References
- Deiters A, Martin, SF. Synthesis of oxygen-and nitrogen-containing heterocycles by ring-closing metathesis. Chem Rev 2004;104:2199–238
- Harbert CA, Plattner JJ, Welch WM, et al. Neuroleptic activity in 5-aryltetrahydro-gamma-carbolines. J Med Chem 1980;23:635–43
- Abou-Gharbia M, Patel UR, Webb MB, et al. Antipsychotic activity of substituted gamma-carbolines. J Med Chem 1987;30:1818–23
- Paris D, Cottin M, Demonchaux P, et al. Synthesis, structure–activity relationships, and pharmacological evaluation of pyrrolo[3,2,1-ij]quinoline derivatives: potent histamine and platelet activating factor antagonism and 5-lipoxygenase inhibitory properties. Potential therapeutic application in asthma. J Med Chem 1995;38:669–85
- Anzini M, Cappelli A, Vomero S, et al. Novel, potent, and selective 5-HT3 receptor antagonists based on the arylpiperazine skeleton: synthesis, structure, biological activity, and comparative molecular field analysis studies. J Med Chem 1995;38:2692–704
- Bendale P, Olepu S, Suryadevara PK, et al. Second generation tetrahydroquinoline-based protein farnesyltransferase inhibitors as antimalarials. J Med Chem 2007;50:4585–605
- Bulbule VJ, Rivas K, Verlinde CLMJ, et al. 2-Oxotetrahydroquinoline-based antimalarials with high potency and metabolic stability. J Med Chem 2008;51:384–7
- Konishi M, Ohkuma H, Tsuno T, et al. Crystal and molecular structure of dynemicin A: a novel 1,5-diyn-3-ene antitumor antibiotic. J Am Chem Soc 1990;112:3715–16
- Wender PA, Zercher CK, Beckham S, et al. A photochemically triggered DNA cleaving agent: synthesis, mechanistic and DNA cleavage studies on a new analog of the anti-tumor antibiotic dynemicin. J Org Chem 1993;58:5867–69
- Gudmundsson KS, Boggs SD, Catalano JG, et al. Imidazopyridine-5,6,7,8-tetrahydro-8-quinolinamine derivatives with potent activity against HIV-1. Bioorg Med Chem Lett 2009;19:6399–403
- Jarvest RL, Armstrong SA, Berge JM, et al. Definition of the heterocyclic pharmacophore of the bacterial methionyl tRNA synthetase inhibitors: potent antibacterially active non-quinolone analogues. Bioorg Med Chem Lett 2004;14:3937–41
- Yamada N, Kadowaki S, Takahashi K, et al. MY-1250, a major metabolite of the anti-allergic drug repirinast, induces phosphorylation of a 78-kDa protein in rat mast cells. Biochem Pharmacol 1992;44:1211–13
- Faber K, Stueckler H, Kappe T. Non-steroidal anti-inflammatory agents. 1. Synthesis of 4-hydroxy-2-oxo- 1,2–dihydroquinolin-3-yl alkanoic acids by the Wittig reaction of quinisatines. J Heterocycl Chem 1984;21:1177–81
- Sridharan V, Suryavanshi PA, Menéndez JC. Advances in the chemistry of tetrahydroquinolines. Chem Rev 2011;111:7157–259
- Dai Y, Hartandi K, Ji Z, et al. Discovery of N-(4-(3-amino-1H-indazol-4-yl)phenyl)-N′-(2-fluoro-5-methylphenyl) urea (ABT-869), a 3-aminoindazole-based orally active multitargeted receptor tyrosine kinase inhibitor. J Med Chem 2007;50:1584–97
- Jones TK, Goldman ME, Pooley CLF, et al. Preparation of quinolines and fused quinolines as steroid receptor modulators. 1996; WO9619458A2
- D'Amato V, Rosa R, D'Amato C, et al. The dual PI3K/mTOR inhibitor PKI-587 enhances sensitivity to cetuximab in EGFR-resistant human head and neck cancer models. Br J Cancer 2014;110:2287–95
- Buonora P, Olsen JO, Oh T. Recent developments in imino Diels–Alder reactions. Tetrahedron 2001;57:6099–138
- Kouznetsov VV, Bohorquez ARR, Stahenko EE. Three-component imino Diels–Alder reaction with essential oil and seeds of anise: generation of new tetrahydroquinolines. Tetrahedron Lett 2007;48:8855–60
- Lin XF, Cui SL, Wang YG. A highly efficient synthesis of 1,2,3,4-tetrahydroquinolines by molecular iodine-catalyzed domino reaction of anilines with cyclic enol ethers. Tetrahedron Lett 2006;47:4509–12
- Yadav JS, Reddy BVS, Rao RS, et al. InCl3-catalyzed hetero-Diels–Alder reaction: an expeditious synthesis of pyranoquinolines. Tetrahedron 2002;58:7891–6
- Zhou R, Huang W, Ren W, et al. Synthesis of cis or trans 4-heteroaromatic substituted furano and pyrano[3,2-c]tetrahydroquinolines by one pot imino Diels–Alder reactions. Heterocycles 2013;87:2495–500