Advanced search
Publication Cover
Synthetic Communications
An International Journal for Rapid Communication of Synthetic Organic Chemistry
Volume 26, 1996 - Issue 20
Submit an article Journal homepage
72
Views
32
CrossRef citations to date
0
Altmetric
Original Articles

Synthesis and Application of Some New Thienopyrimidine Derivatives as Antimicrobial Agents

Z.A. Hozien Department of Chemistry, Faculty of Science, Assiut University, Assiut, Egypt
,
F.M. Atta Department of Chemistry, Faculty of Science, Assiut University, Assiut, Egypt
,
Kh.M. Hassan Department of Chemistry, Faculty of Science, Assiut University, Assiut, Egypt
,
A.A. Abdel-Wahab Department of Chemistry, Faculty of Science, Assiut University, Assiut, Egypt
&
S.A. Ahmed Department of Chemistry, Faculty of Science, Assiut University, Assiut, Egypt
Pages 3733-3755 | Received 15 Apr 1996, Published online: 21 Aug 2006

Citations (32)

Keep up to date with the latest research on this topic with citation updates for this article.

Subscribe to citation updates

Read on this site (9)

Ahmed F. Saber, Mostafa Sayed, Mahmoud S. Tolba, Adel M. Kamal El-Dean, Reda Hassanien & Mostafa Ahmed. (2021) A facile method for preparation and evaluation of the antimicrobial efficiency of various heterocycles containing thieno[2,3-d]pyrimidine. Synthetic Communications 51:3, pages 398-409.
Read now
Refaah A. Alshahrani, Adil A. Gobouri, Naif A. Alshanbari, Saleh A. Ahmed & Shams H. Abdel-Hafez. (2018) Synthesis of some new pyrimidine selanyl derivatives. Phosphorus, Sulfur, and Silicon and the Related Elements 193:6, pages 345-349.
Read now
RamakrishnaV. S. Nirogi, Rama Sastri Kambhampati, Prabhakar Kothmirkar, Sobhanadri Arepalli, Narasimha ReddyG. Pamuleti, AnilK. Shinde & P.K. Dubey. (2011) Convenient and Efficient Synthesis of Some Novel Fused Thieno Pyrimidines Using Gewald's Reaction. Synthetic Communications 41:19, pages 2835-2851.
Read now
Yong Sun, Nian-Yu Huang & Ming-Wu Ding. (2010) Efficient Synthesis of 6-(1H-1,2,4-Triazol-1-yl)-thieno[2,3-d]pyrimidin-4(3H)-ones via an Iminophosphorane. Synthetic Communications 40:13, pages 1985-1991.
Read now
Xiao-Hua Zeng, Min Liu, Ming-Wu Ding & Hong-Wu He. (2010) Facile Synthesis of 2-Alkylthio-5,6,7,8-tetrahydrobenzothieno[2,3-d]pyrimidin-4(3H)-ones. Synthetic Communications 40:10, pages 1453-1460.
Read now
A.A. Amer, O.A. Omran & A. Khodairy. (2009) Utility of Hydrazinopiperidinomethanethione in Synthesis of Thiadiazole, Thiadiazine, and Pyrazole Derivatives. Phosphorus, Sulfur, and Silicon and the Related Elements 184:7, pages 1653-1664.
Read now
Amer Anwar Amer. (2008) Synthesis and Reactions of Some New Thiazolylpyrazole Derivatives and Related Compounds. Phosphorus, Sulfur, and Silicon and the Related Elements 183:9, pages 2330-2343.
Read now
M.E. Azab, H.M. F. Madkour & M.A. E. Ibraheem. (2006) The Utility of 2-(5,6,7,8-Tetrahydrobenzo[b]thieno-[2,3-d]pyrimidin-4-yloxy) Acethydrazide in Heterocyclic Synthesis. Phosphorus, Sulfur, and Silicon and the Related Elements 181:6, pages 1299-1313.
Read now
H. M. Moustafa, A. Khodairy & A. M. M. El-Saghier. (2003) Synthesis of Some New Polyfused Thienothiophenes Part 4: Synthesis of Thienopyrimidine, Thienotriazine, Thienoimidazotriazine, Thienotriazolotriazine, and Thienotetrazolotriazine Derivatives. Phosphorus, Sulfur, and Silicon and the Related Elements 178:6, pages 1211-1224.
Read now

