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Xenobiotica
the fate of foreign compounds in biological systems
Volume 28, 1998 - Issue 3
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Research Article

Inhibition of human hepatic cytochrome P4502E1 by azole antifungals, CNS-active drugs and nonsteroidal anti-inflammatory agents

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Pages 293-301 | Published online: 22 Sep 2008

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Jae Yong Choi, Chul Hoon Kim, Tae Joo Jeon, Byoung Soo Kim, Chi Hoon Yi, Kwang Sun Woo, Young Beom Seo, Sang Jin Han, Kyeong Min Kim, Dae Ik Yi, Minkyung Lee, Dong Goo Kim, Jung Young Kim, Kyo Chul Lee, Tae Hyun Choi, Gwangil An & Young Hoon Ryu. (2012) Effective MicroPET imaging of brain 5‐HT 1A receptors in rats with [ 18 F]MeFWAY by suppression of radioligand defluorination . Synapse 66:12, pages 1015-1023.
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G Merino, A J Molina, J L García, M M Pulido, J G Prieto & A I Alvarez. (2003) Effect of clotrimazole on microsomal metabolism and pharmacokinetics of albendazole. Journal of Pharmacy and Pharmacology 55:6, pages 757-764.
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Hugues Ouellet, Jonathan B. Johnston & Paul R. Ortiz de Montellano. (2010) The Mycobacterium tuberculosis cytochrome P450 system. Archives of Biochemistry and Biophysics 493:1, pages 82-95.
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J. J. Aaron, M. D. Gaye Seye, S. Trajkovska & N. Motohashi. 2009. Bioactive Heterocycles VII. Bioactive Heterocycles VII 153 231 .
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Robert L. Haining & Mari Nichols-Haining. (2007) Cytochrome P450-catalyzed pathways in human brain: Metabolism meets pharmacology or old drugs with new mechanism of action?. Pharmacology & Therapeutics 113:3, pages 537-545.
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Toshiro NIWAToshifumi SHIRAGAAkira TAKAGI. (2005) Drug-Drug Interaction of Antifungal Drugs抗真菌剤の薬物相互作用—薬物代謝酵素に及ぼす影響—. YAKUGAKU ZASSHI 125:10, pages 795-805.
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Christian Wolff, Michel Gillard, Bruno Fuks & Pierre Chatelain. (2005) [3H]linopirdine binding to rat brain membranes is not relevant for M-channel interaction. European Journal of Pharmacology 518:1, pages 10-17.
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Toshiro NiwaSachiko Inoue-YamamotoToshifumi ShiragaAkira Takagi. (2005) Effect of Antifungal Drugs on Cytochrome P450 (CYP) 1A2, CYP2D6, and CYP2E1 Activities in Human Liver Microsomes. Biological and Pharmaceutical Bulletin 28:9, pages 1813-1816.
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Katalin Monostory, Eszter Hazai & László Vereczkey. (2004) Inhibition of cytochrome P450 enzymes participating in p-nitrophenol hydroxylation by drugs known as CYP2E1 inhibitors. Chemico-Biological Interactions 147:3, pages 331-340.
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David E. Moody. 2004. Handbook of Drug Interactions. Handbook of Drug Interactions 3 88 .
Bryan D. MarksRonald W. SmithHeidi A. BraunTony A. GoossensMarie ChristensonMary S. OzersConnie S. LebakkenOlga V. Trubetskoy. (2002) A High Throughput Screening Assay to Screen for CYP2E1 Metabolism and Inhibition Using a Fluorogenic Vivid ® P450 Substrate . ASSAY and Drug Development Technologies 1:1, pages 73-81.
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Eszter Hazai, László Vereczkey & Katalin Monostory. (2002) Reduction of Toxic Metabolite Formation of Acetaminophen. Biochemical and Biophysical Research Communications 291:4, pages 1089-1094.
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Chin‐Eng Ong, Sally Coulter, Donald J. Birkett, C. Ramana Bhasker & John O. Miners. (2008) The xenobiotic inhibitor profile of cytochrome P4502C8. British Journal of Clinical Pharmacology 50:6, pages 573-580.
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Karthik Venkatakrishnan, Lisa L. von Moltke & David J. Greenblatt. (2000) Effects of the Antifungal Agents on Oxidative Drug Metabolism. Clinical Pharmacokinetics 38:2, pages 111-180.
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