Taste-masked and affordable donepezil hydrochloride orally disintegrating tablet as promising solution for non-compliance in Alzheimer’s disease patients

References

• Sunada H, Bi YX. Preparation, evaluation and optimization of rapidly disintegrating tablets. Powder Technol 2002;122:188–98
   Web of Science ®Google Scholar
• US Food and Drug Administration, CDER Data Standards Manual. Guidance for industry: orally disintegrating tablet. 2008 December. FDA. 2011 Nov 29. Available from: http://www.fda.gov/cder/dsm/DRG/drg00201.htm
   Google Scholar
• British Pharmacopoeia. Vol. 3 – General Monograph: Tablets; 2009:5
   Google Scholar
• Hirani JJ, Rathod DA, Vadalia KR. Orally disintegrating tablets: a review. Trop J Pharm Res 2009;8:161–72
   Web of Science ®Google Scholar
• Pillai R, Karatgi P. Orally disintegrating tablets: the path to improved patient compliance and enhanced life cycle management. Pharmtech Europe 2009;21:37–41
   Google Scholar
• Camarco W, Ray D, Druffner A. Selecting superdisintegrants for orally disintegrating formulations. PT. 2011. Available from: http://pharmtech.findpharma.com/pharmtech/Manufacturing/Selecting-Superdisintegrants-for-Orally-Disintegra/ArticleStandard/Article/detail/378398 [last accessed 2 Feb 2014]
   Google Scholar
• Makino T, Yamada M, Kikuta J. Fast dissolving tablet and its production. European Patent. 0553777 A2; 1993
   Google Scholar
• Dobetti L. Fast melting tablets: development and technologies. Pharm Tech 2001;(Suppl):44–50
   Google Scholar
• Deepak K, Harish D, Saini TR. Mouth dissolving tablets: a review. Indian Drugs 2004;41:187–93
   Google Scholar
• Gohel M, Patel M, Amin A, et al. Formulation design and optimization of mouth dissolve tablets of nimesulide using vacuum drying technique. AAPS PharmSciTech 2004;5:10–15
   Web of Science ®Google Scholar
• Abdelbary G, Prinderre P, Eouani C, et al. The preparation of orally disintegrating tablets using a hydrophilic waxy binder. Int J Pharma 2004;278:423–33
   PubMed Web of Science ®Google Scholar
• Kuno Y, Kojima M, Ando S, Nakagami H. Evaluation of rapidly disintegrating tablets manufactured by phase transition of sugar alcohols. J Control Release 2005;105:16–22
   PubMed Web of Science ®Google Scholar
• Maniruzzaman M, Boateng JS, Chowdhry BZ, et al. A review on the taste masking of bitter APIs: hot-melt extrusion (HME) evaluation. Drug Dev Ind Pharm 2014;40:145–56
   Google Scholar
• Yan YD, Jong SW, Kang JH, et al. Preparation and evaluation of taste-masked donepezil hydrochloride orally disintegrating tablets. Biol Pharm Bull 2010;33:1364–70
   PubMed Web of Science ®Google Scholar
• Joseph TD, Robert LT, Gary CY, et al. Pharmacotherapy: a pathophysiologic approach. 6th ed. New York: McGraw Hill; 2005
   Google Scholar
• Martin RF. Effective pharmacologic management of Alzheimer disease. AMJMED 2007;120:388–97
   Web of Science ®Google Scholar
• United State Pharmacopoeia 29-NF 24, Pg. 3017
   Google Scholar
• Carr RL. Evaluating flow properties of solids. Chem Eng 1965;72:163–8
   Google Scholar
• Rowe RC, Sheskey PJ, Quinn ME. Pharmaceutical excipients. 6th ed. London: Pharmaceutical Press; 2009
   Google Scholar
• Sherwood BE, Staniforth JH, Hunter EA. Pharmaceutical excipient having improved compressibility. US Patent 6,521,261, 2003
   Google Scholar
• Du J, Hoag S. The influence of excipients on the stability of the moisture sensitive drugs asprin and niacinamide: comparison of tablets containing lactosemonohydrate with tablets containing anhydrous lactose. Pharm Dev Technol 2001;6:159–66
