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Research Article

Comparison of a novel spray congealing procedure with emulsion-based methods for the micro-encapsulation of water-soluble drugs in low melting point triglycerides

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Pages 365-378 | Received 15 Aug 2007, Accepted 19 Feb 2008, Published online: 08 Oct 2008

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Read on this site (6)

Hongyi Ouyang, Soon Jun Ang, Zong Yang Lee, Tze Ning Hiew, Paul Wan Sia Heng & Lai Wah Chan. (2022) Effect of drug load and lipid–wax blends on drug release and stability from spray-congealed microparticles. Pharmaceutical Development and Technology 27:10, pages 1069-1082.
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Santo Scalia, Paul M Young & Daniela Traini. (2015) Solid lipid microparticles as an approach to drug delivery. Expert Opinion on Drug Delivery 12:4, pages 583-599.
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Ching Mien Oh, Qiyun Guo, Paul Wan Sia Heng & Lai Wah Chan. (2014) Spray-congealed microparticles for drug delivery – an overview of factors influencing their production and characteristics. Expert Opinion on Drug Delivery 11:7, pages 1047-1060.
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Rodrigo Molina Martins, Silvia Siqueira, Marcela Olaia Machado & Luis Alexandre Pedro Freitas. (2013) The effect of homogenization method on the properties of carbamazepine microparticles prepared by spray congealing. Journal of Microencapsulation 30:7, pages 692-700.
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Santo Scalia, Daniela Traini, Paul M. Young, Marcello Di Sabatino, Nadia Passerini & Beatrice Albertini. (2013) Comparison of spray congealing and melt emulsification methods for the incorporation of the water-soluble salbutamol sulphate in lipid microparticles. Pharmaceutical Development and Technology 18:1, pages 266-273.
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Leena Peltonen, Hanna Valo, Ruzica Kolakovic, Timo Laaksonen & Jouni Hirvonen. (2010) Electrospraying, spray drying and related techniques for production and formulation of drug nanoparticles. Expert Opinion on Drug Delivery 7:6, pages 705-719.
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Articles from other publishers (17)

