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ORIGINAL ARTICLE

Effect of Leuprolide and Cetrorelix on Cell Growth, Apoptosis, and GnRH Receptor Expression in Primary Cell Cultures from Human Prostate Carcinoma

, Ph.D., , M.S.c., , M.D., , V.M.D., , Ph.D., , V.M.D., , Ph.D. & , M.D. show all
Pages 261-268 | Published online: 11 Jun 2009

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Catherine Sánchez, Alejandro Mercado, Héctor R. Contreras, Felipe Carvajal V, Apolo Salgado, Christian Huidobro & Enrique A. Castellón. (2021) Membrane translocation and activation of GnRH receptor sensitize prostate cancer cells to radiation. International Journal of Radiation Biology 97:11, pages 1555-1562.
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Nicola Arrighi, Serena Bodei, Danilo Zani, Claudio Simeone, Sergio Cosciani Cunico, Cristina Missale, Pierfranco Spano & Sandra Sigala. (2010) Nerve growth factor signaling in prostate health and disease. Growth Factors 28:3, pages 191-201.
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Christian Doehn, Martin Sommerauer & Dieter Jocham. (2009) Degarelix and its therapeutic potential in the treatment of prostate cancer. Clinical Interventions in Aging 4, pages 215-223.
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Christian Doehn, Martin Sommerauer & Dieter Jocham. (2009) Degarelix for prostate cancer. Expert Opinion on Investigational Drugs 18:6, pages 851-860.
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R. Elancheran, V. L. Maruthanila, M. Ramanathan, S. Kabilan, R. Devi, A. Kunnumakara & Jibon Kotoky. (2015) Recent discoveries and developments of androgen receptor based therapy for prostate cancer. MedChemComm 6:5, pages 746-768.
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Peter Hammerer & Stephan Madersbacher. (2013) Reply. BJU International 111:3.
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Catherine A. Sánchez, Alejandro J. Mercado, Héctor R. Contreras, Juan C. Cabezas, Christian C. Huidobro & Enrique A. Castellón. (2012) Pharmacoperone IN3 enhances the apoptotic effect of leuprolide in prostate cancer cells by increasing the gonadotropin-releasing hormone receptor in the cell membrane. Anti-Cancer Drugs 23:9, pages 959-969.
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Laurent Boccon-Gibod, Egbert van der Meulen & Bo-Eric Persson. (2011) An update on the use of gonadotropin-releasing hormone antagonists in prostate cancer. Therapeutic Advances in Urology 3:3, pages 127-140.
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Mariela Bilotas, Gabriela Meresman, Ricardo Buquet, Carlos Sueldo & Rosa Inés Barañao. (2010) Effect of vascular endothelial growth factor and interleukin-1β on apoptosis in endometrial cell cultures from patients with endometriosis and controls. Journal of Reproductive Immunology 84:2, pages 193-198.
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Xiang Zou, Chen feng Ji & Yu bin Ji. (2009) Effect of Asparagus Saponins on HepG2 Apoptosis and Mitochondrial Membrane Potential and ROS Level. Effect of Asparagus Saponins on HepG2 Apoptosis and Mitochondrial Membrane Potential and ROS Level.
Catherine Sánchez, Patricia Mendoza, Héctor R. Contreras, Jorge Vergara, James A. McCubrey, Christian Huidobro & Enrique A. Castellón. (2009) Expression of multidrug resistance proteins in prostate cancer is related with cell sensitivity to chemotherapeutic drugs. The Prostate 69:13, pages 1448-1459.
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Cristiana Angelucci, Gina Lama, Fortunata Iacopino, Silvia Ferracuti, Aldo V. Bono, Robert P. Millar & Gigliola Sica. (2009) GnRH receptor expression in human prostate cancer cells is affected by hormones and growth factors. Endocrine 36:1, pages 87-97.
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Marisa Clementi, Catherine Sánchez, Dixan A. Benitez, Héctor R. Contreras, Christian Huidobro, Juan Cabezas, Cristian Acevedo & Enrique A. Castellón. (2009) Gonadotropin releasing hormone analogs induce apoptosis by extrinsic pathway involving p53 phosphorylation in primary cell cultures of human prostatic adenocarcinomas. The Prostate 69:10, pages 1025-1033.
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Dong-Ki Kim, Ji Sook Yang, Kaushik Maiti, Jong-Ik Hwang, Kyungjin Kim, Dongseung Seen, Younghee Ahn, Cheolju Lee, Byeong-Cheol Kang, Hyuk Bang Kwon, Jun Cheon & Jae Young Seong. (2009) A Gonadotropin-Releasing Hormone-II Antagonist Induces Autophagy of Prostate Cancer Cells. Cancer Research 69:3, pages 923-931.
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Wai‐Kin So, Jung‐Chien Cheng, Song‐Ling Poon & Peter C. K. Leung. (2008) Gonadotropin‐releasing hormone and ovarian cancer: a functional and mechanistic overview. The FEBS Journal 275:22, pages 5496-5511.
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Elahe A. Mostaghel, Robert B. Montgomery & Daniel W. Lin. (2008) The basic biochemistry and molecular events of hormone therapy. Current Prostate Reports 6:2, pages 47-55.
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D A Benitez, E Pozo-Guisado, M Clementi, E Castellón & P M Fernandez-Salguero. (2007) Non-genomic action of resveratrol on androgen and oestrogen receptors in prostate cancer: modulation of the phosphoinositide 3-kinase pathway. British Journal of Cancer 96:10, pages 1595-1604.
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Elahe A. Mostaghel, Robert B. Montgomery & Daniel W. Lin. (2007) The basic biochemistry and molecular events of hormone therapy. Current Urology Reports 8:3, pages 224-232.
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