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Research Article

Inhibition of Ache: Structure-Activity Relationship Among Conformational Transition of Trp84 and Bimolecular Rate Constant

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Pages 547-556 | Received 20 Jan 2000, Published online: 27 Sep 2008

References

  • Rosenberry T. L. Acetylcholineaterase. Adv. Enzymol. 1975; 43: 103–218
  • Fersht A. R. Enzyme Structure and Mechanism, 2nd ed. W.H. Freeman & Company, NY 1985; 150–152
  • Sussman J. L., Harel M., Frolow F., Oefner C., Goldman A., Toker L., Silman I. Science 1991; 253: 872–879, Entry PDB 2ACE; authors: M. Harel, M.L. Raves, I. Silman & J.L. Sussman (23 June 1996).
  • Pathak D., Ngai K. L., Ollis D. L. J. Mol. Biol. 1988; 204(2)435–445
  • Pathak D., Ollis D. J. Mol. Biol. 1990; 214(2)497–525
  • Ordentlinch A., Barak D., Kronman C., Flahner Y., Leitner M., Segall Y., Ariel N., Cohen S., Velan B., Shafferman A. J. Biol. Chem. 1993; 268(23)17083–17095
  • Ordentlinch A., Barak D., Kronman C., Ariel N., Segall Y., Velan B., Shafferman A. J. Biol. Chem. 1995; 270(5)2082–2091
  • Leszczynski J. F., Rose G. D. Science 1986; 234: 849–855
  • Taylor P. Neurology 1998; 51(1Suppl 1)S30, discussion S65–7
  • Knopman D. S. Geriatrics 1998; 53: S31–34
  • Marta M., Gatta F., Pomponi M. Biochim. Biophys. Acta 1992; 1120(3)262–266
  • Ellman G. L., Courtney K. D., Andres V., Jr., Featherstone M. Biochem. Pharmacol. 1961; 7: 88–95
  • Nishioka T., Kitamura K., Fujita T., Nakajima M. Pestic. Biochem. Physiol. 1976; 6: 320–327
  • Harel M., Quinn D. M., Nair H. K., Silman I., Sussman J. J. Am. Chem. Soc. 1996; 118: 2340–2346
  • Hammond G. S. J. Am. Chem. Soc. 1955; 77: 334
  • Chen Y. L., Nielsen J., Hedberg K., Dunaiskis A., Jones S., Russo L., Ives J., Liston D. J. Med. Chem. 1992; 35: 1429–1434
  • Atack J. R., Yu Q. S., Liu C., Brzostowska M., Chrisey L., Brossi A., Greig N. H., Soncrant T. T., Rapoport S. I., Radunz H. H. Helv Chim Acta 1991; 74: 761–766
  • Pomponi M., Marta M., Sacchi S., Colella A., Patamia M., Gatta F., Capone F., Oliverio A., Pavone F. FEBS Lett. 1997; 409(2)155–160
  • Gilson M. K., Straatsma T. P., McCammon J. A., Ripoll D. R., Faerman C. H., Axelsen P. H., Silman I., Sussman J. L. Science 1994; 263: 1276–1278
  • Kronman C., Ordentlich A., Barak D., Velan B., Shafferman A. J. Biol. Chem. 1994; 269(45)27819–27822
  • Faerman C., Ripoll D., Bon S., LeFeuvre Y., Morel N., Massoulie J., Sussman J. L., Silman I. FEBS Lett. 1996; 386(1)65–71
  • Marquardt D. W.J. Soc. Ind. Appl. Math. 1963; 11: 431–441

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