Hongyi Ouyang, Annabel Shi Yin Poh, Paul Wan Sia Heng & Lai Wah Chan. (2020) Effect of Surfactants on the Melt Viscosity and Extent of Drug Embedment of Paraffin Wax Blends in Spray Congealing. Journal of Pharmaceutical Innovation 17:2, pages 414-428.
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Serena Bertoni, Beatrice Albertini, Joanna Ronowicz-Pilarczyk, Natalia Calonghi & Nadia Passerini. (2021) Solvent-Free Fabrication of Biphasic Lipid-Based Microparticles with Tunable Structure. Pharmaceutics 14:1, pages 54.
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G.D Sorita, A Santamaria-Echart, A.M Gozzo, O.H Gonçalves, F.V Leimann, E Bona, Y Manrique, I.P.M Fernandes, I.C.F.R Ferreira & M.F Barreiro. (2021) Lipid composition optimization in spray congealing technique and testing with curcumin-loaded microparticles. Advanced Powder Technology 32:5, pages 1710-1722.
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Leon Yoon Ho, Zi Shun Xiang, Renuga Gopal & Saif A. Khan. (2021) Microfluidics-enabled particle engineering of monodisperse solid lipid microparticles with uniform drug loading and diverse solid-state outcomes. International Journal of Pharmaceutics 596, pages 120230.
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Kerstin Traub-Hoffmann, Katrin Gegenfurtner, Kay-Uwe Kraft & Wolfgang Friess. (2020) Spray congealed solid lipid microparticles as a sustained release delivery system for Gonadorelin [6-D-Phe]: Production, optimization and in vitro release behavior. European Journal of Pharmaceutics and Biopharmaceutics 154, pages 18-32.
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Hongyi Ouyang, Chen Yee Ang, Paul Wan Sia Heng & Lai Wah Chan. (2019) Effects of Drug Particle Size and Lipid Additives on Drug Release from Paraffin Wax Formulations Prepared by Spray Congealing Technique. AAPS PharmSciTech 20:7.
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Serena Bertoni, Luisa S Dolci, Beatrice Albertini & Nadia Passerini. (2018) Spray congealing: a versatile technology for advanced drug-delivery systems. Therapeutic Delivery 9:11, pages 833-845.
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Hongyi Ouyang, Audrey Zheng, Paul Heng & Lai Chan. (2018) Effect of Lipid Additives and Drug on the Rheological Properties of Molten Paraffin Wax, Degree of Surface Drug Coating, and Drug Release in Spray-Congealed Microparticles. Pharmaceutics 10:3, pages 75.
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O.C. Paucar, F.L. Tulini, M. Thomazini, J.C.C. Balieiro, E.M.J.A. Pallone & C.S. Favaro-Trindade. (2016) Production by spray chilling and characterization of solid lipid microparticles loaded with vitamin D 3. Food and Bioproducts Processing 100, pages 344-350.
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Julice Dutra Lopes, Carlos Raimundo Ferreira Grosso, Guilherme de Andrade Calligaris, Lisandro Pavie Cardoso, Rodrigo Corrêa Basso, Ana Paula Badan Ribeiro & Priscilla Efraim. (2017) Solid lipid microparticles of hardfats produced by spray cooling as promising crystallization modifiers in lipid systems. European Journal of Lipid Science and Technology 117:11, pages 1733-1744.
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Julice Dutra Lopes, Carlos Raimundo Ferreira Grosso, Guilherme de Andrade Calligaris, Lisandro Pavie Cardoso, Rodrigo Corrêa Basso, Ana Paula Badan Ribeiro & Priscilla Efraim. (2015) Solid lipid microparticles of hardfats produced by spray cooling as promising crystallization modifiers in lipid systems. European Journal of Lipid Science and Technology 117:11, pages 1733-1744.
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Darren S. Miller, Anne Michelle Parsons, John Bresland, Paul Herde, Duc Minh Pham, Angel Tan, Hung-yao Hsu, Clive A. Prestidge, Tim Kuchel, Rezaul Begg, Syed Mahfuzul Aziz & Ross N. Butler. (2015) A simple and inexpensive enteric-coated capsule for delivery of acid-labile macromolecules to the small intestine一种用于递送酸度敏感大分子到小肠的简易且廉价的肠溶胶囊. Journal of Zhejiang University-SCIENCE B 16:7, pages 586-592.
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Marcello Di Sabatino, Beatrice Albertini, Vicky L. Kett & Nadia Passerini. (2012) Spray congealed lipid microparticles with high protein loading: Preparation and solid state characterisation. European Journal of Pharmaceutical Sciences 46:5, pages 346-356.
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Nadia Passerini, Sheng Qi, Beatrice Albertini, Mario Grassi, Lorenzo Rodriguez & Duncan Q.M. Craig. (2010) Solid lipid microparticles produced by spray congealing: Influence of the atomizer on microparticle characteristics and mathematical modeling of the drug release. Journal of Pharmaceutical Sciences 99:2, pages 916-931.
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Rasil Al-Kassas, Ryan F Donnelly & Paul A McCarron. (2009) Aminolevulinic acid-loaded Witepsol microparticles manufactured using a spray congealing procedure: implications for topical photodynamic therapy. Journal of Pharmacy and Pharmacology 61:9, pages 1125-1135.
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I. Ilić, R. Dreu, M. Burjak, M. Homar, J. Kerč & S. Srčič. (2009) Microparticle size control and glimepiride microencapsulation using spray congealing technology. International Journal of Pharmaceutics 381:2, pages 176-183.
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Ryan F. Donnelly, Paul A. McCarron, Rasil Al‐Kassas, Asta Juzeniene, Petras Juzenas, Vladimir Iani, A. David Woolfson & Johan Moan. (2009) Influence of formulation factors on PpIX production and photodynamic action of novel ALA‐loaded microparticles. Biopharmaceutics & Drug Disposition 30:2, pages 55-70.
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