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Xenobiotica
the fate of foreign compounds in biological systems
Volume 37, 2007 - Issue 5
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Research Article

Gemfibrozil and its glucuronide inhibit the hepatic uptake of pravastatin mediated by OATP1B1

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Pages 474-486 | Received 12 Jan 2007, Accepted 13 Feb 2007, Published online: 22 Sep 2008

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Mariana Mauro, Jose Salvador Lepera, Bruno Borsari, Jorge Manuel Vieira Capela & Natália Valadares de Moraes. (2018) Effect of inhalation exposure to toluene on the activity of organic anion transporting polypeptide (Oatp) using pravastatin as a probe drug in rats. Xenobiotica 48:7, pages 734-738.
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Aleksi Tornio, Pertti J. Neuvonen, Mikko Niemi & Janne T. Backman. (2017) Role of gemfibrozil as an inhibitor of CYP2C8 and membrane transporters. Expert Opinion on Drug Metabolism & Toxicology 13:1, pages 83-95.
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Fabian Müller & Martin F Fromm. (2011) Transporter-Mediated Drug–Drug Interactions. Pharmacogenomics 12:7, pages 1017-1037.
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Alice C Rodrigues. (2010) Efflux and uptake transporters as determinants of statin response. Expert Opinion on Drug Metabolism & Toxicology 6:5, pages 621-632.
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