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Journal of Biomolecular Structure and Dynamics Volume 40, 2022 - Issue 18
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Research Articles

Synthesis, α-glucosidase and α-amylase inhibitory activities, acute toxicity and molecular docking studies of thiazolidine-2,4-diones derivatives

Saad Fettacha Laboratory of Pharmacology and Toxicology, Biopharmaceutical and Toxicological Analysis Research Team, Faculty of Medicine and Pharmacy, Mohammed V University in Rabat, Rabat, MoroccoView further author information
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Fatima Zahra Tharib Equipe de Chimie des Plantes et de Synthèse Organique et Bioorganique, URAC23, Faculty of Science, Geophysics, Natural Patrimony and Green Chemistry (GEOPAC) Research Center, Mohammed V University in Rabat, Rabat, MoroccoView further author information
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Zakaria Hafidic Laboratoire de Physico-Chimie des Matériaux Inorganiques et Organiques, Centre des Sciences des Matériaux, Ecole Normale Supérieure-Rabat, Mohammed V University in Rabat, Rabat, MoroccoORCID Iconhttps://orcid.org/0000-0001-8554-5189View further author information
ORCID Icon,
Hamza Tachallaitb Equipe de Chimie des Plantes et de Synthèse Organique et Bioorganique, URAC23, Faculty of Science, Geophysics, Natural Patrimony and Green Chemistry (GEOPAC) Research Center, Mohammed V University in Rabat, Rabat, MoroccoView further author information
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Khalid Karrouchid Laboratory of Analytical Chemistry and Bromatology, Faculty of Medicine and Pharmacy, Mohammed V University in Rabat, Rabat, MoroccoView further author information
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Mohammed El achouric Laboratoire de Physico-Chimie des Matériaux Inorganiques et Organiques, Centre des Sciences des Matériaux, Ecole Normale Supérieure-Rabat, Mohammed V University in Rabat, Rabat, MoroccoView further author information
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Yahia Cherraha Laboratory of Pharmacology and Toxicology, Biopharmaceutical and Toxicological Analysis Research Team, Faculty of Medicine and Pharmacy, Mohammed V University in Rabat, Rabat, MoroccoORCID Iconhttps://orcid.org/0000-0001-7890-9028View further author information
ORCID Icon,
Hassan Sefriouie Moroccan Foundation for Science, Innovation & Research (MAScIR), Centre de Biotechnologie Médicale, Rabat, MoroccoView further author information
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Khalid Bougrinb Equipe de Chimie des Plantes et de Synthèse Organique et Bioorganique, URAC23, Faculty of Science, Geophysics, Natural Patrimony and Green Chemistry (GEOPAC) Research Center, Mohammed V University in Rabat, Rabat, Morocco;f Mohammed VI Polytechnic University, Benguerir, MoroccoCorrespondence[email protected] [email protected]
ORCID Iconhttps://orcid.org/0000-0001-9553-8310View further author information
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My El Abbes Faouzia Laboratory of Pharmacology and Toxicology, Biopharmaceutical and Toxicological Analysis Research Team, Faculty of Medicine and Pharmacy, Mohammed V University in Rabat, Rabat, MoroccoCorrespondence[email protected] [email protected]
ORCID Iconhttps://orcid.org/0000-0003-3863-4677View further author information
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Pages 8340-8351 | Received 19 Dec 2020, Accepted 26 Mar 2021, Published online: 13 Apr 2021

