References
- Jacobsen D., McMartin K. E. Methanol and ethylene glycol poisonings. Mechanism of toxicity, clinical course, diagnosis and treatment. Med Toxicol 1986; 1: 309–334
- Li T. K., Theorell H. Human liver alcohol dehydrogenase: inhibition by pyrazole and pyrazole analogs. Acta Chem Scand 1969; 23: 892–902
- McMartin K. E., Makar A. B., Martin G., Palese M., Tephly T. R. Methanol poisoning I. The role of formic acid in the development of metabolic acidosis in the monkey and the reversal by 4-methylpyrazole. Biochem Med 1975; 13: 319–333
- McMartin K. E., Hedstrom K. G., Tolf B. R., Östling-Wintzell H., Blomstrand R. Studies on the metabolic interactions between 4-methylpyrazole and methanol using the monkey as an animal model. Arch Biochem Biophys 1980; 199: 606–614
- Clay K. L., Murphy R. C. On the metabolic acidosis of ethylene glycol intoxication. Toxicol Appl Pharmacol 1977; 39: 39–49
- Hardman J. G., Limbird L. E. Goodman and Gilman's The Pharmacological Basis of Therapeutics. McGraw-Hill, New York 1996; 1682–1683
- Pietruszko R. Human liver alcohol dehydrogenase: inhibition of methanol activity by pyrazole, 4-methylpyrazole, 4-hydroxymethylpyrazole and 4-carboxypyrazole. Biochem Pharmacol 1975; 24: 1603–1607
- Blomstrand R., Theorell H. Inhibitory effect on ethanol oxidation in man after administration of 4-methylpyrazole. Life Sri II 1970; 9: 631–640
- Magnusson G., Nyberg J. A., Bodin N. O., Hansson E. Toxicity of pyrazole and 4-methylpyrazole in mice and rats. Expereraia 1972; 28: 1198–1200
- Blomstrand R., Ingemansson S. O., Jensen M., Hedstrom C. G. Normal electroretinogram and no toxicity signs after chronic and acute administration of the alcohol dehydrogenase inhibitor 4-methylpyrazole to the cynomolgus monkey (Macaca Fascicularis) - a possible new treatment of methanol poisoning. Drug Alcohol Depend 1984; 13: 9–20
- Jacobsen D., Sebastian C. S., Blomstrand R., McMartin K. E. 4-Methylpyrazole: a controlled study of safety in healthy human subjects after single, ascending doses. Alcohol Oin Exp Res 1988; 12: 516–522
- Jacobsen D., Sebastian C. S., Barron S. K., Carriere E. W., McMartin K. E. Effects of 4-methylpyrazole, methanol/ethylene glycol antidote, in healthy humans. J Emerg Med 1990; 8: 455–461
- Jacobsen D., Barron S. K., Sebastian C. S., Blomstrand R., McMartin K. E. Non-linear kinetics of 4-methyl-pyrazole in healthy human subjects. Eur J Clin Pharmacol 1989; 37: 599–604
- Jacobsen D., Sebastian C. S., Dies D. F., Breau R. L., Spann E. G., Barron S. K., McMartin K. E. Kinetic interactions between 4-methylpyrazole and ethanol in healthy humans. Alcohol Clin Exp Res 1996, in press
- Baud F. J., Bismuth C., Gamier R., et al. 4-Methylpyrazole may be an alternative to ethanol therapy for ethylene glycol intoxication in man. J Toxicol Oin Toxicol 1986–87; 24: 463–483
- Baud F. J., Galliot M., Astier A., et al. Treatment of ethylene glycol poisoning with intravenous 4-methylpyrazole. New Engl J Med 1988; 319: 97–100
- Harry P., Turcant A., Bouachour G., Houze P., Alquier P., Allain P. Efficacy of 4-methylpyrazole in ethylene glycol poisoning: clinical and toxicokinetic aspects. Hum Exp Toxicol 1994; 13: 61–64
- Jacobsen D., Ovrebo S., Arnesen E., Paus P. N. Pulmonary excretion of methanol in man. Scand J Oin Lab Invest 1983; 43: 377–379
- Jobard E., Harry P., Turcant A., Roy P. M., Allain P. 4-Methylpyrazole and hemodialysis in ethylene glycol poisoning. J Toxicol Oin Toxicol 1996; 34: 373–377