156
Views
9
CrossRef citations to date
0
Altmetric
Research Article

The dissolution and solid-state behaviours of coground ibuprofen–glucosamine HCl

, , , &
Pages 1682-1692 | Received 30 Jul 2014, Accepted 17 Nov 2014, Published online: 11 Dec 2014

References

  • Otsuka M, Kaneniwa N. Effects of grinding on the physicochemical properties of cephalexin. Chem Pharm Bull 1984;32:1071–9
  • Ford JL. The current status of solid dispersions. Pharm Acta Helv 1986;61:69–88
  • Takeuchi H, Handa T, Kawashima Y. Enhancement of the dissolution rate of a poorly watersoluble drug (tolbutamide) by a spray-drying solvent deposition method and disintegrants. J Pharm Pharmacol 1987;39:769–73
  • Nyström C, Westerberg M. The use of ordered mixtures for improving the dissolution rate of low solubility compounds. J Pharm Pharmacol 1986;38:161–5
  • Nozawa Y, Suzuki K, Miyagishima A, Hirota S. Solid-phase complexing of ibuprofen to β-cyclodextrin by roll mixing. Powder Tech 1994;79:269–71
  • Moyano JR, Gines JM, Arias MJ, Rabasco AM. Study of the dissolution characteristics of oxazepam via complexation with beta-cyclodextrin. Int J Pharm 1995;114:95–102
  • Buckton G, Beezer AE. The relationship between particle-size and solubility. Int J Pharm 1991;82:R7–10
  • Martini A, Torricelli C, Deponti R. Physico-pharmaceutical characteristics of steroid cross-linked polyvinylpyrrolidone coground systems. Int J Pharm 1991;75:141–6
  • Yamaguchi G, Sakamoto K. Effect of dry grinding on gibbsite B. Chem Soc Jpn 1959;32:1364–8
  • Mochalin VN, Sagar A, Gour S, Gogotsi Y. Manufacturing nanosized fenofibrate by salt assisted milling. Pharm Res 2009;26:1365–70
  • Kubo M, Oumi Y, Miura R, et al. Atomic control of layer-by-layer epitaxial growth on SrTiO3(001): molecular-dynamics simulations. Phys Rev B 1997;56:13535–42
  • Liversidge G, Cundy K. Particle size reduction for improvement of oral bioavailability of hydrophobic drugs: I absolute oral bioavailability of nanocrystalline danazol in beagle dogs. Int J Pharm 1995;125:91–7
  • Sugimoto M, Okagaki T, Narisawa S, et al. Improvement of dissolution characteristics and bioavailability of poorly water-soluble drugs by novel cogrinding method using water-soluble polymer. Int J Pharm 1998;160:11–19
  • Yamada H, Takahashi S, Fujita H, et al. Cytokine-induced neutrophil chemoattractants in healing of gastric ulcers in rat – expression of > 40-kDa chemo-attractant in delayed ulcer healing by indomethacin. Dig Dis Sci 1999;44:889–95
  • Sarkari M, Brown J, Chen XX, et al. Enhanced drug dissolution using evaporative precipitation into aqueous solution. Int J Pharm 2002;243:17–31
  • Moneghini M, Kikic I, Voinovich D, et al. Processing of carbamazepine PEG 4000 solid dispersions with supercritical carbon dioxide: preparation, characterisation, and in vitro dissolution. Int J Pharm 2001;222:129–38
  • Camarada CC, Dowless G. Glucosamine sulfate for osteoarthritis. Ann Pharmaco Ther 1998;832:580–7
  • Pujalte JM, Llavore EP, Ylescupidez FR. Double-blind clinical evaluation of oral glucosamine sulfate in the basic treatment of osteoarthrosis. Curr Med Res Opin 1980;7:110–14
  • Horton D. Monosaccharide amino sugars. In: Jeanloz RW, ed. The amino sugars, the chemistry and biology of compounds containing amino sugars, Vol IA. Academic Press Inc: 1969:4–18
  • Clegg DO, Jackson CG. Glucosamine. In: Coates PM, ed. Encyclopedia of dietary supplements. USA: Marcel Dekker; 2005:79–87
  • Al-Hamidi H, Mohammad Amin M, Edwards AA, Nokhodchi A. To enhance dissolution rate of poorly water soluble drugs: glucosamine hydrochloride as a potential carrier in solid dispersion formulations. Colloids Surf B-Biointerfaces 2010;76:170–8
  • Al-Hamidi H, Edwards AA, Douroumis D, et al. Effect of glucosamine HCl on dissolution and solid state behaviours of piroxicam upon milling. Colloids Surf B Biointerfaces 2013;103:189–99
  • Khan KA. Concept of dissolution efficiency. J Pharm Pharmacol 1975;27:48–9
  • Shaw LR, Irwin WJ, Grattan TJ, Conway BR. The effect of selected water-soluble excipients on the dissolution of paracetamol and Ibuprofen. Drug Dev Ind Pharm 2005;31:515–25
  • Pendleton A, Arden N, Dougados M, et al. EULAR recommendations for the management of knee osteoarthritis: report of a task force of the standing committee for International Clinical Studies Including Therapeutic Trials (ESCISIT). Ann Rheum Dis 2000;59:936–44
  • Atkinson RM, Bedford C, Child KJ, Tomich EG. Effect of particle size on blood griseofulvin-levels in man. Nature 1962;193:588–9
  • Liversidge GG, Conzentino P. Drug particle size reduction for decreasing gastric irritancy and enhancing absorption of naproxen in rats. Int J Pharm 1995;125:309–13
  • Barzegar-Jalali M, Valizadeh H, Dastmalchi S, et al. Enhancing dissolution rate of carbamazepine via cogrinding with Crospovidone and hydroxypropylmethylcellulose. Iran J Pharm Res 2007;6:159–65
  • Barzegar-Jalali M, Valizadeh H, Siahi-Shadbad MR, et al. Cogrinding as an approach to enhance dissolution rate of a poorly water soluble drug (gliclazide). Powder Tech 2010;197:150–8
  • Yonemochi E, Kitahara S, Maeda S, et al. Physicochemical properties of amorphous clarithromycin obtained by grinding and spray drying. Eur J Pharm Sci 1999;7:331–8

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.