Articles from other publishers (23)

Jiao-dan Wang, Qiao-li Lin, Jun Qiu, Xiao-feng Gou, Cheng-wen Hua, Jun-long Zhao & Bang Chen. (2017) NO2-Fe(III)PcCl@C -catalyzed one-pot synthesis of tetrahydropyridine derivatives. Russian Journal of General Chemistry 87:4, pages 821-828.
Crossref
DipenK Sureja, SandipP Dholakia & KantilalR Vadalia. (2016) Synthesis of some novel pyrazolo[3,4-d] pyrimidin-4(5H)-one derivatives as potential antimicrobial agent. Journal of Pharmacy And Bioallied Sciences 8:4, pages 321.
Crossref
S. Bugge, E. M. Skjønsfjell, F. B. Willumsen, E. Sundby & B. H. Hoff. (2014) Improved and Scalable Preparation of 6-Bromo-4-Chlorothieno[2,3-d]Pyrimidine. Chemistry of Heterocyclic Compounds 50:8, pages 1177-1187.
Crossref
Sobhi M. Gomha & Mohamed G. Badrey. (2013) A Convenient Synthesis of Some New Thiazole and Pyrimidine Derivatives Incorporating a Naphthalene Moiety. Journal of Chemical Research 37:2, pages 86-90.
Crossref
Jiangping Lou, Zhen Liu, Yan Li, Mi Zhou, Zhengxi Zhang, Shu Zheng, Renxiao Wang & Jian Li. (2011) Synthesis and anti-tumor activities of N′-benzylidene-2-(4-oxothieno[2,3-d]pyrimidin-3(4H)-yl)acetohydrazone derivatives. Bioorganic & Medicinal Chemistry Letters 21:22, pages 6662-6666.
Crossref
Takao HoriuchiYasuyuki TakedaNoriyasu HaginoyaMasaki MiyazakiMotoko NagataMayumi KitagawaKouichi AkahaneKouichi Uoto. (2011) Discovery of Novel Thieno[2,3-d]pyrimidin-4-yl Hydrazone-Based Cyclin-Dependent Kinase 4 Inhibitors: Synthesis, Biological Evaluation and Structure-Activity Relationships. Chemical and Pharmaceutical Bulletin 59:8, pages 991-1002.
Crossref
Hoon-Young Son & Yang-Heon Song. (2010) A Convenient Synthesis of New 3,7-Diphenylthieno[3,2-e]bis[1,2,4] triazolo[4,3-a:4',3'-c]pyrimidine Derivatives by Oxidative Cyclization Using Alumina-supported Calcium Hypochlorite. Bulletin of the Korean Chemical Society 31:8, pages 2242-2246.
Crossref
Takao Horiuchi, Motoko Nagata, Mayumi Kitagawa, Kouichi Akahane & Kouichi Uoto. (2009) Discovery of novel thieno[2,3-d]pyrimidin-4-yl hydrazone-based inhibitors of Cyclin D1-CDK4: Synthesis, biological evaluation and structure–activity relationships. Part 2. Bioorganic & Medicinal Chemistry 17:23, pages 7850-7860.
Crossref
Sheng‐Zhen Xu, Min‐Hui Cao, Chang‐Shui Chen & Ming‐Wu Ding. (2009) Efficient synthesis of benzothieno[3,2‐ d ]‐1,2,4‐triazolo [1,5‐ a ]pyrimidin‐5(1 H )‐ones via a tandem aza‐Wittig/heterocumulene‐mediated annulation . Journal of Heterocyclic Chemistry 46:5, pages 903-908.
Crossref
Takao Horiuchi, Jun Chiba, Kouichi Uoto & Tsunehiko Soga. (2009) Discovery of novel thieno[2,3-d]pyrimidin-4-yl hydrazone-based inhibitors of Cyclin D1-CDK4: Synthesis, biological evaluation, and structure–activity relationships. Bioorganic & Medicinal Chemistry Letters 19:2, pages 305-308.
Crossref
T.J. Delia. 2008. Comprehensive Heterocyclic Chemistry III. Comprehensive Heterocyclic Chemistry III 339 430 .
Gerardo Blanco, José M. Quintela & Carlos Peinador. (2007) Efficient one-pot preparation of bis(pyrazino[2′,3′:4,5]thieno[3,2-d]pyrimidin-4-yl)benzenes based on an aza–Wittig/mediated annulation strategy. Tetrahedron 63:9, pages 2034-2041.
