In Vitro Permeation Study of a Mucoadhesive Drug Delivery System for Controlled Delivery of Nonoxynol-9

References

• Cramer D. W., Goldman M. B., Schiff I. The relationship of tubal infertility to barrier method and oral contraceptive use. JAMA 1987; 257: 2446–2450
   PubMed Web of Science ®Google Scholar
• Lauv W. C., Austin H., Alexander W. J., Stagno S., Cheeks J. A. Clinical trial of nonoxynol-9 for preventing gonococcal and chlamydial infections. J. Infec. Dis. 1988; 158: 518–523
   PubMed Web of Science ®Google Scholar
• Judson F. N., Ehret J. M., Bodin G. F., Levin M. J., Rietmeiyer C. A. In vitro evaluations of condoms with and without nonoxynol-9 as physical and chemical barriers against chlamydia trachomatis, Herpes simplex virus type 2 and human immunodeficiency virus. Sex Trans. Dis. 1989; 16: 51–56
   PubMed Web of Science ®Google Scholar
• Barbone F., Austin H., Lauv W. C., Alexander W. J. A follow-up study of methods of contraception, sexual activity and rates of trichomoniasis candidiasis and bacterial vaginosis. Am. J. Obstet. Gynecol. 1990; 163: 510–514
   PubMed Web of Science ®Google Scholar
• Miller C. J., Alexander N. J., Gettie A. The effect of contraceptives containing N-9 on the genital transmission of simian immunodeficiency virus in rhesus macaques. Fert. Steril. 1992; 57: 1126
   PubMed Web of Science ®Google Scholar
• Moench T. R., Whaley K. J., Mandrell T. D. The cat/feline immunodeficiency virus model for transmission by an infected cell inoculum. AIDS 1993; 7: 797
   PubMed Web of Science ®Google Scholar
• Vorhauser B. W., Dobbie T. A., Jr. Disposable spermicide releasing diaphragm, U. S. Patent. 4,393,871, July 19, 1983
   Google Scholar
• Roddy R. E., Cordero M., Cordero C., Fortney J. A. A dosing study of nonoxynol-9 and genital irritation. Int. J. STD AIDS 1993; 4: 286–290
   Web of Science ®Google Scholar
• Lee C. H., Anderson M., Chien Y. W. The characterization of in vitro spermicidal activity of chelating agent on human sperm. J. Pharm Sci. 1995, in press
   Web of Science ®Google Scholar
• Lee C. H., Bagdon R., Chien Y. W. Comparative in vitro spermicidal activity and synergistic effect of chelating agents with nonoxynol-9 on human sperm functionality. J. Pharm Sci. 1996; 85: 91–95
   PubMed Web of Science ®Google Scholar
• Knuth K., Mansoor A., Robinson J. R. Hydrogel delivery systems for vaginal and oral applications: Formulation and biological consideration. Adv. Drug Del. Rev. 1993; 11: 137–164
   Web of Science ®Google Scholar
• Ishida M., Nambu N., Nagai T. Ointment-type oral mucosal dosage form of carbopol containing prednisolone for treatment of aphtha. Chem. Pharm. Bull. 1983; 31: 1010–1014
   PubMed Web of Science ®Google Scholar
• Robinson J. R., Bologna W. J. Vaginal and reproductive system treatment using a bioadhesive polymer. J. Cont. Rel. 1994; 28: 87–94
   Web of Science ®Google Scholar
• Lee C. H., Chien Y. W. Development and evaluation of a mucoadhesive drug-delivery system for dual-controlled delivery of nonoxynol-9 (I). J. Cont. Rel. 1995, in press
   Web of Science ®Google Scholar
• Aungst B. J., Rogers N. J. Site dependence of absorption-promoting actions of laureth-9, Na salicylate, Na2EDTA, and aprotinin on rectal, nasal, and buccal insulin delivery. Pharm Res. 1988; 5: 305–308
   PubMed Web of Science ®Google Scholar
