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Research Article

Film-coated matrix mini-tablets for the extended release of a water-soluble drug

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Pages 623-630 | Received 17 Sep 2013, Accepted 24 Jan 2014, Published online: 24 Feb 2014

References

  • Kirsch JD, Drennen JK. Determination of film-coated tablet parameters by near-infrared spectroscopy. J Pharmaceut Biomed Anal 1995;13:1273–81
  • Hemati M, Cherif R, Saleh K, Pont V. Fluidized bed coating and granulation: influence of process-related variables and physicochemical properties on the growth kinetics. Powder Technol 2003;130:18–34
  • Behzadi SS, Toegel S, Viernstein H. Innovations in coating technology. Recent Patents Drug Deliv Formul 2008;2:209–30
  • Patel JK, Shah AM, Sheth NR. Aqueous-based film coating of tablets: study the effect of critical process parameters. Int J PharmTech Res 2009;2:235–40
  • Cahyadi C, Heng PWS, Chan LW. Optimization of process parameters for a quasi-continuous tablet coating. J Am Assoc Pharm Sci 2010;12:119–31
  • Rege BD, Gawel J, Kou JH. Identification of critical process variables for coating actives onto tablets via statistically designed experiments. Int J Pharm 2002;237:87–94
  • Tang L, Schwartz JB, Porter SC, et al. Drug release from film-coated chlorpheniramine maleate nonpareil beads: effect of water-soluble polymer, coating level, and soluble core material. Pharm Dev Technol 2000;5:383–90
  • Tobiska S, Kleinebudde P. Coating uniformity and coating efficiency in a Bohle lab-coater using oval tablets. Eur J Pharm Biopharm 2003;56:3–9
  • Smith GW, Macleod GS, Fell JT. Mixing efficiency in side-vented coating equipment. Am Assoc Pharm Sci 2003;4:71–5
  • Sadeghi F, Ford JL, Rajabi-Siahboomi A. The influence of drug type on the release profiles from Surelease-coated pellets. Int J Pharm 2003;254:123–35
  • Ahmed A, Souad S. Effect of viscosity grades of ethylcellulose on the sustained release properties of indomethacin from its matrix tablets. Afr J Pharm Pharmacol 2008;2:153–6
  • Murtaza G. Ethylcellulose microparticles: a review. Acta Poloniae Pharmaceut 2012;69:11–22
  • Cavalcanti OA, Petenuc B, Bedin AC, et al. Characterisation of ethylcellulose films containing natural polysaccharides by thermal analysis and FTIR spectroscopy. Acta Farm Bonaerense 2003;23:53–7
  • Rohera BD, Parikh NH. Influence of type and level of water soluble additives on drug release and surface and mechanical properties of Surelease® films. Pharm Dev Technol 2002;7:421–32
  • Sadeghi F, Ford JL, Rubinstein MH, Rajabi-Siahboomi AR. Study of drug release from pellets coated with Surelease containing hydroxypropylmethylcellulose. Drug Dev Ind Pharm 2001;27:419–30
  • Emeje MO, Kunle OO, Ofoefule SI. Compaction characteristics of ethylcellulose in the presence of some channeling agents: Technical Note. J Am Assoc Pharm Sci 2006;7:1–4
  • Sahni E, Chaudhuri B. Experiments and numerical modeling to estimate the coating variability in a pan coater. Int J Pharm 2011;418:286–96
  • Li CL, Martini LG, Ford JL, Roberts M. The use of hypromellose in oral drug delivery. J Pharm Pharmacol 2005;57:533–46
  • World Health Organization. Development of paediatric medicines – Points to consider in pharmaceutical development; 2012
  • Ishida M, Abe K, Hashizume M, Kawamura M. A novel approach to sustained pseudoephedrine release: differentially coated mini-tablets in HPMC capsules. Int J Pharm 2008;359:46–52
  • Lingam M, Ashok T, Venkateswarlu V, Rao YM. Design and evaluation of a novel matrix type multiple units as biphasic gastroretentive drug delivery systems. AAPS PharmSciTech 2008;9:1253–61
