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Synthetic Communications
An International Journal for Rapid Communication of Synthetic Organic Chemistry
Volume 50, 2020 - Issue 1
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ARTICLE

Synthesis and molecular docking of some new bis-thiadiazoles as anti-hypertensive α-blocking agents

Waleed A. M. A. El-EnanyDepartment of Chemistry, Faculty of Science, University of Cairo, Giza, Egypt;
,
Sobhi M. GomhaDepartment of Chemistry, Faculty of Science, University of Cairo, Giza, Egypt; ;Department of Chemistry, Faculty of Science, Islamic University in Almadinah Almonawara, Almadinah Almonawara, Saudi Arabia; Correspondence[email protected]
ORCID Iconhttp://orcid.org/0000-0001-6744-7817
ORCID Icon,
Ahmed K El-ZiatyChemistry Department, Faculty of Science, Ain Shams University, Cairo, Egypt;
,
Wesam HusseinDepartment of Chemistry, Faculty of Science, Islamic University in Almadinah Almonawara, Almadinah Almonawara, Saudi Arabia;
,
Mohamed M. AbdullaAtosPharma, Elkatyba Land, Belbis, ElSharkya, Egypt;
,
Shaimaa A. HassanDepartment of Chemistry, Faculty of Science, University of Cairo, Giza, Egypt;
,
Hanan A. SallamChemistry Department, Faculty of Science, Ain Shams University, Cairo, Egypt;
&
Rania S. AliDepartment of Basic Science, Faculty of Industrial Education, Helwane University, Cairo, Egypt
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Pages 85-96 | Received 23 Aug 2019, Published online: 31 Oct 2019

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Sapan Shah, Dinesh Chaple, Vijay H. Masand, Magdi E.A Zaki, Sami A. Al-Hussain, Ashish Shah, Sumit Arora, Rahul Jawarkar & Mohammad Tauqeer. (2023) In silico study to recognize novel angiotensin-converting-enzyme-I inhibitors by 2D-QSAR and constraint-based molecular simulations. Journal of Biomolecular Structure and Dynamics 0:0, pages 1-20.
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Mahmoud F. Ismail, Hassan M. F. Madkour, Marwa S. Salem, Ali M. M. Mohamed & Aly Fahmy Aly. (2021) Design, synthesis and insecticidal activity of new 1,3,4-thiadiazole and 1,3,4-thiadiazolo[3,2-a]pyrimidine derivatives under solvent-free conditions. Synthetic Communications 51:17, pages 2644-2660.
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Sayed K. Ramadan, Ahmed K. El-Ziaty & Eman A. E. El-Helw. (2021) Synthesis and antioxidant evaluation of some heterocyclic candidates from 3-(1,3-diphenyl-1H-pyrazol-4-yl)-2-(4-oxo-4H-benzo[d][1,3]oxazin-2-yl)propenonitrile. Synthetic Communications 51:8, pages 1272-1283.
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Samir Bondock, Tallah Albarqi & Mohamed Abboud. (2021) Advances in the synthesis and chemical transformations of 5-acetyl-1,3,4-thiadiazolines. Journal of Sulfur Chemistry 42:2, pages 202-240.
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Articles from other publishers (11)

Sobhi M. Gomha, Sayed M. Riyadh, Magda H. Abdellattif, Tariq Z. Abolibda, Hassan M. Abdel-aziz, AbdElAziz. A. Nayl, Alaa M. Elgohary & Abdo A. Elfiky. (2022) Synthesis and In Silico Study of Some New bis-[1,3,4]thiadiazolimines and bis-Thiazolimines as Potential Inhibitors for SARS-CoV-2 Main Protease. Current Issues in Molecular Biology 44:10, pages 4540-4556.
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Tushar S. Basu Baul, Maheswara Rao Addepalli, Bietlaichhai Hlychho, Antonin Lyčka, Praseeda Vamadevan, Shashank Saurav, Sunil K. Manna & M. Fátima C. Guedes da Silva. (2022) O,N,S-tris-chelating ligand scaffolds flanked with cyclohexyl or adamantyl substituents anchored with diorganotin(IV) moieties: synthesis, structures and cytotoxicity. Inorganica Chimica Acta 537, pages 120935.
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S. Ramakrishna Reddy, G. Ganga Reddy, Ch. Venkata Ramana Reddy & E. Laxminarayana. (2022) Synthesis, Characterization, and Molecular Docking Study of N-[4-(1H-Benzimidazol-2-yl)-1,3-thiazol-2-yl]-1-[(E)-phenyldiazenyl)-1-phenylmethanimines. Russian Journal of Organic Chemistry 58:6, pages 858-864.
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S. Abu-Melha, M. M. Edrees, N. A. Kheder, A. M. Saad, S. M. Riyadh, M. M. Abdel-Aziz, M. A. Abdelmoaz & S. M. Gomha. (2022) Synthesis and Anti-Tubercular (Tb) Evaluation of Bis[4-Ethylidineamino[1,2,4]Triazole-3-Thiol] Tethered by 1,4-Dihydropyridine. Russian Journal of Bioorganic Chemistry 48:2, pages 345-352.
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Şükriye Çakmak, Başak Koşar Kırca, Aysel Veyisoğlu, Hasan Yakan, Cem Cüneyt Ersanlı & Halil Kütük. (2022) Experimental and theoretical investigations on a furan-2-carboxamide-bearing thiazole: synthesis, molecular characterization by IR/NMR/XRD, electronic characterization by DFT, Hirshfeld surface analysis and biological activity. Acta Crystallographica Section C Structural Chemistry 78:3, pages 201-211.
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Asmaa Aboelnaga, Eman Mansour, Asmaa M Fahim & Ghada H. Elsayed. (2022) Synthesis, anti-proliferative activity, gene expression, docking and DFT investigation of novel pyrazol-1-yl-thiazol-4(5H)-one derivatives. Journal of Molecular Structure 1251, pages 131945.
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Syeda Uroos Qazi, Asia Naz, Aqeel Imran & Jamshed Iqbal. (2022) Urease inhibitory kinetics, molecular docking, SAR and ADME studies of imine analogues. New Journal of Chemistry 46:7, pages 3512-3520.
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Emranul Kabir & Monir Uzzaman. (2022) A review on biological and medicinal impact of heterocyclic compounds. Results in Chemistry 4, pages 100606.
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Syeda Uroos Qazi, Asia Naz, Abdul Hameed, Faisal Abdulrhman Osra, Saquib Jalil, Jamshed Iqbal, Syed Adnan Ali Shah & Agha Zeeshan Mirza. (2021) Semicarbazones, thiosemicarbazone, thiazole and oxazole analogues as monoamine oxidase inhibitors: Synthesis, characterization, biological evaluation, molecular docking, and kinetic studies. Bioorganic Chemistry 115, pages 105209.
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Prachi T. Acharya, Zeel A. Bhavsar, Divya J. Jethava, Dhaval B. Patel & Hitesh D. Patel. (2021) A review on development of bio-active thiosemicarbazide derivatives: Recent advances. Journal of Molecular Structure 1226, pages 129268.
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Begüm Nurpelin Sağlık, Betül Kaya Çavuşoğlu, Ulviye Acar Çevik, Derya Osmaniye, Serkan Levent, Yusuf Özkay & Zafer Asım Kaplancıklı. (2020) Novel 1,3,4-thiadiazole compounds as potential MAO-A inhibitors – design, synthesis, biological evaluation and molecular modelling. RSC Medicinal Chemistry 11:9, pages 1063-1074.
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