160
Views
9
CrossRef citations to date
0
Altmetric
Research Article

Development of a prospective isopropyl alcohol-loaded pharmaceutical base using simultaneous in vitro/in vivo characterization methods of skin performance

, , , , , , , & show all
Pages 960-971 | Received 27 Dec 2012, Accepted 04 Apr 2013, Published online: 20 May 2013

References

  • Lukic M, Jaksic I, Krstonosic V, et al. A combined approach in characterization of an effective w/o hand cream: the influence of emollient on textural, sensorial and in vivo skin performance. Int J Cosmet Sci 2012;34:140–9
  • Piispanen P, Persson M, Claesson P, Norin T. Surface properties of surfactants derived from natural products. Part 1: syntheses and structure/property relationships – solubility and emulsification. J Surfact Deterg 2004;7:147–59
  • Savic S, Tamburic S, Savic M. From conventional towards new – natural surfactants in drug delivery systems design: current status and perspectives. Expert Opin Drug Deliv 2010;7:353–69
  • Iglauer S, Wu Y, Shuler P, et al. Alkyl polyglycoside surfactant-alcohol cosolvent formulations for improved oil recovery. Colloids Surf A Physicochem Eng Asp 2009;339:48–59
  • Moddaresi M, Brown M, Tamburic S, Jones S. Tocopheryl acetate disposition in porcine and human skin when administered using lipid nanocarriers. J Pharm Pharmacol 2010;62:762–9
  • Mugglestone C, Mariz S, Lane M. The development and registration of topical pharmaceuticals. Int J Pharm 2012;435:22–6
  • Russell LM, Guy RH. Measurement and prediction of the rate and extent of drug delivery into and through the skin. Expert Opin Drug Deliv 2009;6:355–69
  • Godin B, Touitou E. Transdermal skin delivery: predictions for humans from in vivo, ex vivo and animal models. Adv Drug Deliv Rev 2007;59:1152–61
  • Narkar Y. Bioequivalence for topical products – an update. Pharm Res 2010;27:2590–601
  • Lademann J, Jacobi U, Surber C, et al. The tape stripping procedure – evaluation of some critical parameters. Eur J Pharm Biopharm 2009;72:317–23
  • Au WL, Skinner M, Kanfer I. Comparison of tape stripping with the human skin blanching assay for the bioequivalence assessment of topical clobetasol propionate formulations. J Pharm Pharmaceut Sci 2010;13:11–20
  • Baudonnet L, Grossiord J-L, Rodriguez F. Physicochemical characterization and in vitro release of salicylic acid from O/W emulsions prepared with Montanov 68: effect of formulation parameters. Drug Dev Ind Pharm 2004;30:975–84
  • Vucinic-Milankovic N, Savic S, Vuleta G, Vucinic S. The physicochemical characterization and in vitro/in vivo evaluation of natural surfactants-based emulsions as vehicles for diclofenac diethylamine. Drug Dev Ind Pharm 2007;33:221–34
  • Jaksic I, Lukic M, Malenovic A, et al. Compounding of a topical drug with prospective natural surfactant-stabilized pharmaceutical bases: physicochemical and in vitro/in vivo characterization – a ketoprofen case study. Eur J Pharm Biopharm 2012;80:164–75
  • Surber C, Tassopoulos T, Smith EW. Ointments, creams and lotions used as topical drug delivery vehicles. In: Bronaugh R, Maibach H, eds. Topical absorption of dermatological products. New York: Marcel Dekker, 2001:511–17
  • Deutsches Arzneibuch. Stuttgart: Deutscher Apotheker Verlag; 2006
  • Savic S, Vuleta G, Daniels R, Müller-Goymann C. Colloidal microstructure of binary systems and model creams stabilized an alkylpolyglucoside non-ionic emulsifier. Colloid Polym Sci 2005;283:439–51
  • Dragicevic-Curic N, Winter S, Stupar M, et al. Temoporfin-loaded liposomal gels: viscoelastic properties and in vitro skin penetration. Int J Pharm 2009;373:77–84
  • Winkler A, Müller-Goymann C. Comparative permeation studies for δ-aminolevulinic acid and its n-butyl ester through stratum corneum and artificial skin constructs. Eur J Pharm Biopharm 2002;53:281–7
  • Michel C, Purmann T, Mentrup E, et al. Effect of liposomes on percutaneous penetration of lipophilic materials. Int J Pharm 1992;84:93–105
