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Qiqi Huang, Tianli Lai, Qu Wang & Lianxiang Luo. (2023) mPGES-1 Inhibitor Discovery Based on Computer-Aided Screening: Pharmacophore Models, Molecular Docking, ADMET, and MD Simulations. Molecules 28:16, pages 6059.
Crossref
Crossref
Thota Ganesh. (2023) Targeting EP2 Receptor for Drug Discovery: Strengths, Weaknesses, Opportunities, and Threats (SWOT) Analysis. Journal of Medicinal Chemistry 66:14, pages 9313-9324.
Crossref
Crossref
Madison N Sluter, Qianqian Li, Nelufar Yasmen, Yu Chen, Lexiao Li, Ruida Hou, Ying Yu, Chao-Yie Yang, Bernd Meibohm & Jianxiong Jiang. (2023) The inducible prostaglandin E synthase (mPGES-1) in neuroinflammatory disorders. Experimental Biology and Medicine 248:9, pages 811-819.
Crossref
Crossref
Madison N. Sluter, Rajib Bhuniya, Xinrui Yuan, Andhavaram Ramaraju, Yu Chen, Ying Yu, Keyur R. Parmar, Zaid H. Temrikar, Ashish Srivastava, Bernd Meibohm, Jianxiong Jiang & Chao-Yie Yang. (2023)
Novel, Brain-Permeable, Cross-Species Benzothiazole Inhibitors of Microsomal Prostaglandin E Synthase-1 (mPGES-1) Dampen Neuroinflammation
In Vitro
and
In Vivo
. ACS Pharmacology & Translational Science 6:4, pages 587-599.
Crossref
Crossref
Marianna Potenza, Assunta Giordano, Maria G. Chini, Anella Saviano, Christian Kretzer, Federica Raucci, Marina Russo, Gianluigi Lauro, Stefania Terracciano, Ines Bruno, Maria Iorizzi, Robert K. Hofstetter, Simona Pace, Francesco Maione, Oliver Werz & Giuseppe Bifulco. (2022)
Identification of 2-Aminoacyl-1,3,4-thiadiazoles as Prostaglandin E
2
and Leukotriene Biosynthesis Inhibitors
. ACS Medicinal Chemistry Letters 14:1, pages 26-34.
Crossref
Crossref
Demiana S. Mikhail, Hala B. El‐Nassan, Sally T. Mahmoud & Samar H. Fahim. (2022) Nonacidic thiophene‐based derivatives as potential analgesic and design, synthesis, biological evaluation, and metabolic stability study. Drug Development Research 83:8, pages 1739-1757.
Crossref
Crossref
Igor José dos Santos Nascimento, Thiago Mendonça de Aquino & Edeildo Ferreira da Silva Júnior. (2022)
Computer-Aided Drug Design of Anti-inflammatory Agents Targeting
Microsomal Prostaglandin E
2
Synthase-1 (mPGES-1)
. Current Medicinal Chemistry 29:33, pages 5397-5419.
Crossref
Crossref
Azize Gizem Ergül, Tuğçe Gür Maz, Christian Kretzer, Abdurrahman Olğaç, Paul M. Jordan, Burcu Çalışkan, Oliver Werz & Erden Banoglu. (2022) Novel potent benzimidazole-based microsomal prostaglandin E2 synthase-1 (mPGES-1) inhibitors derived from BRP-201 that also inhibit leukotriene C4 synthase. European Journal of Medicinal Chemistry 231, pages 114167.
Crossref
Crossref
Maria A. Theodoropoulou, Anastasia Psarra, Martin Erhardt, Aikaterini Nikolaou, Anna-Dimitra D. Gerogiannopoulou, Dimitra Hadjipavlou-Litina, Daiki Hayashi, Edward A. Dennis, Andrea Huwiler & George Kokotos. (2022) N-Acylated and N-Alkylated 2-Aminobenzothiazoles Are Novel Agents That Suppress the Generation of Prostaglandin E2. Biomolecules 12:2, pages 267.
Crossref
Crossref
Kassandra T. Ávila-Alvarez, Mónica L. Chávez-González, Elda P. Segura-Ceniceros, José L. Martínez-Hernández, Roberto Arredondo-Valdes, Mayela Govea-Salas, Erika Nava-Reyna, Anna Ilyina & Rodolfo Ramos-González. 2022. Value-Addition in Food Products and Processing Through Enzyme Technology. Value-Addition in Food Products and Processing Through Enzyme Technology
413
425
.
