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Polycyclic Aromatic Compounds Volume 40, 2020 - Issue 4
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Articles

New Biscoumarin Derivatives as Potent α-Glucosidase Inhibitors: Synthesis, Biological Evaluation, Kinetic Analysis, and Docking Study

Maryam Mohammadi-KhanaposhtaniCellular and Molecular Biology Research Center, Health Research Institute, Babol University of Medical Sciences, Babol, Iran; View further author information
,
Hoda YahyaviFaculty of Chemistry and Physics, Department of Chemistry, Alzahra University, Tehran, Iran; View further author information
,
Ebrahim BarzegaricMedical Biology Research Center, Kermanshah University of Medical Sciences, Kermanshah, Iran; View further author information
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Somaye ImanparastDepartment of Pharmaceutical Biotechnology, Faculty of Pharmacy and Biotechnology Research Center, Tehran University of Medical Sciences, Iran; View further author information
,
Majid M. HeraviFaculty of Chemistry and Physics, Department of Chemistry, Alzahra University, Tehran, Iran; View further author information
,
Mohammad Ali FaramarziDepartment of Pharmaceutical Biotechnology, Faculty of Pharmacy and Biotechnology Research Center, Tehran University of Medical Sciences, Iran; View further author information
,
Alireza ForoumadiDepartment of Medicinal Chemistry, Faculty of Pharmacy and Pharmaceutical Sciences Research Center, Tehran University of Medical Sciences, Tehran, Iran; View further author information
,
Hossein AdibiEndocrinology and Metabolism Research Center, Endocrinology and Metabolism Clinical Sciences Institute, Tehran University of Medical Sciences, Tehran, IranView further author information
,
Bagher LarijaniEndocrinology and Metabolism Research Center, Endocrinology and Metabolism Clinical Sciences Institute, Tehran University of Medical Sciences, Tehran, IranCorrespondence[email protected] [email protected]
View further author information
&
Mohammad MahdaviEndocrinology and Metabolism Research Center, Endocrinology and Metabolism Clinical Sciences Institute, Tehran University of Medical Sciences, Tehran, IranCorrespondence[email protected] [email protected]
View further author information
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Pages 915-926 | Received 20 Apr 2018, Accepted 04 Aug 2018, Published online: 02 Nov 2018

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Soukaina Chehab, Youssef Merroun, Rachida Ghailane, Said Boukhris & Abdelaziz Souizi. (2023) Na2Ca(HPO4)2, an Efficient, Reusable Eco-Friendly Catalyst for the Synthesis of 1,8-Dioxo-Octahydroxanthenes and Biscoumarin Derivatives. Polycyclic Aromatic Compounds 43:6, pages 4906-4923.
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K. R. Kadam, G. R. Pandhare, A. S. Waghmare, V. D. Murade, N. R. Kamble & V. T. Kamble. (2023) Silica Chemisorbed Bis(Hydrogensulphato)Benzene (SiO2-BHSB) as a New, Environmentally Benign and Recyclable Catalyst for an Efficient Synthesis of Biscoumarin Scaffolds in Water Based Solvent. Polycyclic Aromatic Compounds 43:1, pages 647-664.
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Emad Elahabaadi, Amir Ahmad Salarian & Ehsan Nassireslami. (2022) Design, Synthesis, and Molecular Docking of Novel Hybrids of Coumarin-Dithiocarbamate Alpha-Glucosidase Inhibitors Targeting Type 2 Diabetes Mellitus. Polycyclic Aromatic Compounds 42:7, pages 4317-4327.
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Seyed Esmaeil Sadat-Ebrahimi, Hiva Babania, Maryam Mohammadi-Khanaposhtani, Mohammad Sadegh Asgari, Somayeh Mojtabavi, Mohammad Ali Faramarzi, Azadeh Yahya-Meymandi, Samaneh Zareie, Bagher Larijani, Mahmoud Biglar, Hossein Rastgar, Alireza Foroumadi & Mohammad Mahdavi. (2022) Design, Synthesis, and Biological Evaluation of New Indole-Acrylamide-1,2,3-Triazole Derivatives as Potential α-Glucosidase Inhibitors. Polycyclic Aromatic Compounds 42:6, pages 3157-3165.
