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Synthetic Communications
An International Journal for Rapid Communication of Synthetic Organic Chemistry
Volume 36, 2006 - Issue 2
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Original Articles

New Synthesis of Donepezil Through Palladium‐Catalyzed Hydrogenation Approach

Chandrashekar R. Elati Department of Research and Development, Dr. Reddy's Laboratories Ltd., Hyderabad, Andhra Pradesh, India
,
Naveenkumar Kolla Department of Research and Development, Dr. Reddy's Laboratories Ltd., Hyderabad, Andhra Pradesh, India
,
Subrahmanyeswara Rao Chalamala Department of Research and Development, Dr. Reddy's Laboratories Ltd., Hyderabad, Andhra Pradesh, India
,
Pravinchandra J. Vankawala Department of Research and Development, Dr. Reddy's Laboratories Ltd., Hyderabad, Andhra Pradesh, India
,
Venkataraman Sundaram Department of Research and Development, Dr. Reddy's Laboratories Ltd., Hyderabad, Andhra Pradesh, India
,
Himabindu Vurimidi Institute of Science and Technology, J. N. T. University, Hyderabad, Andhra Pradesh, India
&
Vijayavitthal T. Mathad Department of Research and Development, Dr. Reddy's Laboratories Ltd., Hyderabad, Andhra Pradesh, IndiaCorrespondence[email protected]
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Pages 169-174 | Received 11 Jul 2005, Published online: 15 Aug 2006

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Keshvar Rahimpour, Roghaye Nikbakht, Alireza Aghaiepour & Reza Teimuri-Mofrad. (2018) Synthesis of 2-(4-amino substituted benzylidene) indanone analogues from aromatic nucleophilic substitution (SNAr) reaction. Synthetic Communications 48:17, pages 2253-2259.
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R. Janaki Rama Rao, A.K. S. Bhujanga Rao & Y.L. N. Murthy. (2007) Efficient and Industrially Viable Synthesis of Donepezil. Synthetic Communications 37:17, pages 2847-2853.
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Articles from other publishers (30)

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James T. BrewsterIIII, Simone Dell’Acqua, Danny Q. Thach & Jonathan L. Sessler. (2018) Classics in Chemical Neuroscience: Donepezil. ACS Chemical Neuroscience 10:1, pages 155-167.
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Reza Teimuri-Mofrad, Roghaye Nikbakht & Mahdi Gholamhosseini-Nazari. (2016) A convenient and efficient method for the synthesis of new 2-(4-amino substituted benzilidine) indanone derivatives. Research on Chemical Intermediates 42:10, pages 7501-7511.
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Christoph Schlepphorst, Biplab Maji & Frank Glorius. (2016) Ruthenium-NHC Catalyzed α-Alkylation of Methylene Ketones Provides Branched Products through Borrowing Hydrogen Strategy. ACS Catalysis 6:7, pages 4184-4188.
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Shailendra Kumar Dubey, Manita Kharbanda, Sushil Kumar Dubey & Chandra Shekhar Mathela. (2010) A New Commercially Viable Synthetic Route for Donepezil Hydrochloride: Anti-Alzheimer's Drug. Chemical and Pharmaceutical Bulletin 58:9, pages 1157-1160.
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Navanath Niphade, Anil Mali, Kunal Jagtap, Ramesh Chandra Ojha, Pravinchandra J. Vankawala & Vijayavitthal T. Mathad. (2008) An Improved and Efficient Process for the Production of Donepezil Hydrochloride: Substitution of Sodium Hydroxide for n -Butyl Lithium via Phase Transfer Catalysis . Organic Process Research & Development 12:4, pages 731-735.
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Pelayo CampsXavier FormosaCarles GaldeanoTània GómezDiego Muñoz-TorreroMichele ScarpelliniElisabet ViaynaAlbert BadiaM. Victòria ClosAntoni CaminsMercè PallàsManuela BartoliniFrancesca ManciniVincenza AndrisanoJoan EstelrichMònica LizondoAxel Bidon-ChanalF. Javier Luque. (2008) Novel Donepezil-Based Inhibitors of Acetyl- and Butyrylcholinesterase and Acetylcholinesterase-Induced β-Amyloid Aggregation. Journal of Medicinal Chemistry 51:12, pages 3588-3598.
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Chandrashekar R. Elati, Naveenkumar Kolla, Subrahmanyeswara Rao Chalamala, Pravinchandra J. Vankawala, Venkataraman Sundaram, Himabindu Vurimidi & Vijayavittahl T. Mathad. (2006) New Synthesis of Donepezil Through Palladium‐Catalyzed Hydrogenation Approach.. ChemInform 37:22.
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saikh wabaidur, Saraswati Patel, Sonika Jain, Ritika Gururani, Jaya Dwivedi, Seikh Mohammad wabaidur & Swapnil Sharma. (2021) Insights on Greener Synthetic Strategies and Structure-Activity Relationship of Donepezil and its Derivatives. SSRN Electronic Journal.
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