Kathiravan M K, Swethan Babu, Chitra Vellapandian, Vigneshwaran Namasivayam & Senthilkumar Palaniappan. 2022. Systems Biomedicine Approaches in Cancer Research. Systems Biomedicine Approaches in Cancer Research
71
95
.
Shafinaz Nur, Md. Mohotasin Hossain, Nadia Islam, Abu Montakim Tareq, Nujhat Binte Hanif, Riniara Khatun & Mohammed Abu Sayeed. (2021) Scrutinizing pharmacological efficiency for Acacia auriculiformis by experimental and computational approach. Future Journal of Pharmaceutical Sciences 7:1.
Crossref
Crossref
Lenisa Dandara dos Santos, Thamires Quadros Froes, Miriam Cristina Contin de Melo, Gloria Emília Petto de Souza, Denis de Melo Soares & Marcelo Santos Castilho. (2021) Triazol-phenyl Antipyretic Derivatives Inhibit mPGES-1 mRNA Levels in LPS-Induced RAW 264.7 Macrophage Cells. Anti-Inflammatory & Anti-Allergy Agents in Medicinal Chemistry 20:3, pages 271-281.
Crossref
Crossref
Simone Di Micco, Stefania Terracciano, Dafne Ruggiero, Marianna Potenza, Maria C. Vaccaro, Katrin Fischer, Oliver Werz, Ines Bruno & Giuseppe Bifulco. (2021) Identification of 2-(thiophen-2-yl)acetic Acid-Based Lead Compound for mPGES-1 Inhibition. Frontiers in Chemistry 9.
Crossref
Crossref
Anastasia Psarra, Maria A. Theodoropoulou, Martin Erhardt, Marina Mertiri, Christiana Mantzourani, Sofia Vasilakaki, Victoria Magrioti, Andrea Huwiler & George Kokotos. (2021) α-Ketoheterocycles Able to Inhibit the Generation of Prostaglandin E2 (PGE2) in Rat Mesangial Cells. Biomolecules 11:2, pages 275.
Crossref
Crossref
X. Jiang, H. Renkema, B. Pennings, S. Pecheritsyna, J. C. Schoeman, T. Hankemeier, J. Smeitink & J. Beyrath. (2021) Mechanism of action and potential applications of selective inhibition of microsomal prostaglandin E synthase-1-mediated PGE2 biosynthesis by sonlicromanol’s metabolite KH176m. Scientific Reports 11:1.
Crossref
Crossref
Lauri Tuure, Antti Pemmari, Mari Hämäläinen, Teemu Moilanen & Eeva Moilanen. (2020) Regulation of gene expression by MF63, a selective inhibitor of microsomal PGE synthase 1 (mPGES1) in human osteoarthritic chondrocytes. British Journal of Pharmacology 177:18, pages 4134-4146.
Crossref
Crossref
Madhuranayaki Thulasingam & Jesper Z. Haeggström. (2020) Integral Membrane Enzymes in Eicosanoid Metabolism: Structures, Mechanisms and Inhibitor Design. Journal of Molecular Biology 432:18, pages 4999-5022.
Crossref
Crossref
Jun Chul Park, Atsushi Hagiwara, Heum Gi Park & Jae-Seong Lee. (2020) The glutathione S-transferase genes in marine rotifers and copepods: Identification of GSTs and applications for ecotoxicological studies. Marine Pollution Bulletin 156, pages 111080.
Crossref
Crossref
Luigia Di Francesco, Annalisa Bruno, Emanuela Ricciotti, Stefania Tacconelli, Melania Dovizio, Paloma Guillem-Llobat, Maria Alessandra Alisi, Beatrice Garrone, Isabella Coletta, Giorgina Mangano, Claudio Milanese, Garret A. FitzGerald & Paola Patrignani. (2020) Pharmacological Characterization of the Microsomal Prostaglandin E2 Synthase-1 Inhibitor AF3485 In Vitro and In Vivo. Frontiers in Pharmacology 11.
Crossref
Crossref
Filip Bergqvist, Ralf Morgenstern & Per-Johan Jakobsson. (2020) A review on mPGES-1 inhibitors: From preclinical studies to clinical applications. Prostaglandins & Other Lipid Mediators 147, pages 106383.
Crossref
Crossref
Shilpa Choudhary & Carol Pilbeam. 2020. Principles of Bone Biology. Principles of Bone Biology
1247
1269
.
Tony Avril & Eric Chevet. (2019) Stress signaling in pain control. Science 365:6450, pages 224-225.