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Jay Soni, Nusrat Sahiba, Ayushi Sethiya, Pankaj Teli, Dinesh Kr. Agarwal, Anu Manhas, Prakash Chandra Jha, Deepkumar Joshi & Shikha Agarwal. (2022) Biscoumarin Derivatives as Potent anti-Microbials: Graphene Oxide Catalyzed Eco-Benign Synthesis, Biological Evaluation and Docking Studies. Polycyclic Aromatic Compounds 42:6, pages 2970-2990.
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Articles from other publishers (23)

Mohammed El Behery, Ibrahim M. El-Deen, Manar A. El-Zend & Lamiaa A.A. Barakat. (2023) Design, synthesis and evaluation the bioactivities of novel 8‑methoxy-1-azacoumarin-3-carboxamide derivatives as anti-diabetic agents. Journal of Molecular Structure 1294, pages 136486.
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Ajay Thakur, Ruchi Bharti, Monika Verma, Renu Sharma, Ajay Sharma, Anshi GuptaVipasha Sharma. (2023) Ultra-Sonicated One-Pot Synthesis of Potent Bioactive Biscoumarin and Polycyclic Pyranodichromenone Scaffolds in Aqueous Media: A Complementary Tool to Organic Synthesis. Synthesis 55:19, pages 3129-3144.
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Fariba Peytam, Faezeh sadat Hosseini, Malak Hekmati, Bahareh Bayati, Mahdis Sadeghi Moghadam, Zahra Emamgholipour, Loghman Firoozpour, Somayeh Mojtabavi, Mohammad Ali Faramarzi, Seyed Esmaeil Sadat-Ebrahimi, Maliheh Barazandeh Tehrani & Alireza Foroumadi. (2023) Imidazo[1,2-c]quinazolines as a novel and potent scaffold of α-glucosidase inhibitors: design, synthesis, biological evaluations, and in silico studies. Scientific Reports 13:1.
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Faeze Yousefnejad, Mahyar Mohammadi-Moghadam-Goozali, Mohammad Hosein Sayahi, Mohammad Halimi, Ali Moazzam, Maryam Mohammadi-Khanaposhtani, Somayeh Mojtabavi, Mehdi Asadi, Mohammad Ali Faramarzi, Bagher Larijani, Massoud Amanlou & Mohammad Mahdavi. (2023) Design, synthesis, in vitro, and in silico evaluations of benzo[d]imidazole-amide-1,2,3-triazole-N-arylacetamide hybrids as new antidiabetic agents targeting α-glucosidase. Scientific Reports 13:1.
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Thi-Hong-Truc Phan, Kowit Hengphasatporn, Yasuteru Shigeta, Wanting Xie, Phornphimon Maitarad, Thanyada Rungrotmongkol & Warinthorn Chavasiri. (2023) Designing Potent α-Glucosidase Inhibitors: A Synthesis and QSAR Modeling Approach for Biscoumarin Derivatives. ACS Omega 8:29, pages 26340-26350.
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Mahtab Rahmani Gavanrudi, Mohammad Halimi, Hossein Najafzadehvarzi, Majid Alikhani, Ali MoazzamSoghra Farzipour, Samanesadat Hosseini, Somayeh Mojtabavi, Mohammad Ali Faramarzi, Ensieh Nasli‐Esfahani, Maryam Mohammadi‐Khanaposhtani & Mohammad Mahdavi. (2023) Discovery of Phthalimide‐1,2,3‐triazole‐ N ‐phenylacetamide Hybrids as Potent α‐Glucosidase Inhibitors: Design, Synthesis, ADMET Prediction, and in vitro and in silico Enzymatic Evaluations . ChemistrySelect 8:26.
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Sajedeh Safapoor, Mohammad Halimi, Minoo Khalili Ghomi, Milad Noori, Navid Dastyafteh, Shahrzad Javanshir, Samanesadat Hosseini, Somayeh Mojtabavi, Mohammad Ali Faramarzi, Ensieh Nasli-Esfahani, Bagher Larijani, Azadeh Fakhrioliaei, Mohammad G. Dekamin, Maryam Mohammadi-Khanaposhtani & Mohammad Mahdavi. (2023) Synthesis, ADMT prediction, and in vitro and in silico α-glucosidase inhibition evaluations of new quinoline–quinazolinone–thioacetamides . RSC Advances 13:28, pages 19243-19256.