• Suzuka T., Furuya A., Kamada A., Nishihata T. Effect of phenothiazines, disodium ethylenediamine-tetraacetic acid and diethyl maleate on in vitro rat colonic transport of cefmetazole and inulin. J. Pharmacobio-Dyn. 1987; 10: 63–71
   PubMedGoogle Scholar
• Burgos M. H., Roig de Varnas-Linares C. E. UI-trastructure of the vaginal mucosa. The Human Vagina, E. S.E. Hafez, T. N. Evans. North Holland Publishing Co., New York 1978; 63–93
   Google Scholar
• Richardson J. L., Illum L. The vaginal route of peptide and protein drug delivery. Adv. Drug Del. Rev. 1992; 8: 341–366
   Web of Science ®Google Scholar
• Lee P. I. Dimensional changes during drug release from a glassy hydrogel matrix. Polym. Commun. 1983; 24: 45–47
   Web of Science ®Google Scholar
• Transdermal Controlled Systemic Medications, Y. W. Chien. Marcel Dekker, New York 1987; 25–59
   Google Scholar
• Toddywala R., Chien Y. W. Evaluation of silicone-based pressure-sensitive adhesives for transdermal drug delivery. I. Effect of penetrant hydrophilicity. J. Cont. Rel. 1990; 14: 29–41
   Web of Science ®Google Scholar
• Higuch T. Mechanisms of sustained action medication: Theoretical analysis of the rate of release of solid drugs dispersed in solid matrices. J. Pharm. Sci. 1963; 52: 1145–1149
   PubMed Web of Science ®Google Scholar
• Tojo K. P., Masi J. A., Chien Y. W. Hydrody-namic characteristics of an in vitro drug permeation cell. Ind. Eng. Chem. Fundam. 1985; 24: 368
   Google Scholar
• Tojo K. P., Keshary P., Chien Y. W. Design and calibration of in vitro permeation apparatus. Transdermal Controlled Systemic Medications, Y. W. Chien. Marcel Dekker, New York 1987; 127–158
   Google Scholar
• Keshary P., Huang Y. C., Chien Y. W. Mechanism of transdermal controlled nitroglycerin administration (III): Control of skin permeation rate and optimization. Drug Dev. Ind. Pharm. 1985; 11: 1213–1253
   Web of Science ®Google Scholar
• Kabadi M. B., Chien Y. W. Intravaginal controlled administration of flurogestone acetate III: Development of rate-control vaginal devices. Drug Dev. Ind. Pharm. 1985; 11: 1271–1312
   Web of Science ®Google Scholar
• Kabadi M. B., Chien Y. W. Intravaginal controlled administration of flurogestone acetate IV: In vitro and in vivo correlation for intravaginal drug delivery from rate-control vaginal pessary. Drug Dev. Ind. Pharm. 1985; 11: 1313–1361
   Web of Science ®Google Scholar
• Ruckebush Y., Phaneuf L., Dunlop R. Reproductive life and cycles in animals. Physiology of small and large animals, Y. Ruckebush, L. Phaneuf, R. Dunlop. B. C. Decker, Philadelphia 1991; 573–587
   Google Scholar
• Corbo D. C., Liu J. C., Chien Y. W. Characterization of the barrier properties of mucosal membrane. J. Pharm. Sci. 1990; 79: 202
   PubMed Web of Science ®Google Scholar
• Yu K. Intravaginal delivery of nonoxynol-9: In vitro characterization. Ph.D. thesis, Rutgers University. 1994
   Google Scholar
• Tomeczek L., Reid G., Cuperus P. L., Mcgroarty J. A., van der Mei H. C., Bruce A. W., Khoury A. E., Busscher H. J. Correlation between hydro-phobicity and resistence to nonoxynol-9 and vancomycin for urogenital isolates of lactobacilli. FEMS Microbiol. Lett. 1992; 94: 101–104
   Web of Science ®Google Scholar
• Leung S. S., Robinson J. R. The contribution of anionic polymer structural features to mucoadhesion. J. Com. Release 1988; 5: 223
   Google Scholar