Crossref
Crossref
Sun-Hee Kim, Jason Roszik, Sung-Nam Cho, Dai Ogata, Denái R. Milton, Weiyi Peng, David G. Menter, Suhendan Ekmekcioglu & Elizabeth A. Grimm. (2019) The COX2 Effector Microsomal PGE2 Synthase 1 is a Regulator of Immunosuppression in Cutaneous Melanoma. Clinical Cancer Research 25:5, pages 1650-1663.
Crossref
Crossref
Karin Larsson, Anna Kock, Per Kogner & Per-Johan Jakobsson. 2019. The Role of Bioactive Lipids in Cancer, Inflammation and Related Diseases. The Role of Bioactive Lipids in Cancer, Inflammation and Related Diseases
89
100
.
Carol Pilbeam. 2020. Bone Regulators and Osteoporosis Therapy. Bone Regulators and Osteoporosis Therapy
157
175
.
Gianluigi Lauro, Vincenza Cantone, Marianna Potenza, Katrin Fischer, Andreas Koeberle, Oliver Werz, Raffaele Riccio & Giuseppe Bifulco. (2018) Discovery of 3-hydroxy-3-pyrrolin-2-one-based mPGES-1 inhibitors using a multi-step virtual screening protocol. MedChemComm 9:12, pages 2028-2036.
Crossref
Crossref
Ashish Gupta, Neha Chaudhary & Polamarasetty Aparoy. (2018) MM-PBSA and per-residue decomposition energy studies on 7-Phenyl-imidazoquinolin-4(5H)-one derivatives: Identification of crucial site points at microsomal prostaglandin E synthase-1 (mPGES-1) active site. International Journal of Biological Macromolecules 119, pages 352-359.
Crossref
Crossref
Andreas Koeberle & Oliver Werz. (2018) Natural products as inhibitors of prostaglandin E2 and pro-inflammatory 5-lipoxygenase-derived lipid mediator biosynthesis. Biotechnology Advances 36:6, pages 1709-1723.
Crossref
Crossref
Mayuri Napagoda, Jana Gerstmeier, Hannah Butschek, Sybille Lorenz, Dinusha Kanatiwela, Mallique Qader, Ajith Nagahawatte, Sudhara De Soyza, Gaya Bandara Wijayaratne, Aleš Svatoš, Lalith Jayasinghe, Andreas Koeberle & Oliver Werz. (2018) Lipophilic extracts of Leucas zeylanica, a multi-purpose medicinal plant in the tropics, inhibit key enzymes involved in inflammation and gout. Journal of Ethnopharmacology 224, pages 474-481.
Crossref
Crossref
Preeti Kanikarla-Marie, Scott Kopetz, Ernest T. Hawk, Steven W. Millward, Anil K. Sood, Paolo Gresele, Michael Overman, Kenneth Honn & David G. Menter. (2018) Bioactive lipid metabolism in platelet “first responder” and cancer biology. Cancer and Metastasis Reviews 37:2-3, pages 439-454.
Crossref
Crossref
Nagarajan Muthukaman, Sanjay Deshmukh, Macchindra Tambe, Dnyandeo Pisal, Shital Tondlekar, Mahamadhanif Shaikh, Neelam Sarode, Vidya G. Kattige, Pooja Sawant, Monali Pisat, Vikas Karande, Srinivasa Honnegowda, Abhay Kulkarni, Dayanidhi Behera, Satyawan B. Jadhav, Ramchandra R. Sangana, Girish S. Gudi, Neelima Khairatkar-Joshi & Laxmikant A. Gharat. (2018) Alleviating CYP and hERG liabilities by structure optimization of dihydrofuran-fused tricyclic benzo[ d ]imidazole series – Potent, selective and orally efficacious microsomal prostaglandin E synthase-1 (mPGES-1) inhibitors: Part-2. Bioorganic & Medicinal Chemistry Letters 28:7, pages 1211-1218.
Crossref
Crossref
Nerino Allocati, Michele Masulli, Carmine Di Ilio & Luca Federici. (2018) Glutathione transferases: substrates, inihibitors and pro-drugs in cancer and neurodegenerative diseases. Oncogenesis 7:1.
Crossref
Crossref
Sofia Vasilakaki, Oleksandr Pastukhov, Thomas Mavromoustakos, Andrea Huwiler & George Kokotos. (2018) Small Peptides Able to Suppress Prostaglandin E2 Generation in Renal Mesangial Cells. Molecules 23:1, pages 158.
Crossref
Crossref
Ioana Mozos, Clemens Malainer, Jarosław Horbańczuk, Cristina Gug, Dana Stoian, Constantin Tudor Luca & Atanas G. Atanasov. (2017) Inflammatory Markers for Arterial Stiffness in Cardiovascular Diseases. Frontiers in Immunology 8.
Crossref
Crossref