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Research Article

Effect of permeation enhancers on the iontophoretic transport of metoprolol tartrate and the drug retention in skin

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Pages 19-25 | Received 14 Feb 2010, Accepted 14 Jul 2010, Published online: 21 Aug 2010

References

  • Aqil, M., Sultana, Y., Ali, A. (2006). Transdermal delivery of beta-blockers. Expert Opin Drug Deliv. 3:405–18.
  • Anroop, B., Ghosh, B., Parcha, V., Khanam, J. (2008). Comparative skin permeability of metoprolol tartrate and its ester prodrugs by passive permeation and iontophoresis. Asian J Pharm Sci. 3:1–11.
  • Banga, A.K., Chien, Y.W. (1993). Characterization of in vitro transdermal iontophoretic delivery of insulin. Drug Dev Ind Pharm. 19:2069–87.
  • Borras-Bolasco, J., Diez-Sales, O., Lopez, A., Herraez-Dominguez, M. (2004). A mathematical approach to predicting the percutaneous absorption enhancing effect of sodium lauryl sulphate. Int J Pharm. 269:121–9.
  • Chesnoy, S., Durand, D., Doucet, J., Couarraze, G. (1999). Structural parameters involved in the permeation of propranolol HCl by iontophoresis and enhancers. J Contr Rel. 58:163–75.
  • Choi, E.H., Lee, S.H., Ahn, S.K., Hwang, S.M. (1999). The pretreatment effect of chemical skin penetration enhancers in transdermal drug delivery using iontophoresis. Skin Pharmacol Appl Skin Physiol. 12:326–35.
  • Choi, M.J., Maibach, H.I. (2005). Liposomes and niosomes as topical drug delivery systems. Skin Pharmacol Physiol. 18:209–19.
  • Cosco, D., Celia, C., Cilurzo, F., Trapasso, E., Paolino, D. (2008). Colloidal carriers for the enhanced delivery through the skin. Expert Opin Drug Deliv. 5:737–55.
  • de Figueiredo Alves, S.T., Gomes, M.A.S., Clapauch, R. (2000). Comparison of gel and patch estradiol replacement in Brazil, a tropical country. Maturitas. 36:69–74.
  • Doliwa, A., Santoyo, S., Ygartua, P. (2001). Transdermal iontophoresis and skin retention of piroxicam from gels containing piroxicam: hydroxypropyl-beta-cyclodextrin complexes. Drug Dev Ind Pharm. 27:751–8.
  • Fang, J., Huang, Y., Wu, P., Tsai, Y. (1996). Transdermal iontophoresis of sodium nonivamide acetate II: optimization and evaluation on solutions and gels. Int J Pharm. 145:175–86.
  • Fang, J., Kuo, C., Huang, Y., Wu, P., Tsai, Y. (1999). Transdermal delivery of sodium nonivamide acetate from volatile vehicles: effects of polymers. Int J Pharm. 176:157–67.
  • Femenia-Font, A., Balaguer-Fernandez, C., Merino, V., Rodilla, V., Lopez-Castellano, A. (2005). Effect of chemical enhancers on the in vitro percutaneous absorption of sumatriptan succinate. Eur J Pharm Biopharm. 61:50–5.
  • Ghosh, B., Jain, A., Ashok, P., Patel, B., Tarafdar, K. (2009). Passive and iontophoretic permeation of glipizide gel: an in vitro and in vivo study. Curr Drug Deliv. 6:444–50.
  • Ghosh, T.K., Adimola, J.A., Pfister, W.R., Yum, S.I. (1997). Transdermal delivery of beta adrenergic therapeutics. In: Ghosh, T.K., Pfister, W.R., Yum, S.I., eds. Transdermal and topical drug delivery systems. Illinois: Interpharm Press Inc, 299–320.
  • Green, P.G., Hadgraft, J., Ridout, G. (1989). Enhanced in vitro skin permeation of cationic drugs. Pharm Res. 6:628–32.
  • Hadgraft, J. (1999). Passive enhancement strategies in topical and transdermal drug delivery. Int J Pharm. 184:1–6.
  • Jamakandi, V.G., Ghosh, B., Desai, B.G., Khanam, J. (2006). Recent trends in transdermal cardiovascular therapy. Indian J Pharm Sci. 68:556–61.
  • Kaliszan, R., Nasal, A., Turowski, M. (1995). Binding site for basic drugs on α1- acid glycoprotein as revealed by chemometric analysis of biochromatographic data. Biomed Chrom. 9:211–5.
  • Merclin, N., Bramer, T., Desmán, K. (2004). Iontophoretic delivery of 5-aminolevulinic acid and its methyl ester using a carbopol gel as vehicle. J Contr Rel. 98:57–65.
  • Mitragotri, S. (2000). Synergistic effect of enhancers for transdermal drug delivery. Pharm Res. 17:1354–9.
  • Mutalik, S., Parekh, H.S., Davies, N.M., Udupa, N. (2009). A combined approach of chemical enhancers and sonophoresis for the transdermal delivery of tizanidine hydrochloride. Drug Deliv. 16:82–91.
  • Nair, V., Panchagnula, R. (2003). Poloxamer gel as vehicle for transdermal iontophoretic delivery of arginine vasopressin: evaluation of in vivo performance in rats. Pharmacol Res. 47:555–62.
  • Pillai, O., Panchagnula, R. (2003). Transdermal delivery of insulin from poloxamer gel: ex vivo and in vivo skin permeation studies in rat using iontophoresis and chemical enhancers. J Contr Rel. 89:127–40.
  • Prakash, A., Markham, A. (2000). Metoprolol: a review of its use in chronic heart failure. Drugs. 60:647–78.
  • Sachdeva, V., Siddoju, S., Yu, Y.Y., Kim, H.D., Friden, P.M., Banga, A.K. (2010). Transdermal iontophoretic delivery of terbinafine hydrochloride: quantitation of drug levels in stratum corneum and underlying skin. Int J Pharm. 388:24–31.
  • Shokri, J., Nokhodchi, A., Dashbolaghi, A., Zadeh, D.H., Jalali, M.B. (2001). The effect of surfactants on the skin penetration of diazepam. Int J Pharm. 228:99–107.
  • Wang, Y., Thakur, R., Fan, Q., Michnaik, B. (2005). Transdermal iontophoresis: combination strategies to improve transdermal iontophoretic drug delivery. Eur J Pharm Biopharm. 60:179–91.

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