Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 18, Issue 2 (2003)

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Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 18, Issue 2 (2003)

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Research Article

Article
Structure–Activity Relationships of Human Urotensin II and Related Analogues on Rat Aortic Ring Contraction
Patricia Labarrère†David Chatenet†Jérôme Leprince†Céline Marionneau†Gervaise Loirand, Marie-Christine Tonon, Christophe Dubessy, Elizabeth Scalbert, Bruno Pfeiffer, Pierre Renard, Bernard Calas, Pierre Pacaud & Hubert Vaudry
Pages: 77-88
Published online: 03 Oct 2008
AbstractforStructure–Activity Relationships of Human Urotensin II and Related Analogues on Rat Aortic Ring Contraction | References | PDF (349.1 KB)
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Article
New Analogues of the Anticancer E7070: Synthesis and Pharmacology
G. Laconde, N. Pommery, P. Depreux, P. Berthelot & J.-P. Hénichart
Pages: 89-94
Published online: 03 Oct 2008
AbstractforNew Analogues of the Anticancer E7070: Synthesis and Pharmacology | References | PDF (169.7 KB)
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Article
Design, Synthesis and Pharmacological Evaluation of New Anticancer Fused Pentacycles
Sarah Chackal, Raymond Houssin, Nicole Pommery & Jean-Pierre Henichart
Pages: 95-99
Published online: 03 Oct 2008
AbstractforDesign, Synthesis and Pharmacological Evaluation of New Anticancer Fused Pentacycles | References | PDF (152.2 KB)
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Article
Indolizino[1,2-b]quinolines Derived from A–D Rings of Camptothecin: Synthesis and DNA Interaction
Aurore Perzyna, Raymond Houssin, Jean-François Goossens, Nicole Pommery, Carine Marty, Michael Facompré, Pierre Colson, Claude Houssier, Christian Bailly & Jean-Pierre Hénichart
Pages: 101-109
Published online: 03 Oct 2008
AbstractforIndolizino[1,2-b]quinolines Derived from A–D Rings of Camptothecin: Synthesis and DNA Interaction | References | PDF (406.4 KB)
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Article
New Ursolic and Betulinic Derivatives as Potential Cytotoxic Agents
I. Baglin, A. Poumaroux, M. Nour, K. Tan, A.C. Mitaine-Offer, M.A. Lacaille-Dubois, B. Chauffert & C. Cavé
Pages: 111-117
Published online: 03 Oct 2008
AbstractforNew Ursolic and Betulinic Derivatives as Potential Cytotoxic Agents | References | PDF (207.9 KB)
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Article
Design, Synthesis and In Vitro Evaluation of Novel Benzo[b]thiophene Derivatives as Serotonin N-acetyltransferase (AANAT) Inhibitors
C. Mesangeau, S. Yous, P. Chavatte, G. Ferry, V. Audinot, J.A. Boutin, P. Delagrange, C. Bennejean, P. Renard & D. Lesieur
Pages: 119-125
Published online: 03 Oct 2008
AbstractforDesign, Synthesis and In Vitro Evaluation of Novel Benzo[b]thiophene Derivatives as Serotonin N-acetyltransferase (AANAT) Inhibitors | References | PDF (189.9 KB)
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Article
Synthesis and Pharmacological Study of Rho-Kinase Inhibitors: Pharmacomodulations on the Lead Compound Fasudil
Cédric Logé, Xavier Siomboing, Valérie Wallez, Elizabeth Scalbert, Caroline Bennejean, Christelle Cario-Tourmaniantz, Gervaise Loirand, Bernard Gressier, Pierre Pacaud & Michel Luyckx
Pages: 127-138
Published online: 03 Oct 2008
AbstractforSynthesis and Pharmacological Study of Rho-Kinase Inhibitors: Pharmacomodulations on the Lead Compound Fasudil | References | PDF (296.7 KB)
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Article
Synthesis and Anti-histaminic Evaluation of N-Phenyl-(alkyl)-5-(dialkylamino)methyl-2-amino-2-oxazolines
J.J. Bosc, F. Pourageaud, P.O. Girodet, M. Molimard & C. Jarry
Pages: 139-145
Published online: 03 Oct 2008
AbstractforSynthesis and Anti-histaminic Evaluation of N-Phenyl-(alkyl)-5-(dialkylamino)methyl-2-amino-2-oxazolines | References | PDF (133.2 KB)
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Article
