153
Views
0
CrossRef citations to date
0
Altmetric
Research Article

Effects of hexagonal boron nitride on dry compression mixture of Avicel DG and Starch 1500

&
Pages 415-427 | Received 05 Nov 2014, Accepted 27 Jan 2015, Published online: 26 Feb 2015

References

  • Bastos MO, Friedrich RB, Beck RCR. Effects of filler-binders and lubricants on physicochemical properties of tablets obtained by direct compression: a 22 factorial design. Lat Am J Pharm 2008;27: 578–583
  • Otsuka M, Yamane I, Matsuda Y. Effects of lubricant mixing on compression properties of various kinds of direct compression excipients and physical properties of the tablets. Advanced Powder Technol 2004;15:477–493
  • Wang J, Wen H, Desai D. Lubrication in tablet formulations. Eur J Pharm Biopharm 2010;75:1–15
  • Santl M, Ilija I, Vrecer F, Baumgartner A. A compressibility and compactibility study of real tableting mixtures: the effect of granule particle size. Acta Pharm 2012;62:325–340
  • Mosig J, Kleinebudde P. Evaluation of lubrication methods: how to generate a comparable lubrication for dry granules and powder material for tableting processes. Powder Technol 2014;266:156–166
  • Pingali K, Mendez R, Lewis D, et al. Mixing order of glidant and lubricant-influence on powder and tablet properties. Int J Pharm 2011;409:269–277
  • Kikuta J, Kitamori N. Effect of mixing time on the lubricating properties of magnesium stearate and the final characteristics of the compressed tablet. Drug Dev Ind Pharm 1994;20:343–355
  • Bacher C, Olsen PM, Sonnergaard JM. Compressibility and compactibility of granules produced by wet and dry granulation. Int J Pharm 2008;358:69–74
  • Kara A, Tobyn MJ, Stevens R. An application for zirconia as a pharmaceutical die set. J Eur Ceram Soc 2004;24:3091–3101
  • Yamamura T, Ohta T, Ogawa Y, et al. Effects of automated external lubrication on tablet properties and the stability of eprazinone hydrochloride. Int J Pharm 2009;370:1–7
  • Dawes J, Allenspach C, Gamble JF, et al. Application of external lubrication during the roller compaction of adhesive pharmaceutical formulations. Pharm Dev Technol 2013;18:246–256
  • Patel S, Kaushal AM, Bansal AK. Lubrication potential of magnesium Stearate studied on instrumented rotary tablet press. AAPS PharmSciTech 2007;8:57–64
  • Late SG, Yu Y-Y, Banga AK. Effects of disintegration promoting agent, lubricants and moisture treatment on optimized fast disintegrating tablets. Int J Pharm 2009;365:4–11
  • Turkoglu M, Sakr A. Tablet dosage forms. In: Florence AT, Siepmann J, eds. Modern pharmaceutics. Basic principles and systems. Vol. 1. Pinehurst, North Caroline, USA: PharmaceuTech, Inc.; 2009:481–497
  • Ugurlu T, Turkoglu M. Hexagonal boron nitride as a tablet lubricant and a comparison with conventional lubricants. Int J Pharm 2008;353:45–51
  • Ugurlu T, Halacoğlu MD. Effects of some lubricants and evaluation of compression parameters on directly compressible powders. Pharm Dev Technol 2014;19:347–354
  • Halacoglu MD, Ugurlu T. Compression parameters of Hexagonal Boron Nitride on direct compression mixture of microcrystalline cellulose and modified starch. Pharm Dev Technol 2014;20:1–8
  • Baraton MI, Merle T, Quintard P, Lorenzelli V. Surface activity of a boron nitride powder: a vibrational study. Langmuir 1993;9:1486–1491
  • Golberg D, Bando Y, Huang Y, et al. Boron nitride nanotubes and nanosheets. ACS Nano 2010;4:2979–2993
  • Ciofani G, Raffa V, Menciassi A, Cuschieri A. Boron nitride nanotubes: an innovative tool for nanomedicine. Nano Today 2009;4:8–10
  • Turkoglu M, Sahin I, San T. Evaluation of hexagonal boron nitride as a new tablet lubricant. Pharm Dev Technol 2005;10:381–388
  • Staniforth JN, Aulton ME. Powder flow. In: Aulton ME, ed. Aulton’s pharmaceutics, the design and manufacture of medicines. Philadelphia: Churchill Livingstone Elsevier; 2007:168–179
  • European Pharmacopoeia 7.0 (2.9.36). Powder flow. Strasbourg: Council of Europe; 2011:305–311
  • Fell JT, Newton JM. Determination of tablet strength by the diametrical compression test. J Pharm Sci 1970;59:688–691
  • Davies PN, Worthington HEC, Podczeck F, Newton JM. The determination of the mechanical strength of tablets of different shapes. Int J Pharm 2003;258:153–163
  • Röscheisen G, Schmidt PC. The combination of factorial design and simplex method in the optimization of lubricants for effervescent tablets. Eur J Biopharm 1995;41:302–308
  • Delacourte A, Predella P, Leterme P, et al. A method for quantitative evaluation of the effectiveness of the lubricants used in tablet tecnology. Drug Dev Ind Pharm 1993;19:1047–1060
  • Heckel RW. Density pressure relationship in powder compaction. Transect Metal Soc AIME 1961;221:671–675