  • Hathout RM, Mansour S, Geneidi AS, Mortada ND. Visualization, dermatopharmacokinetic analysis and monitoring the conformational effects of a microemulsion formulation in the skin stratum corneum. J Colloid Interf Sci 2011;354:124–30
  • Fullerton A, Fischer T, Lahti A, et al. Guidelines for measurement of skin colour and erythema. A report from the Standardization Group of the European Society of Contact Dermatitis. Contact Dermatitis 1996;35:1–10
  • Berardesca E. EEMCO guidance for the assessment of stratum corneum hydration: electrical methods. Skin Res Technol 1997;3:126–32
  • Rogiers V. EEMCO guidance for the assessment of transepidermal water loss in cosmetic sciences. Skin Pharmacol Appl Skin Physiol 2001;14:117–28
  • Hoffmann B, Platz G. Phase and aggregation behaviour of alkylglycosides. Curr Opin Colloid Interface Sci 2001;6:171–7
  • Junginger HE. Pharmaceutical emulsions and creams. In: Sjöblom J, ed. Emulsions – a fundamental and practical approach. Netherlands: Kluwer Academic Publishers; 1992:189–205
  • British Pharmacopoeia. London: British Pharmacopoeial Commission, Stationary Office; 2009
  • Barnes HA. Rheology of emulsions – a review. Colloids Surf A 1994;91:89–95
  • Tadros T. Application of rheology for assessment and prediction of the long-term physical stability of emulsions. Adv Colloid Interface Sci 2004;108–109:227–58
  • Hadgraft J. Passive enhancement strategies in topical and transdermal drug delivery. Int J Pharm 1999;184:1–6
  • Tamburic S, Craig DQM, Vuleta G, Milic J. A comparison of electrical and rheological techniques for the characterization of creams. Int J Pharm 1996;137:243–8
  • Csóka I, Csányi E, Zapantis G, et al. In vitro and in vivo percutaneous absorption of topical dosage forms: case studies. Int J Pharm 2005;291:11–19
  • Schaefer UF, Hansen S, Schneider M, et al. Models for skin absorption and skin toxicity testing. In: Ehrhardt C, Kim KJ, eds. Drug absorption studies. In situ, in vitro and in silico models. New York: Springer; 2008:3–33
  • Oliveira G, Beezer A, Hadgraft J, Lane M. Alcohol enhanced permeation in model membranes. Part I. Thermodynamic and kinetic analyses of membrane permeation. Int J Pharm 2010;393:61–7
  • Saino V, Monti D, Burgalassi S, et al. Optimization of skin permeation and distribution of ibuprofen by using nanostructures (coagels) based on alkyl vitamin C derivatives. Eur J Pharm Biopharm 2010;76:443–9
  • Darlenski R, Sassning S, Tsankov N, Fluhr JW. Non-invasive in vivo methods for investigation of the skin barrier physical properties. Eur J Pharm Biopharm 2009;72:295–303
  • Arellano A, Santoyo S, Martin C, Ygartua P. Influence of propylene glycol and isopropyl myristate on the in vitro percutaneous penetration of diclofenac sodium from carbopol gels. Eur J Pharm Sci 1998;7:129–35
  • Harada S, Horisawa E, Kano S, Sugibayashi K. Formulation study of topically applied o/w lotion containing vitamin D3 derivative, focusing on skin permeability of the drug. Drug Dev Ind Pharm 2011;37:917–25
  • Levintova Y, Plakogiannis F, Bellantone R. An improved in vitro method for measuring skin permeability that controls excess hydration of skin using modified Franz diffusion cells. Int J Pharm 2011;419:96–106
  • Lau WM, White AW, Heard CM. Topical delivery of a naproxen-dithranol co-drug: in vitro skin penetration, permeation, and staining. Pharm Res 2010;27:2734–42
  • Dias M, Hadgraft J, Lane M. Influence of membrane–solvent–solute interactions on solute permeation in model membranes. Int J Pharm 2007;336:108–14
  • Herkenne C, Naik A, Kalia Y, et al. Effect of propylene glycol on ibuprofen absorption into human skin in vivo. J Pharm Sci 2008;97:185–97
  • Russell LM, Wiedersberg S, Delgado-Charro MB. The determination of stratum corneum thickness: an alternative approach. Eur J Pharm Biopharm 2008;69:861–70
  • Yariv D, Efrat R, Libster D, et al. In vitro permeation of diclofenac salts from lyotropic liquid crystalline systems. Colloids Surf B: Biointerfaces 2010;78:185–92

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.