Synthesis and Initial Results for MAO-B Inhibition by New N-Propargyl-3-pyrrol-1-ylindanamine Derivatives, Analogues of Rasagiline
Jean Guillon, Guillaume Hébert, Patrick Dallemagne, Jean-Michel Léger, Céline Vidaillac, Corinne Thé, Vincent Lisowski, Sylvain Rault, Jacques Demotes-Mainard & Christian Jarry
Pages: 147-153
Published online: 03 Oct 2008
AbstractforSynthesis and Initial Results for MAO-B Inhibition by New N-Propargyl-3-pyrrol-1-ylindanamine Derivatives, Analogues of Rasagiline | References | PDF (239.1 KB)
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Article
Retinoic Acid Metabolism Inhibition by 3-Azolylmethyl-1H-indoles and 2, 3 or 5-(α-Azolylbenzyl)-1H-indoles
Marc Le Borgne, Pascal Marchand, Guillaume Le Baut, Masoud Ahmadi, H. John Smith & Paul J. Nicholls
Pages: 155-158
Published online: 03 Oct 2008
AbstractforRetinoic Acid Metabolism Inhibition by 3-Azolylmethyl-1H-indoles and 2, 3 or 5-(α-Azolylbenzyl)-1H-indoles | References | PDF (134.7 KB)
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Article
Synthesis and Cytotoxic Activity Against a Non-small-cell Bronchopulmonary Carcinoma Line (NSCLC-N6) of Benzofuran Enantiomeric Derivatives
J.J. Hélesbeux, O. Duval, D. Séraphin, C. Roussakis & P. Richomme
Pages: 159-165
Published online: 03 Oct 2008
AbstractforSynthesis and Cytotoxic Activity Against a Non-small-cell Bronchopulmonary Carcinoma Line (NSCLC-N6) of Benzofuran Enantiomeric Derivatives | References | PDF (200.8 KB)
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Article
Synthesis and Cytotoxic Evaluation of Novel Thiazolocarbazoles. Part II1
Hadjila Chabane, Christelle Lamazzi, Valerie Thiery, Alain Pierre, Stephane Leonce, Bruno Pfeiffer, Pierre Renard, Gérald Guillaumet & Thierry Besson
Pages: 167-174
Published online: 03 Oct 2008
AbstractforSynthesis and Cytotoxic Evaluation of Novel Thiazolocarbazoles. Part II1 | References | PDF (241.4 KB)
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Article
Synthesis and Anti-HIV Activity of Some Heterodimers [NRTI]-Glycyl-Succinyl-[Trovirdine Analogue] of Known HIV-1 Reverse Transcriptase Inhibitors
Elena Sugeac, Christine Fossey, Daniel Ladurée, Sylvie Schmidt, Geraldine Laumond & Anne-marie Aubertin
Pages: 175-186
Published online: 03 Oct 2008
AbstractforSynthesis and Anti-HIV Activity of Some Heterodimers [NRTI]-Glycyl-Succinyl-[Trovirdine Analogue] of Known HIV-1 Reverse Transcriptase Inhibitors | References | PDF (315.6 KB)
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Article
Synthesis of 5-Substituted-2,3-dihydro-1,4-benzoxathiins: Biological Evaluation as Melatonin Receptors Ligands
Isabelle Charton, Franck Suzenet, Jean A. Boutin, Valérie Audinot, Philippe Delagrange, Caroline Bennejean, Pierre Renard & Gérald Guillaumet
Pages: 187-193
Published online: 03 Oct 2008
AbstractforSynthesis of 5-Substituted-2,3-dihydro-1,4-benzoxathiins: Biological Evaluation as Melatonin Receptors Ligands | References | PDF (174.7 KB)
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Article
Synthesis, Pharmacological Study and Modeling of 7-Methoxyindazole and Related Substituted Indazoles as Neuronal Nitric Oxide Synthase Inhibitors
Valérie Collot, Jana Sopkova-de Oliveira Santos, Pascale Schumann-Bard, Nathalie Colloc'h, Eric T. MacKenzie & Sylvain Rault
Pages: 195-199
Published online: 03 Oct 2008
AbstractforSynthesis, Pharmacological Study and Modeling of 7-Methoxyindazole and Related Substituted Indazoles as Neuronal Nitric Oxide Synthase Inhibitors | References | PDF (169.3 KB)
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Article
New N-Pyridinyl(methyl)-N1-substituted-3-indolepropanamides Acting as Topical and Systemic Anti-inflammatory Agents
Anthony Gallard, Muriel Duflos, Marie-Renee Nourrisson, Guillaume Le Baut, Nicole Grimaud & Jean Yves Petit
Pages: 201-208
Published online: 03 Oct 2008
AbstractforNew N-Pyridinyl(methyl)-N1-substituted-3-indolepropanamides Acting as Topical and Systemic Anti-inflammatory Agents | References | PDF (203.5 KB)
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