Synthesis and antileishmanial and antimicrobial activities of some 2,3-disubstituted 3H-quinazolin-4-ones

References

• Zaika LL. Spices and herbs: their antimicrobial activity and its determination. J Food Safet 1975;9:97–118.
   Google Scholar
• Leon LL, Machado GMC, Carvalho-Paes LE, Grimaldi JG. Antigenic differences of Leishmania amazonensis isolate causing diffuse cutaneous leishmaniasis. Trans R Soc Trop Med Hyg 1990;84:678–80.
   PubMed Web of Science ®Google Scholar
• Korolkovas A, Burckhalter JH.Química Farmacêutica. Rio de Janeiro: Guanabara, 1988:39.
   Google Scholar
• Frezard F, Michalick MSM, Soares CF, Demicheli C. Novel methods for encapsulation of meglumine antimoniate into liposomes. Braz J Med Biol Res 2000;33:841–6.
   PubMed Web of Science ®Google Scholar
• Ji-Feng L, Lee J, Dalton AM, Grace B, Libing Y, Baldino CM, et al. Microwave-assisted one-pot synthesis of 2,3-disubstituted 3H-quinazolin-4-ones. Tetrahedron Lett 2005;46:1241–4.
   Web of Science ®Google Scholar
• Seleh MA, Abde-Mageed MF, Abdo MA, Abdel-Basset MS. Synthesis of novel 3H-quinazolin-4-ones containing pyrazolinone, pyrazole and pyrimidinone moieties. Molecules 2003;8:363–73.
   Web of Science ®Google Scholar
• Edward C, Lawson WA, Kinney MJ, Costanzo WJ, Hoekstra JA, Kauffman DK, et al. Structure-function study of quinazolinone-based vitronectin receptor (αVβ3) antagonists: computer-assisted analysis of ligand-receptor interactions. Lett Drug Des Discov 2004;1:14–18.
   Google Scholar
• Haruhiko F, Kobayashi T, Tokitoh T, Ytorii Y, Natsugari H. Synthetic studies on 3-arylquinazolin-4-ones: intramolecular nucleophilic aromatic substitution reaction of 2-carboxamido-3-arylquinazolin-4-ones and its application to the synthesis of secondary aryl amines. Tetrahedron 2005;61:4297–312.
   Web of Science ®Google Scholar
• Wolf JF, Rathnam TL, Sleevi MC, Campbell JA, Greenwood TD. Synthesis and anticonvulsant activity of some new 2-substituted 3-aryl-4(3H)-quinazolinones. J Med Chem 1990;33:161–6.
   PubMed Web of Science ®Google Scholar
• Mhaske SB, Argade NP. The chemistry of recently isolated naturally quinazolinone alkaloids. Tetrahedron 2006;62:9787–826.
   Web of Science ®Google Scholar
• Connolly DJ, Cusack D, O’Sullivan TP, Guiry PJ. Synthesis of quinazolinones and quinazolines. Tetrahedron 2005;61:10153–202.
   Web of Science ®Google Scholar
• Nosova EA, Lipunova GN, Charushin VN. Cyclization of 2-halobenzoylchlorides with dinucleophiles as a versatile approach to fused heterocycles. Russ Chem Bull Int Ed 2004;53:1137.
   Web of Science ®Google Scholar
• Ji-Feng Liu. Rapid synthesis of biologically active qunazolinone – natural products using microwave technology. Curr Organic Synth 2007;4:223–37.
   Web of Science ®Google Scholar
• Witt A, Bergman J. Synthesis and reactions of some 2-vinyl-3H-quinazolin-4-ones. Tetrahedron 2000;56:7245–53.
   Web of Science ®Google Scholar
• Arfan M, Khan R, Imran M, Khan H, Mehmood J. One-pot synthesis and antimicrobial activities of some 2-aryl/alkyl, 3-aminoquinazolin-4(3H)-ones. J Chem Soc Pak 2008;30:299–305.
   Web of Science ®Google Scholar
• Arfan M, Khan R, Anjum S, Ahmad S, Choudhary MI. Water promoted, microwave assisted oxidative novel deamination on N-aminoquinazolone. Chin Chem Lett 2008;19:161–5.
   Web of Science ®Google Scholar
• National Committee for Clinical Laboratory Standards. Method for broth dilution antifungal susceptibility testing yeast; approved standard, M27-A, 15, 10. Tuscon: NCCLS, VA Medical Center, 1996.
   Google Scholar
• National Committee for Clinical Laboratory Standards. Methods for dilution antimicrobial susceptibility tests for bacteria that grow aerobically, 3rd ed. Approved standard. NCCLS document M100-S12. Wayne, PA: NCCLS, 2002.
   Google Scholar
• Carron RA, Marran JM, Montero-Fernandozlago L, and Dominguez AA. Antimicrobial properties of some extracts obtained from some mediterranean plants of medicinal value. Plantes Medicinales ET Phytotherapie 1987;21:195–202.
   Google Scholar
• Atta-ur-rehman Choudhary, MI, Thomsen WJ. Manual of Bioassay Techniques for Natural Products Research. Amsterdam: Harvard Academic Press, 1999:12.
   Google Scholar
• Evan DA, ed. Hand Book on Isolation, Characterization and Cryopreservation of Leishmania. Geneva: WHO, 1989;7:10–12, 28.
   Google Scholar
• Ben Salah A, Zakraoui H, Zaatour A, Ftaiti A, Aafouri B, Garraoui A, et al. A randomized, placebo-controlled trial in Tunisia treating cutaneous leishmaniasis with paromomycin ointment. Am J Trop Med Hyg 1995;53:162–6.
   PubMed Web of Science ®Google Scholar
• Shariat M, Abdollahi S. Synthesis of benzoxazinone derivatives: a new route to 2-(N-phthaloylmethyl)-4H-3,1-benzoxazin-4-one. Molecules 2004;9:705–12.
   PubMed Web of Science ®Google Scholar
• Pei-Wen H, Tsong-Long H, Chin-Chung W, Fang-Rong C, Tsai-Wei W, Yang-Chang W. The evaluation of 2,8-disubstituted benzoxazinone derivatives as anti-inflammatory and anti-platelet aggregation agents. Bioorg Med Chem Lett 2005;15:2786–9.
   PubMed Web of Science ®Google Scholar
• Narasimhulu M, Mahesh KC, Reddy TS, Rajesh K, Venkateswarlu Y. Lanthanum(III) nitrate hexahydrate or p-toluenesulfonic acid catalyzed one-pot synthesis of 4(3H)-quinazolinones under solvent-free conditions. Tetrahedron Lett 2006;47:4381–3.
   Web of Science ®Google Scholar
• Paxton JD.Assay for antifungal activity. In:Hostemann K, Dey PM, Harborne JB, eds. Methods in Plant Biochemistry. London: Academic Press, 1991;6:33.
   Google Scholar