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Research Article

In vivo microdialysis for the evaluation of transfersomes as a novel transdermal delivery vehicle for cinnamic acid

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Pages 301-307 | Received 31 Aug 2012, Accepted 04 Dec 2012, Published online: 25 Jan 2013

References

  • Jain S, Jain P, Umamaheshwari RB, Jain NK. Transfersomes – a novel vesicular carrier for enhanced transdermal delivery: development, characterization, and performance evaluation. Drug Dev Ind Pharm 2003;29:1013–26
  • Cevc G. Self-regulating “smart carriers” for non-invasive and targeted drug delivery. Cell Mol Biol Lett 2002;7:224–5
  • Trommer H, Neubert RH. Overcoming the stratum corneum: the modulation of skin penetration: a review. Skin Pharmacol Physiol 2006;19:106–21
  • Rai K, Gupta Y, Jain A, Jain SK. Transfersomes: self-optimizing carriers for bioactives. PDA J Pharm Sci Technol 2008;62:362–79
  • Alvi IA, Madan J, Kaushik D, et al. Comparative study of transfersomes, liposomes, and niosomes for topical delivery of 5-fluorouracil to skin cancer cells: preparation, characterization, in-vitro release, and cytotoxicity analysis. Anticancer Drugs 2011;22:774–82
  • Geusens B, Strobbe T, Bracke S, et al. Lipid-mediated gene delivery to the skin. Eur J Pharm Sci 2011;43:199–211
  • Vinod KR, Kumar MS, Anbazhagan S, et al. Critical issues related to transfersomes – novel vesicular system. Acta Sci Pol Technol Aliment 2012;11:67–82
  • El Zaafarany GM, Awad GA, Holayel SM, Mortada ND. Role of edge activators and surface charge in developing ultradeformable vesicles with enhanced skin delivery. Int J Pharm 2010;397:164–72
  • Maswadeh H, Demetzos C, Dimas K, et al. Accumulation of vinblastine into transfersomes and liposomes in response to a transmembrane ammonium sulfate gradient and their cytotoxic/cytostatic activity in vitro. Anticancer Res 2001;21:2577–83
  • Simões SI, Delgado TC, Lopes RM, et al. Developments in the rat adjuvant arthritis model and its use in therapeutic evaluation of novel non-invasive treatment by SOD in transfersomes. J Control Release 2005;103:419–34
  • Manda P, Hargett JK, Vaka SR, et al. Delivery of cefotaxime to the brain via intranasal administration. Drug Dev Ind Pharm 2011;37:1306–10
  • Holmgaard R, Nielsen JB, Benfeldt E. Microdialysis sampling for investigations of bioavailability and bioequivalence of topically administered drugs: current state and future perspectives. Skin Pharmacol Physiol 2010;23:225–43
  • Au WL, Skinner MF, Benfeldt E, et al. Application of dermal microdialysis for the determination of bioavailability of clobetasol propionate applied to the skin of human subjects. Skin Pharmacol Physiol 2012;25:17–24
  • Ebah L, Brenchley P, Coupes B, Mitra S. A modified in vivo flow variation technique of microdialysis for sampling uremic toxins in the subcutaneous interstitial compartment. Blood Purif 2011;32:96–103
  • Zhang QL, Hu JH, Jia ZP, et al. Pharmacokinetics of aconitine in rat skin after oral and transdermal gel administrations. Biomed Chromatogr 2012;26:622–6
  • Patel M, Joshi A, Hassanzadeth H, et al. Quantification of dermal and transdermal delivery of meloxicam gels in rabbits. Drug Dev Ind Pharm 2011;37:613–17
  • Jiang B, Zhang ZW. Comparison on phenolic compounds and antioxidant properties of cabernet sauvignon and merlot wines from four wine grape-growing regions in china. Molecules 2012;17:8804–21
  • Huang HC, Jan TR, Yeh SF. Inhibitory effect of curcumin, an anti-inflammatory agent, on vascular smooth muscle cell proliferation. Eur J Pharmacol 1992;221:381–4
  • Liu Z, Zhang X, Wu H, et al. Preparation and evaluation of solid lipid nanoparticles of baicalin for ocular drug delivery system in vitro and in vivo. Drug Dev Ind Pharm 2011;37:475–81
  • Han JZ, Sun J, Zhu QG, et al. A modified LC-MS/MS method for determination of tetramethylpyrazine in microdialysis samples and calibration of home-made linear probes. Biomed Chromatogr 2012;26:1276–81
  • Benson HA. Transfersomes for transdermal drug delivery. Expert Opin Drug Deliv 2006;3:727–37
  • El Maghraby GM, Williams AC, Barry BW. Skin delivery of oestradiol from lipid vesicles: importance of liposome structure. Int J Pharm 2000;204:159–69
  • El Maghraby GM, Barry BW, Williams AC. Liposomes and skin: from drug delivery to model membranes. Eur J Pharm Sci 2008;34:203–22
  • Pierre MB, Dos Santos Miranda Costa I. Liposomal systems as drug delivery vehicles for dermal and transdermal applications. Arch Dermatol Res 2011;303:607–21
  • Cevc G, Blume G. Hydrocortisone and dexamethasone in very deformable drug carriers have increased biological potency, prolonged effect, and reduced therapeutic dosage. Biochim Biophys Acta 2004;1663:61–73
  • Benfeldt E. In vivo microdialysis for the investigation of drug levels in the dermis and the effect of barrier perturbation on cutaneous drug penetration. Studies in hairless rats and human subjects. Acta Derm Venereol Suppl (Stockh) 1999;206:1–59
  • Cevc G, Schätzlein A, Blume G. Transdermal drug carriers: basic properties, optimization and transfer efficiency in the case of epicutaneously applied peptides. J Control Release 1995;36:3–16
  • Duangjit S, Opanasopit P, Rojanarata T, Ngawhirunpat T. Characterization and in vitro skin permeation of meloxicam-loaded liposomes versus transfersomes. J Drug Deliv 2011;2011:Article ID 418316
  • Wei H, Wang S, Xu F, et al. Topical bioequivalence of acyclovir creams using dermal microdialysis in pigs: a new model to evaluate bioequivalence for topical formulations. Drug Dev Ind Pharm 2012;38:785–91
  • Song YK, Hyun SY, Kim HT, et al. Transdermal delivery of low molecular weight heparin loaded in flexible liposomes with bioavailability enhancement: comparison with ethosomes. J Microencapsul 2011;28:151–8
  • Elsayed MM, Abdallah OY, Naggar VF, Khalafallah NM. Deformable liposomes and ethosomes: mechanism of enhanced skin delivery. Int J Pharm 2006;322:60–6

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