1541–1555.
   Web of Science ®Google Scholar
• Guo J-H. (1994). An investigation into the formation of plasticizer channels in plasticized polymer films. Drug Dev Ind Pharm, 20:1883–1893.
   Web of Science ®Google Scholar
• Hsu ER, Gebert MS, Becker NT, Gaertner AL. (2001). The effects of plasticizers and titanium dioxide on the properties of poly(vinyl alcohol) coatings. Pharm Dev Technol, 6:277–284.
   PubMed Web of Science ®Google Scholar
• Yuan J, Shang P, Wu S. (2001). Effects of polyethylene glycol on morphology, thermomechanical properties, and water vapor permeability of cellulose acetate-free films. Pharm Tech, 62–74.
   Google Scholar
• Aulton M, Abdul-Razzak, M, Hogan J. (1981). The mechanical properties of hydroxypropylmethylcellulose films derived from aqueous systems part I: the influence of plasticizers. Drug Dev Ind Pharm, 7:649–668.
   Web of Science ®Google Scholar
• Heinamaki J, Lehtola V, Nikupaavo P, Yliruusi J. (1994). The mechanical and moisture permeability properties of aqueous-based hydroxypropyl methylcellulose coating systems plasticized with polyethylene glycol. Int J Pharm, 112:191–196.
   Web of Science ®Google Scholar
• Honary S, Orafai H. (2002). The effect of different plasticizer molecular weights and concentrations on mechanical and thermomechanical properties of free films. Drug Dev Ind Pharm, 28:711–715.
   PubMed Web of Science ®Google Scholar
• Qussi B, Suess WG. (2006). The influence of different plasticizers and polymers on the mechanical and thermal properties, porosity and drug permeability of free shellac films. Drug Dev Ind Pharm, 32:403–412.
   PubMed Web of Science ®Google Scholar
• Rowe RC, Forse SF. (1980). The effect of polymer molecular weight on the incidence of film cracking and splitting on film coated tablets. j Pharm Pharmacol, 32:583–584.
   PubMed Web of Science ®Google Scholar
• Okutgen E, Hogan J, Aulton M. (1995). Quantitative estimation of internal stress development in aqueous HPMC tablet film coats. Int J Pharm, 119:193–202.
   Web of Science ®Google Scholar
• Rowe RC. (1983). A reappraisal of the equations used to predict the internal stresses in film coatings applied to tablet substrates. J Pharm Pharmacol, 35:112–113.
   PubMed Web of Science ®Google Scholar
• Felton L, McGinity J. (1997). Influence of plasticizers on the adhesive properties of an acrylic resin copolymer to hydrophilic and hydrophobic tablet compacts. Int J Pharm, 154:167–178.
   Web of Science ®Google Scholar