Crossref
Aymn E. Rashad, Mosaad S. Mohamed, Magdy E. A. Zaki & Samar S. Fatahala. (2006) Synthesis and Biological Evaluation of Some Pyrrolo[2,3‐ d ]pyrimidines . Archiv der Pharmazie 339:12, pages 664-669.
Crossref
Balasubramanian Narasimhan, Meena Kumari, Nitin Jain, Avinash Dhake & Chandrasekaran Sundaravelan. (2006) Correlation of antibacterial activity of some N-[5-(2-furanyl)-2-methyl-4-oxo-4H-thieno[2,3-d]pyrimidin-3-yl]-carboxamide and 3-substituted-5-(2-furanyl)-2-methyl-3H-thieno[2,3-d]pyrimidin-4-ones with topological indices using Hansch analysis. Bioorganic & Medicinal Chemistry Letters 16:18, pages 4951-4958.
Crossref
Shu‐Sheng Zhang, Bo Yang, Hui‐Xiang Li & Kui Jiao. (2005) Facile Synthesis and Characterization of Bioactive N ‐[(1‐Ferrocenylethylidene)amino]‐ N ′ ‐ β ‐ D ‐glycopyranosylthiourea . Chinese Journal of Chemistry 23:9, pages 1253-1256.
Crossref
Yong Sun, Sheng-Zhen Xu & Ming-Wu Ding. (2005) A RAPID PARALLEL SYNTHESIS OF 2-DIALKYLAMINO-5,6,7,8-TETRAHYDRO-BENZOTHIENO[2,3-d]PYRIMIDIN-4(3H)-ONES. Heterocyclic Communications 11:5.
Crossref
B. Dietrich. 2005. Comprehensive Organic Functional Group Transformations II. Comprehensive Organic Functional Group Transformations II 725 798 .
A. E. Rashad, O. A. Heikal, A. O. H. El-Nezhawy & F. M. E. Abdel-Megeid. (2005) Synthesis and isomerization of thienotriazolopyrimidine and thienotetrazolopyrimidine derivatives with potential anti-inflammatory activity. Heteroatom Chemistry 16:3, pages 226-234.
Crossref
Salo Gronowitz & Anna-Britta Hörnfeldt. 2004. Thiophenes. Thiophenes 463 557 .
Wagnat W. Wardakhan & Daisy H. Fleita. (2002) Uses of 2‐diazo‐4,5,6,7‐tetrahydrobenzo[ b ]thiophene derivatives in the synthesis of azoles, azines, and their fused derivatives . Heteroatom Chemistry 13:2, pages 108-115.
Crossref
Rafat M. Mohareb & Mona H. Mohamed. (2001) Reaction of 2‐amino‐3‐cyano‐4,5,6,7‐tetrahydrobenzo‐[ b ]thiophene with ethyl acetoacetate: Novel syntheses of pyridines, pyrazoles, and their fused derivatives . Heteroatom Chemistry 12:6, pages 518-527.
Crossref
O.A Abd Allah. (2000) Synthesis and biological studies of some benzopyrano[2,3-c]pyrazole derivatives. Il Farmaco 55:9-10, pages 641-649.
Crossref
Z. A. HOZIEN, F. M. ATTA, KH. M. HASSAN, A. A. ABDEL‐WAHAB & S. A. AHMED. (2010) ChemInform Abstract: Synthesis and Application of Some New Thienopyrimidine Derivatives as Antimicrobial Agents.. ChemInform 28:3.
Crossref

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Order Reprints Request Corporate Permissions

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

Request Academic Permissions

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.

Related research

People also read lists articles that other readers of this article have read.

Recommended articles lists articles that we recommend and is powered by our AI driven recommendation engine.

Cited by lists all citing articles based on Crossref citations.
Articles with the Crossref icon will open in a new tab.