2,186
Views
29
CrossRef citations to date
0
Altmetric
Research Article

Optimized permeation enhancer for topical delivery of 5-fluorouracil-loaded elastic liposome using Design Expert: part II

, , &
Pages 1242-1253 | Received 08 Oct 2015, Accepted 22 Nov 2015, Published online: 24 Dec 2015

References

  • Bhatt PP, Rytting JH, Topp EM. (1991). Influence of Azone® and lauryl alcohol on the transport of acetaminophen and ibuprofen through shed snake skin. Int J Pharm 72:219–26
  • Contreras MD, Sanchez R. (2002). Application of a factorial design to the study of the flow behavior, spreadability and transparency of a Carbopol ETD 2020 gel. Part II. Int J Pharm 234:149–57
  • Cosco D, Paolino D, Maiuolo J, et al. (2015). Ultradeformable liposomes as multidrug carrier of resveratrol and 5-fluorouracil for their topical delivery. Int J Pharm 489:1–10
  • Dahan A, Hoffman A. (2008). Rationalizing the selection of oral lipid based drug delivery systems by an in vitro dynamic lipolysis model for improved oral bioavailability of poorly water soluble drugs. J Control Release 129:1–10
  • Darwhekar G, Jain DK, Choudhary A. (2012). Elastic liposomes for delivery of neomycin sulphate in deep skin infection. Asian J Pharm Sci 7:230–40
  • Diasio RB, Harris BE. (1989). Clinical pharmacology of 5-fluorouracil. Clin Pharmacokinet 16:215–37
  • Draize J, Woodard G, Calvery H. (1944). Methods for the study of irritation and toxicity of substance applied to the skin and mucous membranes. J Pharmacol Exp Ther 82:377–90
  • El Maghraby GM, Williams AC, Barry BW. (2001). Skin delivery of 5-fluorouracil from ultradeformable and standard liposomes in-vitro. J Pharm Pharmacol 53:1069–77
  • Fraile RJ, Baker LH, Buroker TR, et al. (1980). Pharmacokinetics of 5-fluorouracil administered orally, by rapid intravenous and by slow infusion. Cancer Res 40:2223–8
  • Grit M, Underberg WJ, Crommelin DJ. (1993). Hydrolysis of saturated soybean phosphatidylcholine in aqueous liposome dispersions. J Pharm Sci 82:362–6
  • Hussain A, Samad A, Nazish I, Ahmed FJ, et al. (2013). Nanocarrier-based topical drug delivery for an antifungal drug. Drug Dev Ind Pharm 40:527–41
  • Hussain A, Samad A, Ramzan M, et al. (2014a). Elastic liposome-based gel for topical delivery of 5-fluorouracil: in vitro and in vivo investigation. Drug Deliv 14:1–15
  • Hussain A, Samad A, Singh SK, et al. (2014b). Nanoemulsion gel-based topical delivery of an antifungal drug: in vitro activity and in vivo evaluation. Drug Deliv 21:1–16
  • Jain SK, Gupta Y, Jain A, Rai K. (2008). Enhanced transdermal delivery of acyclovir sodium via elastic liposome. Drug Deliv 15:141–7
  • Kaiser N, Kimpfler A, Massing U, et al. (2003). 5-Fluorouracil in vesicular phospholipid gels for anticancer treatment: entrapment and release properties. Int J Pharm 256:123–31
  • Khurana S, Jain NK, Bedi PM. (2013). Nanoemulsion based gel for transdermal delivery of meloxicam: physico-chemical, mechanistic investigation. Life Sci 92:383–92
  • Lai LF, Guo HX. (2011). Preparation of new 5-fluorouracil-loaded zein nanoparticles for liver targeting. Int J Pharm 404:317–23
  • Monti D, Saettone MF, Giannaccini B, Galli-Angeli D. (1995). Enhancement of transdermal penetration of dapiprazole through hairless mouse skin. J Control Release 33:71–7
  • Pagano R, Thompson TE. (1968). Spherical lipid bilayer membranes: electrical and isotopic studies of ion permeability. J Mol Biol 38:41–57
  • Shakeel F, Baboota S, Ahuja A, et al. (2008). Skin permeation mechanism of aceclofenac using novel nanoemulsion formulation. Pharmazie 63:580–4
  • Singh BN, Singh RB, Singh J. (2005). Effects of ionization and penetration enhancers on the transdermal delivery of 5-fluorouracil through excised human stratum corneum. Int J Pharm 298:98–107
  • Singh HP, Tiwary AK, Jain S. (2010). Preparation and in vitro, in vivo characterization of elastic liposomes encapsulating cyclodextrin-colchicine complex for topical delivery of colchicine. Yakugaku Zasshi 130:397–407
  • Tanaka F, Fukuse T, Wada H, Fukushima M. (2000). The history, mechanism and clinical use of oral 5-fluorouracil derivative chemotherapeutic agents. Curr Pharm Biotechnol 1:137–64
  • Touitou E, Abed L. (1985). Effect of propylene glycol, Azone and n-decylmethyl sulfoxide on skin permeation kinetics of 5-fluorouracil. Int J Pharm 27:89–98
  • Tsukada S, Ueda S, Okada R. (1984). Preparation of liposome encapsulated antitumor drugs relationship between lipophilicity of and in vitro drug release. Chem Pharm Bull 32:1929–35
  • Tutrone WD, Saini R, Caglar S, et al. (2003). Topical therapy for actinic keratoses I: 5-fluorouracil and imiquimod. Cutis 71:365–70
  • Utreja P, Jain S, Tiwar AK. (2011). Localized delivery of paclitaxel using elastic liposomes: formulation development and evaluation. Drug Deliv 18:367–76
  • Verma S, Singh SK, Verma PR, Ahsan MN. (2014). Formulation by design of felodipine loaded liquid and solid self nanoemulsifying drug delivery systems using Box–Behnken design. Drug Dev Ind Pharm 40:1358–70
  • Williams AC, Barry BW. (1991). Terpenes and the lipid-protein-partitioning theory of skin penetration enhancement. Pharm Res 8:17–24

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.