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Mehdi Emadi, Mohammad Halimi, Ali Moazzam, Samanesadat Hosseini, Somayeh Mojtabavi, Mohammad Ali Faramarzi, Reza Ghadimi, Ali Akbar Moghadamnia, Ensieh Nasli-Esfahani, Maryam Mohammadi-Khanaposhtani & Mohammad Mahdavi. (2023) Design, synthesis, in vitro anti-α-glucosidase evaluations, and computational studies of new phthalimide-phenoxy-1,2,3-triazole-N-phenyl (or benzyl) acetamides as potential anti-diabetic agents. Scientific Reports 13:1.
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Alia Mushtaq, Uzma Azam, Saba Mehreen & Muhammad Moazzam Naseer. (2023) Synthetic α-glucosidase inhibitors as promising anti-diabetic agents: Recent developments and future challenges. European Journal of Medicinal Chemistry 249, pages 115119.
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Maryam Mohammadi‐Khanaposhtani, Milad Noori, Yousef Valizadeh, Navid Dastyafteh, Minoo Khalili Ghomi, Somayeh Mojtabavi, Mohammad Ali Faramarzi, Samanesadat Hosseini, Mahmood Biglar, Bagher Larijani, Hossein Rastegar, Haleh Hamedifar, Roghieh Mirzazadeh & Mohammad Mahdavi. (2022) Synthesis, α‐glucosidase Inhibition, in silico Pharmacokinetic, and Docking Studies Of Thieno[2,3‐b]Quinoline‐Acetamide Derivatives as New Anti‐Diabetic Agents . ChemistrySelect 7:44.
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Milad Noori, Mryam Rastak, Mohammad Halimi, Minoo Khalili Ghomi, Mrjan Mollazadeh, Maryam Mohammadi-Khanaposhtani, Mohammad Hosein Sayahi, Zahra Rezaei, Somayeh Mojtabavi, Mohammad Ali Faramarzi, Bagher Larijani, Mahmood Biglar, Massoud Amanlou & Mohammad Mahdavi. (2022) Design, synthesis, in vitro, and in silico enzymatic evaluations of thieno[2,3-b]quinoline-hydrazones as novel inhibitors for α-glucosidase. Bioorganic Chemistry 127, pages 105996.
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Homa Azizian, Keyvan Pedrood, Ali Moazzam, Yousef Valizadeh, Kimia Khavaninzadeh, Ali Zamani, Maryam Mohammadi-Khanaposhtani, Somayeh Mojtabavi, Mohammad Ali Faramarzi, Samanesadat Hosseini, Yaghoub Sarrafi, Hossein Adibi, Bagher Larijani, Hossein Rastegar & Mohammad Mahdavi. (2022) Docking study, molecular dynamic, synthesis, anti-α-glucosidase assessment, and ADMET prediction of new benzimidazole-Schiff base derivatives. Scientific Reports 12:1.
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Mohammad Sadegh Asgari, Maryam Mohammadi-Khanaposhtani, Zeinab Sharafi, Mohammad Ali Faramarzi, Hossein Rastegar, Ensieh Nasli Esfahani, Fatemeh Bandarian, Parviz Ranjbar Rashidi, Rahmatollah Rahimi, Mahmood Biglar, Mohammad Mahdavi & Bagher Larijani. (2020) Design and synthesis of 4,5-diphenyl-imidazol-1,2,3-triazole hybrids as new anti-diabetic agents: in vitro α-glucosidase inhibition, kinetic and docking studies. Molecular Diversity 25:2, pages 877-888.
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Madieh Sadeghpour, Abolfazl Olyaei & Alireza Adl. (2021) 4-Aminocoumarin derivatives: synthesis and applications. New Journal of Chemistry 45:13, pages 5744-5763.
