17
Views
2
CrossRef citations to date
0
Altmetric
Research Article

[123I/125I]-RO 43-0463, A site specific tracer for MAO-B mapping with autoradiography as well as with spet

, , , , &
Pages 581-593 | Published online: 26 Sep 2008

References

  • Haefely W. E., Kettler R., Keller H. H., Da Prada M. Ro 19-6327, a reversible and highly selective monoamino oxidase B inhibitor: a novel tool to explore the MAO-B function in humans. Advances in Neurolgy, Vol. 53: Parkinson's Disease: Anatomy, Pathology, and Therapy, M. B. Streifler, A. D. Korczyn, E. Melamed, M. B.H. Youdim. Raven Press, New York 1990; 505–512
  • Kyburz E. New developments in the field of MAO inhibitors. Drug News and Perspectives 1990; 3: 592–599
  • Richards G., Saura J., Ulrich J., Da Prada M. Molecular neuroanatomy of monoamine oxidase in human brainstem. Psychopharmacology 1992; 106: 21–23
  • Strohlin-Benedetti M., Dostert Ph. Monoamine oxidase. brain aging and degenerative diseases. Biochem. Pharmacol. 1989; 38: 555–561
  • Oreland L., Gottfries C. D. Brain monoamine oxidase in aging and in dementia of Alzheimer type. Prog. Neuropsychopharmacol. Biol. Psychiatr. 1986; 10: 533–540
  • Jossan S. S., Gilberg P.-G., Karlsson I., Gottfries C. D., Oreland L. Visualization of brain monoamine oxidase B (MAO-B) in dementia of Alzheimer's type by means of large cryosection autoradiography; a pilot study. J. Neurotransm. 1990; 32: 61–66
  • Parkinson study group. Effect of deprenyl on the progression of disability in early Parkinson's disease. N. Engl. J. Med. 1989; 321: 1364–1371
  • Parkinson study group. DATATOP: a multicenter controlled clinical trial in early Parkinson's disease. Arch. Neurol. 1989; 46: 1052–1060
  • Bench C. J., Price G. W., Lammertsma A. A., Cremer J. C., Luthra S. K., Turton D., Dolan R. J., Kettler R., Dingemanse J., Da Prada M., Biziere K., McClelland G. R., Jamieson V. L., Wood N. D., Frackowiak R. S.J. Measurement of human cerebral monoamine oxidase type B (MAO-B) activity with positron emission tomography (PET): a dose ranging study with the reversible inhibitor Ro 19-6327. Eur. J. Clin. Pharmacol. 1991; 40: 169–173
  • Da Prada M., Kettler R., Keller H. H., Burkard W. P. Ro 19-6327, a reversible, highly, selective inhibitor of type B monoamine oxidase, completely devoid of tyramine-potentiating effects: comparison with selegiline. Progress in catecholamine research, Part B: Central aspects. Alan R. Liss. 1988; 359–363
  • MacWhorter S. E., Baldwin R. M. Synthesis and biodistribution of 123I N-(2-aminoethyl)-5-iodo-2-pyridinecarboxamide (Ro 43-0463). a monoamine oxidase B inhibitor. Nucl. Med. Biol. 1991; 18: 563–564
  • Beer H.-F., Sha L., Novak-Hofer I., Bläuenstein P., Schubiger P. A. Large scale preparation strategy for labelling of [123I]-SCH 23982. a dopamine D1 receptor binding agent. Appl. Radiat. Isot. 1992; 46: 781–787
  • Kettler R., Dr. Hoffmann-La Roche. Basle CH, Personal communication from
  • Cesura A. M., Galva M. D., Imhof R., Kyburz E., Picotti G. B., Da Prada M. [3H]-Ro 19-6327: a reversible ligand and affinity labelling probe for monoamine oxidase-B. Eur. J. Pharmacol. 1989; 162: 457–465
  • Wyss R., Philipp W. Determination of the monoamine oxidase B inhibitor Ro 19-6327 in plasma by high-performance liquid chromatography using precolumn derivatization with fluorescamine and fluorescence detection. J. Chrom. 1990; 507: 187–198
  • Winchell H. S., Baldwin R. M., Lin T. H. Development of I-123-labeled amines for brain studies: localization of I-123-iodophenylalkyl amines in rat brain. J. Nucl. Med. 1980; 21: 940–946
  • Berman M., Braverman L. E., Burke J., De Groot L., McCormack K. R., Oddie T. H., Rohrer R. H., Wellman H. N., Smith E. M. MIRD/dose estimate report No. 5, summary of current radiation dose estimates to humans from 123I, 124I, 125I, 126I, 130I, 131I, and 132I as sodium iodide. J. Nucl. Med. 1975; 16: 857–860
  • Hasler P. H., Beer H.-F., Frey L. D., Rosetti I., Schubiger P. A. Biodistribution and Estimated Radiation Burden for a New I-123 Labelled Monoamine Oxidase-B Inhibitor (Ro 43-0463). J. Nucl. Biol. Med., accepted
  • Saura M. J., Kettler R., Da Prada M., Richards G. Molecular neuroanatomy of MAO-A and MAO-B. J. Neural Transm. 1990; 32: 49–53
  • Saura J., Kettler R., Da Prada M., Richards J. G. Quantitative enzyme radioautography with 3H-Ro 41-1049 and 3H-Ro 19-6327 in vitro: Localization and Abundance of MAO-A and MAO-B in rat CNS, peripheral organs, and human brain. J. Neuroscience 1992; 12: 1977–1999

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.