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Khalid Karrouchi, Yusuf Sert, M’hammed Ansar, Smaail Radi, Brahim El Bali, Rehan Imad, Anum Alam, Rimsha Irshad, Sheeba Wajid & Muhammad Altaf. (2023) Synthesis, α-Glucosidase Inhibition, Anticancer, DFT and Molecular Docking Investigations of Pyrazole Hydrazone Derivatives. Polycyclic Aromatic Compounds 43:6, pages 5021-5040.
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Khalid Karrouchi, Saad Fettach, El Hassane Anouar, Imene Bayach, Hanan Albalwi, Suhana Arshad, Nada Kheira Sebbar, Hamza Tachalait, Khalid Bougrin, My El Abbes Faouzi & Benacer Himmi. (2023) Synthesis, Spectroscopic Characterization, DFT, Molecular Docking and Antidiabetic Activity of N-Isonicotinoyl Arylaldehyde Hydrazones. Polycyclic Aromatic Compounds 43:2, pages 1469-1481.
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Yasmine Zine, Adel Krid, Raouf Boulcina, Dominique Harakat, Anthony Robert, Chawki Bensouici & Abdelmadjid Debache. Synthesis, Biological Evaluation, DFT Calculations and Molecular Docking of 5-Arylidene-Thiazolidine-2,4-Dione Derivatives. Polycyclic Aromatic Compounds 0:0, pages 1-24.
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Said Dadou, Ahmet Altay, Cemile Baydere, El Hassane Anouar, Burçin Türkmenoğlu, Mohammed Koudad, Necmi Dege, Abdelouahad Oussaid, Noureddine Benchat & Khalid Karrouchi. Chalcone-based imidazo[2,1-b]thiazole derivatives: synthesis, crystal structure, potent anticancer activity, and computational studies. Journal of Biomolecular Structure and Dynamics 0:0, pages 1-16.
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Dilip C. Kanjariya, Hem N. Naik, Meet J. Sherashiya, Yogesh T. Naliapara, Iqrar Ahmad, Harun Patel, Dhanji Rajani & Smita Jauhari. α-Amylase and mycobacterium-TB H37Rv antagonistic efficacy of novel pyrazole-coumarin hybrids: an in vitro and in silico investigation. Journal of Biomolecular Structure and Dynamics 0:0, pages 1-18.
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Articles from other publishers (7)

Shankar Gupta, Gurkaran Singh Baweja, GD Gupta & Vivek Asati. (2023) Identification of potential N-substituted 5-benzylidenethiazolidine-2,4‑dione derivatives as α-amylase inhibitors: Computational cum synthetic studies. Journal of Molecular Structure 1287, pages 135596.
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Rafik Saddik, Silvia A. Brandán, Salma Mortada, Cemile Baydere, Othmane Roby, Necmi Dege, Said Tighadouini, Mohamed Tahiri, My Abbes Faouzi & Khalid Karrouchi. (2023) Synthesis, crystal structure, Hirshfeld surface analysis, DFT and antihyperglycemic activity of 9-allyl-2,3,9,10a-tetrahydrobenzo[b]cyclopenta[e][1,4]diazepin-10(1H)-one. Journal of Molecular Structure 1283, pages 135283.
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Ayman M. Ibrahim, Mai E. Shoman, Mamdouh F. A. Mohamed, Alaa M. Hayallah & Gamal El‐Din A. Abuo‐Rahma. (2023) Chemistry and Applications of Functionalized 2,4‐Thiazolidinediones. European Journal of Organic Chemistry 26:19.
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Said Daoui, Şahin Direkel, Munjed M. Ibrahim, Burak Tüzün, Tarik Chelfi, Mohammed Al-Ghorbani, Mustapha Bouatia, Miloud El Karbane, Anass Doukkali, Noureddine Benchat & Khalid Karrouchi. (2023) Synthesis, Spectroscopic Characterization, Antibacterial Activity, and Computational Studies of Novel Pyridazinone Derivatives. Molecules 28:2, pages 678.
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Sabbir Ahmed, Md Ali, Rumana Ruma, Shafi Mahmud, Gobindo Paul, Md Saleh, Mohammed Alshahrani, Ahmad Obaidullah, Sudhangshu Biswas, Md Rahman, Md Rahman & Md Islam. (2022) Molecular Docking and Dynamics Simulation of Natural Compounds from Betel Leaves (Piper betle L.) for Investigating the Potential Inhibition of Alpha-Amylase and Alpha-Glucosidase of Type 2 Diabetes. Molecules 27:14, pages 4526.
Crossref
Dominika Mech, Antonina Kurowska & Nazar Trotsko. (2021) The Bioactivity of Thiazolidin-4-Ones: A Short Review of the Most Recent Studies. International Journal of Molecular Sciences 22:21, pages 11533.
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Amani Toumi, Sarra Boudriga, Khaled Hamden, Ismail Daoud, Moheddine Askri, Armand Soldera, Jean-Francois Lohier, Carsten Strohmann, Lukas Brieger & Michael Knorr. (2021) Diversity-Oriented Synthesis of Spiropyrrolo[1,2- a ]isoquinoline Derivatives via Diastereoselective and Regiodivergent Three-Component 1,3-Dipolar Cycloaddition Reactions: In Vitro and in Vivo Evaluation of the Antidiabetic Activity of Rhodanine Analogues . The Journal of Organic Chemistry 86:19, pages 13420-13445.
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