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Ali Yavari, Maryam Mohammadi-Khanaposhtani, Shahram Moradi, Saeed Bahadorikhalili, Roghayeh Pourbagher, Nasrin Jafari, Mohammad Ali Faramarzi, Ebrahim Zabihi, Mohammad Mahdavi, Mahmood Biglar, Bagher Larijani, Haleh Hamedifar & Mir Hamed Hajimiri. (2021) α-Glucosidase and α-amylase inhibition, molecular modeling and pharmacokinetic studies of new quinazolinone-1,2,3-triazole-acetamide derivatives. Medicinal Chemistry Research 30:3, pages 702-711.
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Marjan Mollazadeh, Maryam Mohammadi-Khanaposhtani, Yousef Valizadeh, Afsaneh Zonouzi, Mohammad Ali Faramarzi, Parsa Hariri, Mahmood Biglar, Bagher Larijani, Haleh Hamedifar, Mohammad Mahdavi & Nima Sepehri. (2020) 2,4-Dioxochroman Moiety Linked to 1,2,3-triazole Derivatives as Novel α-glucosidase Inhibitors: Synthesis, In vitro Biological Evaluation, and Docking Study. Current Organic Chemistry 24:17, pages 2019-2027.
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Maryam Mohammadi‐Khanaposhtani, Hoda Yahyavi, Somaye Imanparast, Fereshte Nazemi Harandi, Mohammad Ali Faramarzi, Alireza Foroumadi, Bagher Larijani, Mahmood Biglar & Mohammad Mahdavi. (2019) Benzoylquinazolinone derivatives as new potential antidiabetic agents: α‐Glucosidase inhibition, kinetic, and docking studies. Journal of the Chinese Chemical Society 67:5, pages 856-863.
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Tadesse Bekele Tafesse, Mohammed Hussen Bule, Mehdi Khoobi, Mohammad Ali Faramarzi, Mohammad Abdollahi & Mohsen Amini. (2020) Coumarin-based Scaffold as α-glucosidase Inhibitory Activity: Implication for the Development of Potent Antidiabetic Agents. Mini-Reviews in Medicinal Chemistry 20:2, pages 134-151.
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Fariba Peytam, Mehdi Adib, Reihaneh Shourgeshty, Loghman Firoozpour, Mahmoud Rahmanian-Jazi, Mehdi Jahani, Setareh Moghimi, Kouros Divsalar, Mohammad Ali Faramarzi, Somayeh Mojtabavi, Fatemeh Safari, Mohammad Mahdavi & Alireza Foroumadi. (2020) An efficient and targeted synthetic approach towards new highly substituted 6-amino-pyrazolo[1,5-a]pyrimidines with α-glucosidase inhibitory activity. Scientific Reports 10:1.
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Pankaj Teli, Ayushi Sethiya & Shikha Agarwal. (2019) An Insight View on Synthetic Protocol, Mechanistic and Biological Aspects of Biscoumarin Derivatives. ChemistrySelect 4:47, pages 13772-13787.
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Zohreh Bakherad, Maryam Mohammadi-Khanaposhtani, Hojjat Sadeghi-Aliabadi, Sepideh Rezaei, Afshin Fassihi, Mohammad Bakherad, Hossein Rastegar, Mahmood Biglar, Lotfollah Saghaie, Bagher Larijani & Mohammad Mahdavi. (2019) New thiosemicarbazide-1,2,3-triazole hybrids as potent α-glucosidase inhibitors: Design, synthesis, and biological evaluation. Journal of Molecular Structure 1192, pages 192-200.
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Manoj Dhameja & Preeti Gupta. (2019) Synthetic heterocyclic candidates as promising α-glucosidase inhibitors: An overview. European Journal of Medicinal Chemistry 176, pages 343-377.
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Ensieh Nasli‐Esfahani, Maryam Mohammadi‐Khanaposhtani, Sepideh Rezaei, Yaghoub Sarrafi, Zeinab Sharafi, Nasser Samadi, Mohammad Ali Faramarzi, Fatemeh Bandarian, Haleh Hamedifar, Bagher Larijani, Mirhamed Hajimiri & Mohammad Mahdavi. (2019) A new series of Schiff base derivatives bearing 1,2,3‐triazole: Design, synthesis, molecular docking, and α‐glucosidase inhibition. Archiv der Pharmazie 352:8.
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