26
Views
11
CrossRef citations to date
0
Altmetric
Research Article

Thrombin Inhibitors Based on Ketone Derivatives of Arginine and Lysine

, , , , &
Pages 43-60 | Received 17 Jun 1994, Published online: 27 Sep 2008

References

  • Jakubowski J. A., Smith G. F., Sall D. J. Ann. Rep. Med. Chem. 1992; 27: 27
  • Tapparelli C., Metternich R., Ehrhardt C., Cook N. S. Trends Pharma. Sci 1993; 14: 14
  • Szelke M., Leckie B. J., Hallett A., Jones D. M., Sueiras-Diaz J., Atrash B., Lever A. F. Nature (Lond.) 1982; 299: 555
  • Szelke M., Jones D. M., Dudman P. A., Atrash B., Sueiras-Diaz J., Leckie B. J. Peptides: Chemistry, Structure and Biology, J. E. Rivier, G. R. Marshall. Escom, Leiden 1990; 78
  • Sharpe R., Szelke M., G.B. Patent 1, 587,809, 1977, corresponding foreign patents
  • Schechter L., Berger A. Biochem. Biophys. Res. Commun. 1967; 27: 27
  • Szelke M., Jones D. M., European Patent 118,280, 1984, G.B. priority date 4–3–83
  • Jones D. M., Atrash B., Teger-Nilsson A. C., Gyzander E., Szelke M. Proceedings of the Thirteenth American Peptide Symposium, R. S. Hodges, J. A. Smith. Escom, Leiden 1994, In Press
  • Di Maio J., Ni E, Gibbs B., Konishi Y. FEBS Lett. 1991; 282: 282
  • Cheng L., Goodwin C. A., Scully M. F., Kakkar V. V., Claeson G. J. Med. Chem. 1992; 35: 35
  • Jim R. T.S. J. Lab. Clin. Med. 1957; 50: 50
  • Lewis J. H., Didisheim P. Arch. Internal Med. (Chicago) 1957; 100: 157
  • Bajusz S., Szell E., Bagdy D., Barabas E., Horvath G., Dioszegi M., Fittler Z., Szabo G., Juhasz A., Tomori E., Szilagyi G. J. Med. Chem. 1990; 33: 33
  • McMurray J. S., Dyckes D. F. J. Org. Chem. 1985; 50: 50
  • Höfle G., Steglich W., Vorbrüggen H. Angew. Chem. Int. Ed. 1978; 17: 17
  • Bodanszky M., Bodanszky A. The Practice of Peptide Synthesis. Springer-Verlag, Berlin, Heidelberg, New York, Tokyo 1984
  • Chen F. M.F., Kuroda K., Benoiton L. Synthesis 1979; 230
  • Maibaum J., Rich D. H. J. Org. Chem. 1988; 53: 53
  • Thaisrivongs S., Pals D. T., Kati W M., Turner S. R., Thomasco L. M., Watt W. J. Med. Chem. 1986; 29: 29
  • Spaltenstein A., Carpino P. A., Miyake F., Hopkins P. B. J. Org. Chem. 1987; 52: 52
  • Dess D. B., Martin J. C. J. Org. Chem. 1983; 48: 48
  • Kitazume T, Ishikawa N. J. Am. Chem. Soc. 1985; 107: 107
  • Kitazume T., Ishikawa N. Chem. Lett. 1981; 1679
  • Edwards P. D. Tet. Lett. 1992; 33: 33
  • Eckert H., List] M., Ugi I. Angew. Chem. 1978; 90: 90
  • Fukuyama T., Laird A. A., Hotchkiss L. M. Et. Lett. 1985; 26: 26
  • Williams D. R., Klingler F. D., Allen E. E., Lichtenthaler F. W. Et. Lett. 1988; 29: 29
  • Cheung S. T., Benoiton N. L. Can. J. Chem. 1977; 55: 55
  • Burkhart J. P., Peet N. P., Bey P. Tet. Lett. 1988; 29: 29
  • Harada H., Tsuhaki A., Kamijo T, Iizuka K., Kiso Y. Chem. Pharm. Bull. 1989; 37: 37
  • Herranz R., Castro-Pichel J., Vinuesa S., Garcia-Mópez M. T. J. Org. Chem. 1990; 55: 55
  • Fittkau S., Jahreis G. Peptides, K. Bláha, P. Maloñ. Walter de Gruyter, Berlin, New York 1983; 617, 1982
  • Thompson R. C. Biochemistry 1974; 13: 13
  • Di Maio J., Gibbs B., Lefebvre J., Konishi Y., Munn D., Yue S. Y. J. Med. Chem. 1992; 35: 35
  • Gelb M. H., Svaren J. P., Abeles R. H. Biochemistry 1985; 24: 24
  • Mehdi S. Bioop. Chem. 1993; 21: 21
  • Schloss J. V. Accounts Chem. Res. 1988; 21: 21
  • Morrison J. F., Walsh C. T. Advances in Enzymology and Related Areas of Molecular Biology, A. Meister. Wiley, New York 1987; 61: 201
  • Sham H. L., Stein H., Rempel C. A., Cohen J., Plattner J. J. FEBS Lett. 1987; 220: 220
  • Brady K., Abeles R. H. Biochemistry 1990; 29: 29
  • Neises B., Tarnus C. Thromb. Haemost. 1991; 65: 65
  • Guichard G., Briand J. P., Friede M. Peptide Res. 1993; 6: 6
  • Hori H., Yasutake A., Minematsu Y., Powers J. C. Peptides, Structure and Function, C. M. Deber, V. J. Hruby, K. D. Kopple. Pierce Chemical Co, Rockford, Illinois 1985; 819
  • Angelastro M. R., Mehdi S., Burkhart J. P., Peet N. P., Bey P. J. Med. Chem. 1990; 33: 33
  • Peet N. P., Burkhart J. P., Angelastro M. R., Giroux E. L., Mehdi S., Bey P., Kolb M., Neises B., Schirlin D. J. Med Chem. 1990; 33: 33
  • Iwanowicz E. J., Lin J., Roberts D. G.M., Michel I. M., Seiler S. M. Bioorg. Med. Chem. Len. 1992; 2: 2
  • Fusetani N., Matsunaga S. J. Am. Chem. Soc. 1990; 112: 112
  • Hagihara M., Schreiber S. L. J. Am. Chem. Soc. 1992; 114: 114
  • Wipf P., Kim H. J. Org. Chem. 1993; 58: 58
  • Mavanoff B. E., Qiu X., Padmanabhan K P, Tulinsky A., Almond H. R., Jr., Andrade-Gordon P., Grew M. N., Kauffman J. A., Nicolaou K. C., Liu A., Brungs R H., Fusetani N. Proc. Nat. Acad. Sci. USA 1993; 90: 90
  • Fenton II J.W., Ofosu F. A., Brezniak D. V., Hassouna H. I. Hematology/Oncology Clinics of North America: Coagulation Disorders II, Vol.7, J. A. Penner, H. I. Hassouna, 1993; 1107
  • Chesebro J. H., Zoldhelyi P., Badimon L., Fuster V. Throm. Haemost. 1991; 66: 66

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.