   PubMed Web of Science ®Google Scholar
• Shayne CG, eds. Preclinical development handbook: ADME and biopharmaceutical properties. New York: John Wiley and Sons Inc.; 2008
   Google Scholar
• Hauschild K, Picker KM. Evaluation of a new coprocessed compound based on lactose and maize starch for tablet formulation. AAPS PharmSci 2004;6:16
   PubMedGoogle Scholar
• Klevan I, Nordström J, Tho I, Alderborn G. A statistical approach to evaluate the potential use of compression parameters for classification of pharmaceutical powder materials. Eur J Pharm Biopharm 2010;75:425–35
   PubMed Web of Science ®Google Scholar
• Kornblum SS, Stoopak SB. A new tablet disintegrating agent: cross-linked polyvinylpyrolidone. J Pharm Sci 1973;62:43–8
   PubMed Web of Science ®Google Scholar
• Gohel MC, Jogani PD. A review of co-processed directly compressible excipients. J Pharm Pharma Sci 2005;8:76–93
   PubMed Web of Science ®Google Scholar
• Pathak N, Kumar A, Methkar V, et al. Formulation and optimization of immediate release tablet of an antialchoholic drug by dry granulation method. Pharmacie Globale IJCP 2011;3:8
   Google Scholar
• Sadeghi F, Mosaffa F, Garekani HA. Effect of particle size, compaction force and presence of aerosil 200 on the properties of matrices prepared from physical mixture of propranolol hydrochloride and eudragit RS or RL. IJBMS 2007;10:197–205
   Google Scholar
• Lachman L, Lieberman H, Kanig J, eds. The theory and practice of industrial pharmacy. 3rd ed. Mumbai: Varghese Publication House; 2009
   Google Scholar
• Abdullah M, Ahmed AM, Al-Jenoobi FI, et al. Formulation and evaluation of dried yeast tablets using different techniques. Eur J Pharm Biopharm 2007;67:253–9
   PubMed Web of Science ®Google Scholar
• Oyi AR, Allagh TS, Olayemi OJ. Comparative binding effects of wheat, rice and maize starches in chloroquine phosphate tablet formulations. RJASET 2009;1:77–80
   Google Scholar
• Quadir A, Kolter K. A comparative study of current superdisintegrants. PT. 2011. Available from: http://pharmtech.findpharma.com/pharmtech/article/articleDetail.jsp?id=378399&sk=&date=&pageID=2 [last accessed 10 Oct 2013].
   Google Scholar
• Park TJ, Ko DH, Kim YJ, Kim YGL. Polymorphic characterization of pharmaceutical solids, donepezil hydrochloride, by C CP/MAS solid-state nuclear magnetic resonance spectroscopy. B Kor Chem Soc 2009;30:2007–10
   Web of Science ®Google Scholar
• Krishna R, Moses JB, Anil K, et al. Identification and characterization of potential impurities of donepezil. J Pharma Biomed 2004;35:1047–58
   PubMed Web of Science ®Google Scholar
• Duke JA. CRC handbook of medicinal herbs. Boca Raton (FL): CRC Press Inc.; 1985
   Google Scholar
• Opinion of the scientific committee on food on glycyrrhizinic acid and its ammonium salt. European commission. Health and Consumer Protection Directorate – General. SCF/CS/ADD/EDUL/225 Final 10 April 2003
   Google Scholar
• Brown D. Orally disintegrating tablet: taste over speed. Drug Develop Deliv 2003;3:58–61
   Google Scholar
• Tan QY, Zhang L, Liu GD, et al. Novel taste-masked orally disintegrating tablets for a highly soluble drug with an extremely bitter taste: design rationale and evaluation. Drug Dev Ind Pharm 2013;39:1364–71
   PubMed Web of Science ®Google Scholar
• Bayarri S, Izquierdo L, Costell E. Sweetening power of aspartame in hydrocolloids gels: influence of texture. Food Hydrocolloids 2007;21:1265–74
   Web of Science ®Google Scholar
• Jim S, Lily HS. Food additives data book. Malden: Blackwell Publishing; 2003
   Google Scholar