  • Dierickx L, Saerens L, Almeida A, et al. Co-extrusion as manufacturing technique for fixed-dose combination mini-matrices. Eur J Pharm Biopharm 2012;81:683–9
  • Munday DL. A comparison of the dissolution characteristics of theophylline from film-coated granules and mini-tablets. Drug Dev Ind Pharm 1994;20:2369–79
  • Mohamed F, Roberts M, Ford JL, et al. The influence of HPMC concentration on release of theophylline or hydrocortisone from extended-release mini-tablets. Drug Dev Ind Pharm 2013;39:1167–74
  • Mohamed FAA, Roberts M, Seton L, et al. Production of extended release mini-tablets using directly compressible grades of HPMC. Drug Dev Ind Pharm 2013;39:1690–7
  • Cantor SL, Hoag SW, Augsburger LL. Formulation and characterization of a compacted multiparticulate system for modified release of water-soluble drugs – Part II theophylline and cimetidine. Drug Dev Ind Pharm 2009;35:568–82
  • Roberts M, Vellucci D, Mostafa S, et al. Development and evaluation of sustained release Compritol® 888 ATO matrix mini-tablets. Drug Dev Ind Pharm 2012;38:1068–76
  • Munday DL, Fassihi AR. Controlled release delivery: effect of coating composition on release characteristics of mini-tablets. Int J Pharm 1989;52:109–14
  • Frohoff-Hülsmann MA, Lippold BC, McGinity JW. Aqueous ethyl cellulose dispersion containing plasticizers of different water solubility and hydroxypropyl methyl-cellulose as coating material for diffusion pellets II: properties of sprayed films. Eur J Pharm Biopharm 1999;48:67–75
  • Gunder W, Lippold BH, Lippold BC. Release of drugs from ethyl cellulose microcapsules (diffusion pellets) with pore formers and pore fusion. Eur J Pharm Sci 1995;3:203–14
  • Ozturk AG, Ozturk SS, Palsson BO, et al. Mechanism of release from pellets coated with an ethylcellulose-based film. J Control Rel 1990;14:203–13
  • Kim M, Jun SW, Lee S, et al. The influence of Surelease and sodium alginate on the in-vitro release of tamsulosin hydrochloride in pellet dosage form. J Pharm Pharmacol 2005;57:735–42
  • Kim M, Kim J, Kang S, et al. Influence of water soluble additives and HPMCP on drug release from Surelease-coated pellets containing tamsulosin hydrochloride. Arch Pharm Res 2007;30:1008–13
  • Sadeghi F, Ford JL, Rubinstein MH, Rajabi-Siahboomi AR. Comparative study of drug release from pellets coated with HPMC or Surelease. Drug Dev Ind Pharm 2000;26:651–60
  • Wilson KE, Crossman E. The influence of tablet shape and pan speed on intra-tablet film coating uniformity. Drug Dev Ind Pharm 1997;23:1239–43
  • Siepmann J, Podual K, Sriwongjanya M, et al. A new model describing the swelling and drug release kinetics from hydroxypropyl methylcellulose tablets. J Pharm Sci 1999;88:65–72
  • Gao P, Skoug JW, Nixon PR, et al. Swelling of hydroxypropyl methylcellulose matrix tablets. 2. Mechanistic study of the influence of formulation variables on matrix performance and drug release. J Pharm Sci 1996;85:732–40
  • Enayatifard R, Saeedi M, Akbari J, et al. Effect of hydroxypropyl methylcellulose and ethyl cellulose content on release profile and kinetics of diltiazem HCl from matrices. Trop J Pharm Res 2009;8:425–32
  • Krenzlin S, Siepmann F, Wils D, et al. Non-coated multiparticulate matrix systems for colon targeting. Drug Dev Ind Pharm 2011;37:1150–9
  • Cahyadi C, Chan LW, Colombo P, Heng PWS. The butterfly effect: a physical phenomenon of hypromellose matrices during dissolution and the factors affecting its occurrence. Int J Pharm 2011;406:31–40

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