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Cheng Hua Jin, Maddeboina Krishnaiah, Domalapally Sreenu, Vura Bala Subrahmanyam, Hyun-Ju Park, So-Jung Park, Yhun Yhong Sheen & Dae-Kee Kim. (2014) 4-([1,2,4]Triazolo[1,5-a]pyridin-6-yl)-5(3)-(6-methylpyridin-2-yl)imidazole and -pyrazole derivatives as potent and selective inhibitors of transforming growth factor-β type I receptor kinase. Bioorganic & Medicinal Chemistry 22:9, pages 2724-2732.
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Adeyemi O. Adedeji, William Severson, Colleen Jonsson, Kamalendra Singh, Susan R. Weiss & Stefan G. Sarafianos. (2013) Novel Inhibitors of Severe Acute Respiratory Syndrome Coronavirus Entry That Act by Three Distinct Mechanisms. Journal of Virology 87:14, pages 8017-8028.
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Xuyu Zu, Qinghai Zhang, Renxian Cao, Jianghua Liu, Jing Zhong, Gebo Wen & Deliang Cao. (2011) Transforming growth factor-β signaling in tumor initiation, progression and therapy in breast cancer: an update. Cell and Tissue Research 347:1, pages 73-84.
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Cheng Hua Jin, Maddeboina Krishnaiah, Domalapally Sreenu, Vura Bala Subrahmanyam, Kota Sudhakar Rao, Annaji Venkata Nagendra Mohan, Chul-Yong Park, Jee-Yeon Son, Yhun Yhong Sheen & Dae-Kee Kim. (2011) Synthesis and biological evaluation of 1-substituted-3-(6-methylpyridin-2-yl)-4-([1,2,4]triazolo[1,5-a]pyridin-6-yl)pyrazoles as transforming growth factor-β type 1 receptor kinase inhibitors. Bioorganic & Medicinal Chemistry Letters 21:20, pages 6049-6053.
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Hyun-Jung Yoon, Ho-Young Song, Jin Hyoung Kim, Kang-Sun Hong, Yeon Joo Kim, Hyung Gyu Park & Dae-Kee Kim. (2011) Role of IN-1233 in the Prevention of Neointimal Hyperplasia after Stent Placement in a Rat Artery Model. Journal of Vascular and Interventional Radiology 22:9, pages 1321-1328.
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Cheng Hua Jin, Domalapally Sreenu, Maddeboina Krishnaiah, Vura Bala Subrahmanyam, Kota Sudhakar Rao, Annaji Venkata Nagendra Mohan, Chul-Yong Park, Jee-Yeon Son, Do-Hyun Son, Hyun-Ju Park, Yhun Yhong Sheen & Dae-Kee Kim. (2011) Synthesis and biological evaluation of 1-substituted-3(5)-(6-methylpyridin-2-yl)-4-(quinoxalin-6-yl)pyrazoles as transforming growth factor-β type 1 receptor kinase inhibitors. European Journal of Medicinal Chemistry 46:9, pages 3917-3925.
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Cheng Hua Jin, Maddeboina Krishnaiah, Domalapally Sreenu, Kota Sudhakar Rao, Vura Bala Subrahmanyam, Chul-Yong Park, Jee-Yeon Son, Yhun Yhong Sheen & Dae-Kee Kim. (2011) Synthesis and biological evaluation of 1-substituted-3(5)-(6-methylpyridin-2-yl)-4-(quinolin-6-yl)pyrazoles as transforming growth factor-β type 1 receptor kinase inhibitors. Bioorganic & Medicinal Chemistry 19:8, pages 2633-2640.
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Purushottam M. Dewang & Dae-Kee Kim. (2010) Synthesis and biological evaluation of 2-pyridyl-substituted pyrazoles and imidazoles as transforming growth factor-β type 1 receptor kinase inhibitors. Bioorganic & Medicinal Chemistry Letters 20:14, pages 4228-4232.
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Jin Hyoung Kim, Ho-Young Song, Jung-Hoon Park, Hyun-Jung Yoon, Hyung Gyu Park & Dae-Kee Kim. (2010) IN-1233, an ALK-5 Inhibitor: Prevention of Granulation Tissue Formation after Bare Metallic Stent Placement in a Rat Urethral Model. Radiology 255:1, pages 75-82.
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Dae-Kee Kim, Sun Hee Jung, Ho Soon Lee & Purushottam M. Dewang. (2009) Synthesis and biological evaluation of benzenesulfonamide-substituted 4-(6-alkylpyridin-2-yl)-5-(quinoxalin-6-yl)imidazoles as transforming growth factor-β type 1 receptor kinase inhibitors. European Journal of Medicinal Chemistry 44:2, pages 568-576.
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Dae-Kee Kim, Jin-Hwi Lim, Jung A. Lee & Purushottam M. Dewang. (2008) Synthesis and biological evaluation of trisubstituted imidazole derivatives as inhibitors of p38α mitogen-activated protein kinase. Bioorganic & Medicinal Chemistry Letters 18:14, pages 4006-4010.
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