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Journal of Receptors and Signal Transduction Volume 28, 2008 - Issue 3
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Research Article

Biochemical Assay-Based Selectivity Profiling of Clinically Relevant Kinase Inhibitors on Mutant Forms of EGF Receptor

EDIT VARKONDI Rational Drug Design Laboratory CRC, Semmelweis University, Budapest, Hungary
,
FERENC PINTER KPS Biotechnology & Healthcare Services Ltd, Budapest, Hungary
,
KISS ROBERT Department of Pharmaceutical Chemistry, Semmelweis University, Budapest, Hungary
,
RICHARD SCHWAB Rational Drug Design Laboratory CRC, Semmelweis University, Budapest, Hungary; KPS Biotechnology & Healthcare Services Ltd, Budapest, Hungary
,
NORA BREZA Rational Drug Design Laboratory CRC, Semmelweis University, Budapest, Hungary; Pathobiochemical Research Group, Hungarian Academy of Sciences, Budapest, Hungary; Vichem Chemie Research Ltd., Budapest, Hungary
,
LASZLO ÖRFI Rational Drug Design Laboratory CRC, Semmelweis University, Budapest, Hungary; Department of Pharmaceutical Chemistry, Semmelweis University, Budapest, Hungary; Vichem Chemie Research Ltd., Budapest, Hungary
,
GYÖRGY KERI Rational Drug Design Laboratory CRC, Semmelweis University, Budapest, Hungary; Pathobiochemical Research Group, Hungarian Academy of Sciences, Budapest, Hungary; Vichem Chemie Research Ltd., Budapest, Hungary
&
ISTVAN PETAK Rational Drug Design Laboratory CRC, Semmelweis University, Budapest, Hungary; KPS Biotechnology & Healthcare Services Ltd, Budapest, Hungary; 1st Department of Pathology and Experimental Cancer Research, Semmelweis University, Budapest, Hungary
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Pages 295-306 | Published online: 10 Oct 2008

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NÓRA BREZA, JÁNOS PATÓ, LÁSZLÓ ŐRFI, BÁLINT HEGYMEGI-BARAKONYI, PÉTER BÁNHEGYI, EDIT VÁRKONDI, GÁBOR BORBÉLY, ISTVÁN PETÁK & GYÖRGY KÉRI. (2008) Synthesis and Characterization of Novel Quinazoline Type Inhibitors for Mutant and Wild-Type EGFR and RICK Kinases. Journal of Receptors and Signal Transduction 28:4, pages 361-373.
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Articles from other publishers (4)

Alessia Di Florio, Veronica Sancho, Paola Moreno, Gianfranco Delle Fave & Robert T. Jensen. (2013) Gastrointestinal hormones stimulate growth of Foregut Neuroendocrine Tumors by transactivating the EGF receptor. Biochimica et Biophysica Acta (BBA) - Molecular Cell Research 1833:3, pages 573-582.
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István Peták, Richárd Schwab, László Őrfi, László Kopper & György Kéri. (2010) Integrating molecular diagnostics into anticancer drug discovery. Nature Reviews Drug Discovery 9:7, pages 523-535.
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Ibrahim F. Benter, Halit Canatan, Mustapha Benboubetra, Mariam H.M. Yousif & Saghir Akhtar. (2009) Global upregulation of gene expression associated with renal dysfunction in DOCA–salt-induced hypertensive rats occurs via signaling cascades involving epidermal growth factor receptor: A microarray analysis. Vascular Pharmacology 51:2-3, pages 101-109.
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Miyako Satouchi. (2009) Selective Use of Gefitinib and Erlotinib on Non-small Cell Lung Cancer Patients. Haigan 49:6, pages 950-956.
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