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Research Article

Buoyancy and Drug Release Patterns of Floating Minitablets Containing Piretanide and Atenolol as Model Drugs

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Pages 73-84 | Received 17 Mar 1997, Accepted 30 Jul 1997, Published online: 27 Sep 2008

References

  • Timmermans J., Moës A. J. Factors controlling the buoyancy and gastric retention capabilities of floating matrix capsules: new data for reconsidering the controversy. J. Pharm. Sci. 1994; 83: 18–24
  • Doelker E. Novel methods of producing controlled release hard gelatin capsules. Proceedings Capsugel Symposium. Hamburg 1988; 7–15
  • Bongiovanni G., Calanchi M., Marconi M. Multiparticulate sustained release matrix system, International Patent Application. A61K9/48,9/20, 1–13, 1992
  • Follonier N., Doelker E. Biopharmaceutical comparison of oral multiple-unit and single-unit sustained-release dosage forms. S. T. P. Pharma 1992; 2: 141–158
  • Kawashima Y., Niwa T., Takeuchi H., Hino T., Itoh Y. Preparation of multiple unit hollow microspheres (microballoons) with acrylic resin containing tranilast and their drug release characteristics (in vitro) and floating behavior (in vivo). J. Controlled Release 1991; 16: 279–290
  • Icnikawa M., Kato T., Kawahara M., Watanabe S., Kayano M. A new multiple-unit oral floating dosage system. II: In vivo evaluation of floating and sustained-release characteristics with p-aminobenzoic acid and isosorbide dinitrate as model drugs. J. Pharm. Sci. 1991; 80: 1153–1156
  • Ruhnke A. Einfluss der Dichte von Pellets auf die Verweildauer im Magen und die Absorption eines Modell-Arzneistoffes. Ph. D. Thesis, University of Hamburg. 1989
  • Lippold B. C., Günther J. In-vivo Prüfung einer muitipartikularen Retard-Schwimmarzneiform. Eur. J. Pharm. Biopharm. 1991; 37: 254–261
  • Colombo P., Conte U., Caramella C., Gazzaniga A., La Manna A. Compressed polymeric mini-matrices for drug release control. J. Controlled Release 1985; 1: 283–289
  • Gazzaniga A., Conte U., Sangalli M. E., Caramella C., La Manna A. A multiple unit modified release system. Polymers in Medicine III, C. Migliaresi, et al. Elsevier Science Publishers B.V., Amsterdam 1988; 201–208
  • Rouge N., Cole E. T., Buri P., Doelker E. Screening of the potentially excipients for floating minitablets. S. T. P. Pharma 1997, in press
  • Brockmeier D., Grigoleit H.-G., Heptner H., Meyer B. H. Kinetics of piretanide absorption from the gastrointestinal tract. Methods Find. Exp. Clin. Pharmacol. 1986; 8: 731–739
  • Brockmeier D., Grigoleit H.-G., Leonhardt H. The absorption of piretanide from the gastro-intestinal tract is site-dependent. Eur. J. Clin. Pharmacol. 1986; 30: 79–82
  • Taylor D. C. Sites and mechanisms of intestinal drug absorption. Pharm. Int. 1986; 7: 179–183
  • Rouge N., Buri P., Doelker E. Drug absorption sites in the gastrointestinal tract and dosage forms for site-specific delivery. Int. J. Pharm. 1996; 136: 117–139
  • Rouge N., Leroux J. C., Cole E. T., Doelker E., Buri P. Prevention of the sticking tendency of the minitablets filled into hard gelatin capsules. Eur. J. Pharm. Biopharm. 1996; 43: 165–171
  • Timmermans J., Moës A. J. Apparatus and method for resultant-weight measuring system, US Patent Application. 5,076,107, 1991
  • Timmermans J. Floating hydrophilic matrix dosage forms for oral use: factors controlling their buoyancy and gastric residence capabilities. Ph.D. Thesis, University of Brussels. 1991
  • Uekama K., Matsubara K., Abe K., Horiuchi Y., Hirayama F., Suzuki N. Design and in vitro evaluation of slow-release dosage form of piretanide: utility of β-cyclodextrin: cellulose derivative combination as a modified-release drug carrier. J. Pharm. Sci. 1990; 79: 244–247
  • Doherty C., York P. Mechanisms of dissolution of furosemide/PVP solid dispersions. Int. J. Pharm. 1987; 34: 197–205
  • Peppas N. A. Analysis of Fickian and non-Fickian drug release from polymers. Pharm. Acta Helv. 1985; 60: 110–111
  • Ritger P. L., Peppas N. A. A simple equation for description of solute release. II. Fickian and anomalous release from swellable device. J. Controlled Release 1987; 5: 37–42
  • Ostberg T., Lund E. M., Graffner C. Calcium alginate matrices for oral multiple unit administration: IV. Release characteristics in different media. Int. J. Pharm. 1994; 112: 241–248
  • Conte U., Maggi L., La Manna A. Swellable/erodible barriers for the modulation of drug release from hydrophilic matrices. Proc. Int. Symp. Controlled Release Bioact. Mater. 1994; 21: 60–61
  • Doelker E. Water-swollen cellulose derivatives in pharmacy. Hydrogels in Medicine and Pharmacy, Vol. II: Polymers, N. A. Peppas. CRC Press, Boca Raton, FL 1987; 115–160
  • Stockwell A. F., Davis S. S., Walker S. E. In vitro evaluation of alginate gel systems as sustained release drug delivery systems. J. Controlled Release 1986; 3: 167–175
  • Krögel I., Bodmeier R. Evaluation of the floating properties of coated drug delivery systems containing effervescent excipient. Eur. J. Pharm. Biopharm. 1996; 42: 21
  • Vazquez M. J., Seijas R. M., Gomez-Amoza J. L., Martinez-Pacheco R., Souto C., Concheiro A. Influence of dissolution medium and technological variables on release of atenolol from hydrophilic hydroxy-propylmethylcellulose. S. T. P. Pharma 1992; 2: 397–403

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