The effects of excipients for topical preparations on the human skin permeability of terpinen-4-ol contained in Tea tree oil: Infrared spectroscopic investigations

References

• Nenoff P, Haustein U, Brandt W. Antifungal activity of the essential oil of Melaleuca alternifolia (tea tree oil) against pathogenic fungi in vitro. Skin Pharmacol Phys 1996;9:388–394.
   Google Scholar
• Hammer KA, Carson CF, Riley TV. Antifungal effects of Melaleuca alternifolia (tea tree) oil and its components on Candida albicans, Candida glabrata and Saccharomyces cerevisiae. J Antimicrob Chemioth 2004;53(6):1081–1085.
   PubMed Web of Science ®Google Scholar
• Hart PH, Brand C, Carson CF, Riley TV, Prager RH, Finlay-Jones JJ. Terpinen-4-ol, the main component of the essential oil of Melaleuca alternifolia (tea tree oil), suppresses inflammatory mediator production by activated human monocytes. Inflamm Res 2000;49:619–626.
   PubMed Web of Science ®Google Scholar
• Guerry M, Chalchat JC, Fusillier C, Vasson MP, Guillot J. Anti-inflammatory effects of Melaleuca alternifolia essential oil on human polymorphonuclear neutrophils and monocytes. Free Radical Res 2004;38(8):805–811.
   PubMed Web of Science ®Google Scholar
• Bassett IB, Pannowitz DL, Barnetson RS. A comparative study of tea tree oil versus benzoyl peroxide in the treatment of acne. Med J Aust 1990;153(8):455–458.
   PubMed Web of Science ®Google Scholar
• Raman A, Weir U, Bloomfield SF. Antimicrobial effects of tea-tree oil and its major components on Staphylococcus aureus, Staph. epidermidis and Propionibacterium acnes. Lett Appl Microbiol 1995;21(4):242–245.
   PubMed Web of Science ®Google Scholar
• Beckmann B, Ippen H. Tea tree oil. Dermatosen in Beruf und Umwelt 1998;46(3):120–124.
   Google Scholar
• Hausen BM, Reichling J, Harkenthal M. Degradation products of monoterpenes are the sensitizing agents of Tea tree oil. Am J Contact Dermatitis 1999;10(2):68–77.
   PubMedGoogle Scholar
• Nielsen JB, Nielsen F. Topical use of tea tree oil reduces the dermal absorption of benzoic acid and methiocarb. Arch Derm Res 2006;297(9):395–402.
   PubMed Web of Science ®Google Scholar
• Cross SE, Russell M, Southwell I, Roberts MS. Human skin penetration of the major components of Australian tea tree oil applied in its pure form and as a 20% solution in vitro. Eur J Pharm Biopharm 2008;69:214–222.
   PubMed Web of Science ®Google Scholar
• Reichling J, Landvatter U, Wagner H, Kostka KH, Schaefer UF. In vitro studies on release and human skin permeation of Australian tea tree oil (TTO) from topical formulations. Eur J Pharm Biopharm 2006;64(2):222–228.
   PubMed Web of Science ®Google Scholar
• Cal K, Krzyzaniak M. Stratum corneum absorption and retention of linalool and terpinen-4-ol applied as gel or oily solution in humans. J Dermatol Sci 2006;42(3):265–267.
   PubMed Web of Science ®Google Scholar
• Cal K. Skin penetration of terpenes from essential oils and topical vehicles. Planta Med 2006;72(4):311–316.
   PubMed Web of Science ®Google Scholar
• Minghetti P, Casiraghi A, Cilurzo F, Montanari L, Marazzi M, Falcone L, Donati V. Comparison of different membranes with cultures of keratinocytes from man for percutaneous absorption of nitroglycerin. J Pharm Pharmacol 1999;51(6):729–734.
   PubMed Web of Science ®Google Scholar
• Bronaugh RL, Stewart RF, Simon M. Methods for in vitro percutaneous absorption studies VII: Use of excised human skin. J Pharm Sci 1986;75:1094–1097.
   PubMed Web of Science ®Google Scholar
• Sugibayashi K, Kobayashi D, Nakagaki E, Hatanaka T, Inoue N, Kusumi S, Kobayashi M, Kimura M, Morimoto Y. Differences in enhancing effect of l-menthol, ethanol and their combination between hairless rat and human skin. Int J Pharm 1995;113:189–197.
   Web of Science ®Google Scholar
• Crank J. The mathematics of diffusion. Oxford, UK: Oxford University Press; 1975.
   Google Scholar
• Vaddi HK, Ho PC, Chan SY. Terpenes in propylene glycol as skin-penetration enhancers: Permeation and partition of haloperidol, Fourier transform infrared spectroscopy and differential scanning calorimetry. J Pharm Sci 2002;91:1639–1651.
   PubMed Web of Science ®Google Scholar
• Bergonzi MC, Bilia AR, Casiraghi A, Cilurzo F, Minghetti P, Montanari L, Vincieri FF. Evaluation of skin permeability of sesquiterpenes of an innovative supercritical carbon dioxide, Arnica extract by HPLC/DAD/MS. Pharmazie 2005;60(1):36–38.
   PubMed Web of Science ®Google Scholar
• Narishetty STK, Panchagnula R. Transdermal delivery system for zidovudine: in vitro, ex vivo and in vivo evaluation. Biopharm Drug Dispos 2004;25(1):9–20.
   PubMed Web of Science ®Google Scholar
• Yamane MA, Williams AC, Barry BW. Effects of terpenes and oleic acid as skin penetration enhancers towards 5-fluorouracil as assessed with time; permeation, partitioning and differential scanning calorimetry. Int J Pharm 1995;116(2):237–251.
   Google Scholar
• Babita K, Kumar V, Rana V, Jain S, Tiwary AK. Thermotropic and spectroscopic behavior of skin: Relationship with percutaneous permeation enhancement. Curr Drug Del 2006;3(1):95–113.
   PubMedGoogle Scholar
• Songkro S, Becket G, Rades T. The effects of p-menthane monoterpenes and related compounds on the percutaneous absorption of propranolol hydrochloride across newborn pig skin. II. Infrared spectroscopic and thermal analysis investigations. STP Pharma Sci 2003;13(6):394–404.
   Google Scholar
• Ayala-Bravo HA, Quintanar-Guerrero D, Naik A, Kalia YN, Cornejo-Bravo JM, Ganem-Quintanar A. Effects of sucrose oleate and sucrose laureate on in vivo human stratum corneum permeability. Pharm Res 2003;20(8):1267–1273.
   PubMed Web of Science ®Google Scholar
• Naik A, Pechtold LARM, Potts RO, Guy RH. Mechanism of oleic acid-induced skin penetration enhancement in vivo in humans. J Control Release 1995;37(3):299–306.
   Web of Science ®Google Scholar
• Panchagnula R, Desu H, Jain A, Khandavilli S. Feasibility studies of dermal delivery of paclitaxel with binary combinations of ethanol and isopropyl myristate: Role of solubility, partitioning and lipid bilayer perturbation. Il Farmaco 2005;11–12:894–899.
   Google Scholar