  • Heckel RW. An analysis of powder compaction phenomena. Transect Metal Soc AIME 1961;221:1001–1008
  • Kuny TJ. Compression behavior of the enzyme β-galactosidase [Ph.D. Thesis]. Switzerland: University of Bassel; 2004
  • Wadke DA, Serajuddin ATM, Jacobsen H. Preformulation testing. In: Lieberman HA, Lachman L, Schwartz JB, eds. Pharmaceutical dosage forms-tablets. Vol. 1, 2nd ed. New York: Marcel Dekker, Inc.; 1989:1–74
  • Staniforth J. Powder flow. In: Aulton ME, ed. Pharmaceutics. The science of dosage form design. London: Churchill Livingstone, Elsevier Limited; 2002:197–210
  • Kılıcarslan M, Mamca R, Imamoglu S, et al. Investigation on the flow properties of different direct tableting agents by using pyridoxine hydrochloride as a model drug. J Fac Pharm, Ankara 2009;38:331–344
  • Singh I, Kumar P. Preformulation studies for direct compression suitability of cefuroxime axetil and paracetamol: a graphical representation using sedem diagram. Acta Pol Pharm-Drug Res 2012;69:87–93
  • Seppala K, Heinamaki J, Hatara J, et al. Development of a new method to get a reliable powder flow characteristics using only 1 to 2 g of powder. AAPS PharmSciTech 2010;11:402–408
  • Shah RB, Tawakkul MA, Khan MA. Comparative evaluation of flow for pharmaceutical powders and granules. AAPS PharmSciTech 2008;9:250–258
  • Villanova JCO, Ayres E, Orefice RL. Design of prolonged release tablets using new solid acrylic excipients for direct compression. Eur J Pharm Biopharm 2011;79:664–673
  • Langridge JR, Wells JI. Dicalcium phosphate dihy-drate-microcrystalline cellulose systems in direct compression tableting. Int J Pharm Tech Prod Mfr 1981;2:1–8
  • Aulton ME, Marok IS. Assessment of work-hardening characteristics of some tableting materials using Meyer's relationship. Int J Pharm Tech Prod Mfr 1981;2:1–6
  • Kochhar SK, Rubinstein MH, Barnes D. Slugging and recompression characterisation of some blends of pharmaceutical excipients. Int J Pharm 1994;112:225–231
  • Kochhar SK, Rubinstein MH, Barnes D. The effects of slugging and recompression on pharmaceutical excipients. Int J Pharm 1995;115:35–43
  • Herting MG, Kleinebudde P. Studies on the reduction of tensile strength of tablets after roll compaction/dry granulation. Eur J Pharm Biopharm 2008;70:372–379
  • Nakagawa H, Kano M, Hasebe S, et al. Real-time monitoring of lubrication properties of magnesium stearate using NIR spectrometer and thermal effusivity sensor. Int J Pharm 2013;441:402–413
  • Avicel DG. Speciality filler/binder for dry granulation. Application Bulletin, FMC Biopolymer. Available from: http://www.fmcbiopolymer.com/Portals/Pharm/Content/Docs/Avicel%20DG%20Brochure%2012-4-09.pdf [last accessed 18 Feb 2015]
  • Shah AC, Mlodozeniec AR. Mechanism of surface lubrication:influence of duration of lubricant-excipient mixing on processing characteristics of powders and properties of compressed tablets. J Pharm Sci 1977;66:1377–1382
  • Wade JB, Martin GP, Long DF. A methodological approach for determining the effects of moisture content on the compaction properties of powders: granular hydroxyapaptite. Powder Technol 2013;246:511–519
  • Alderborn G. Tablets and compaction. In: Aulton ME, ed. Aulton’s pharmaceutics, the design and manufacture of medicines. Philadelphia: Churchill Livingstone Elsevier; 2007:41–482
  • Patel SS, Patel NM. Development of directly compressible co-processed excipient for dispersible tablets using 32 full factorial design. Int J Pharm Pharmaceut Sci 2009;1:125–148
  • Çomoğlu T. An overview of compaction equations. J Fac Pharm Ankara 2007;36:123–133
  • Energy Dispersive Spectroscopy on the SEM: a primer, Bob Hafner, Characterization Facility, University of Minnesota—Twin Cities. Available from: http://www.charfac.umn.edu/instruments/eds_on_sem_primer.pdf [last accessed 18 Feb 2015]
  • Sindel U, Zimmermann I. Measurement of interaction forces between individual powder particles using an atomic force microscope. Powder Technol 2001;117:247–254
  • Binnig G, Rohrer H. Scanning tunneling microscopy. Helv Phys Acta 1982;55:726–735
  • Binnig G, Quate CF, Gerber C. Atomic force microscope. Phys Rev Lett 1986;56:930–933
  • Sahoo P. “Nanotribology” in engineering tribology. New Delhi: PHI Learning Private Limited; 2011
  • Bhushan B. Nanotribology and nanomechanics. Wear 2005;259:1507–1531
  • Bhushan B, Israelachivili JN, Landman U. Nanotribology: friction, wear, and lubrication at the atomic scale. Nature 1995;374:607–616
  • Conroy M, Armstrong J. A comparison of surf ace metrology techniques. J. Phys: Conf Ser 2005;13:458–465
  • Whitehouse DJ. The handbook of surface and nanometrology. Philadelphia, PA: Institute of Physics Publishing; 2003:383–483

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.