109
Views
0
CrossRef citations to date
0
Altmetric
Research Articles

Design of novel quinazolinone derivatives as inhibitors for 5HT7 receptor

, , &
Pages 3-16 | Received 22 Jun 2011, Accepted 31 Jul 2011, Published online: 16 Dec 2011

References

  • Millan MJ. The neurobiology and control of anxious states. Prog Neurobiol 2003, 70, 83–244.
  • Na YH, Hong SH, Lee JH, Park WK, Baek DJ, Koh HY, Cho YS, Choo H, Pae AN. Novel quinazolinone derivatives as 5-HT7 receptor ligands. Bioorg Med Chem 2008, 16, 2570–2578.
  • Hoyer D, Hannon JP, Martin GR. Molecular, pharmacological and functional diversity of 5-HT receptors. Pharmacol Biochem Behav 2002, 71, 533–554.
  • Peter BH, Gregor JS. Functional, molecular and pharmacological advances in 5HT7 receptor research. Trends Pharmacol Sci 2004, 25, 481–486.
  • Schildkraut JJ. The catecholamine hypothesis of affective disorders: a review of supporting evidence. Am J Psychiatry 1965, 122, 509–522.
  • Bourin M. Psychopharmacological treatment of depression. Bull Clin Psychopharmacol 2001, 11, 46–52.
  • Christopher EJ. Electroconvulsive therapy in the medically ill. Curr Psychiatry Rep 2003, 5, 225–230.
  • Cramer RD 3rd, Patterson D, Bunce JD. Comparitive molecular field analysis (CoMFA) 1. Effect of shape on binding of steriods to carrier proteins. J Am Chem Soc 1998, 110, 5959–5967.
  • Cramer RD 3rd, Patterson DE, Bunce JD. Crossvalidation, bootstrapping, and partial least squares compared with multiple regression in conventional QSAR studies. Quant Struct Act Relat 1998, 7, 18–25.
  • Klebe G, Abraham U, Mietzner T. Molecular similarity indices in a comparative analysis (CoMSIA) of drug molecules to correlate and predict their biological activity. J Med Chem 1994, 37, 4130–4146.
  • Sybyl version 6.9, Tripos Associates, St Louis (MO), 1999.
  • Gasteiger J, Marsili M. Iterative partial equalization of orbital electronegativity − a rapid access to atomic charges. Tetrahedron 1980, 36, 3219–3228.
  • Wold S, Johansson A, Cochi M. 3D-QSAR in drug design: theory, methods and application. In: Kubinyi H, ed. PLS-Partial least squares projection to latent structures. ESCOM, Lieden, 1993, 523–550.

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.