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Kei Suzuki, Kazuhiro Taniyama, Takao Aoyama & Yoshiaki Watanabe. (2020) Bergamottin can be used to assess CYP3A-mediated intestinal first-pass metabolism without affecting P-glycoprotein-mediated efflux in rats. Xenobiotica 50:4, pages 401-407.
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David M Stresser, Jialin Mao, Jane R Kenny, Barry C Jones & Kenneth Grime. (2014) Exploring concepts of in vitro time-dependent CYP inhibition assays. Expert Opinion on Drug Metabolism & Toxicology 10:2, pages 157-174.
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Anna-Pia Palmgren, Britt-Marie Fihn, James Bird, Paul Courtney & Ken Grime. (2013) A novel matrix for the short-term storage of cells: utility in drug metabolism and drug transporter studies with rat, dog and human hepatocytes. Xenobiotica 43:6, pages 487-497.
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Yeamin Huh, David E Smith & Meihau Rose Feng. (2011) Interspecies scaling and prediction of human clearance: comparison of small- and macro-molecule drugs. Xenobiotica 41:11, pages 972-987.
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N. Sekiguchi, M. Kato, M. Takada, H. Watanabe, A. Higashida, S. Sakai, M. Ishigai & Y. Aso. (2008) approach for the evaluation of mechanism-based inhibition of cytochrome P450 3A in rats. Xenobiotica 38:4, pages 368-381.
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Robert J Riley, Ken Grime & Richard Weaver. (2007) Time-dependent CYP inhibition. Expert Opinion on Drug Metabolism & Toxicology 3:1, pages 51-66.
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Articles from other publishers (6)
Sofia Chen, Luna Prieto Garcia, Fredrik Bergström, Pär Nordell & Ken Grime. (2017) Intrinsic Clearance Assay Incubational Binding: A Method Comparison. Drug Metabolism and Disposition 45:4, pages 342-345.
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Pär Nordell, Petter Svanberg, James Bird & Ken Grime. (2013) Predicting Metabolic Clearance for Drugs That Are Actively Transported into Hepatocytes: Incubational Binding as a Consequence of in Vitro Hepatocyte Concentration Is a Key Factor. Drug Metabolism and Disposition 41:4, pages 836-843.
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Jane R. Kenny, Dermot F. McGinnity, Ken Grime & Robert J. Riley. 2010. Pharmaceutical Sciences Encyclopedia. Pharmaceutical Sciences Encyclopedia
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Kenneth H. Grime, James Bird, Douglas Ferguson & Robert J. Riley. (2009) Mechanism-based inhibition of cytochrome P450 enzymes: An evaluation of early decision making in vitro approaches and drug–drug interaction prediction methods. European Journal of Pharmaceutical Sciences 36:2-3, pages 175-191.
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A. P. Rupenko, O. V. Kruglik & I. I. Morgulis. (2008) Functional activity of isolated perfused rat liver depends on medium composition. Bulletin of Experimental Biology and Medicine 146:1, pages 107-110.
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A. P. Rupenko, O. V. Kruglik & I. I. Morgulis. (2011) Oxygen supply of rat liver under the conditions of isolated perfusion. Doklady Biological Sciences 418:1, pages 4-6.
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