Citations (27)
Keep up to date with the latest research on this topic with citation updates for this article.
Articles from other publishers (27)
Dorota Łażewska, Maria Kaleta, Paula Zaręba, Justyna Godyń, Mariam Dubiel, Ewelina Honkisz-Orzechowska, Agata Doroz-Płonka, Anna Więckowska, Holger Stark & Katarzyna Kieć-Kononowicz. (2023) Multitargeting Histamine H3 Receptor Ligands among Acetyl- and Propionyl-Phenoxyalkyl Derivatives. Molecules 28:5, pages 2349.
Crossref
Crossref
Hu Luo, Xiaofang Li, Runyue Fan, Yuer Ruan, Liyin Qian, Yao Shen, Zizhen Si, Longhui Li & Yu Liu. (2023) Neuroprotective effect of histamine H3 receptor blockade on methamphetamine-induced cognitive impairment in mice. Pharmacology Biochemistry and Behavior 222, pages 173512.
Crossref
Crossref
Vittoria Borgonetti & Nicoletta Galeotti. (2022) The Histamine H4 Receptor Participates in the Neuropathic Pain-Relieving Activity of the Histamine H3 Receptor Antagonist GSK189254. International Journal of Molecular Sciences 23:22, pages 14314.
Crossref
Crossref
Ziying Li, Xinyi Xiao, Yulin Xue, Huiling Zhou, Chaonan Huang, Mo Zhu, Tao Zhuang, Yin Chen & Ling Huang. (2022) Discovery of a novel class of benzoxazole derivatives as histamine H3 receptor ligands for the treatment of neuropathic pain. Bioorganic Chemistry 127, pages 106039.
Crossref
Crossref
Zsolt Némethy, Béla Kiss, Natasha Lethbridge, Paul Chazot, Tünde Hajnik, Attila Tóth, László Détári, Éva Schmidt, András Czurkó, Diána Kostyalik, Vilmos Oláh, István Hernádi, Ottilia Balázs, E. Sylvester Vizi, István Ledneczki, Sándor Mahó, Viktor Román, Balázs Lendvai & György Lévay. (2022) Convergent cross-species pro-cognitive effects of RGH-235, a new potent and selective histamine H3 receptor antagonist/inverse agonist. European Journal of Pharmacology 916, pages 174621.
Crossref
Crossref
Markus Falkenstein, David Reiner-Link, Aleksandra Zivkovic, Ian Gering, Dieter Willbold & Holger Stark. (2021) Histamine H3 receptor antagonists with peptidomimetic (keto)piperazine structures to inhibit Aβ oligomerisation. Bioorganic & Medicinal Chemistry 50, pages 116462.
Crossref
Crossref
Dorota Łażewska, Paula Zaręba, Justyna Godyń, Agata Doroz-Płonka, Annika Frank, David Reiner-Link, Marek Bajda, Dorota Stary, Szczepan Mogilski, Agnieszka Olejarz-Maciej, Maria Kaleta, Holger Stark, Barbara Malawska & Katarzyna Kieć-Kononowicz. (2021) Biphenylalkoxyamine Derivatives–Histamine H3 Receptor Ligands with Butyrylcholinesterase Inhibitory Activity. Molecules 26:12, pages 3580.
Crossref
Crossref
Ramakrishna Nirogi, Venkata R Grandhi, Rajesh B Medapati, Narender Ganuga, Vijay Benade, Sudhakar Gandipudi, Arunkumar Manoharan, Renny Abraham, Pradeep Jayarajan, Gopinadh Bhyrapuneni, Anil Shinde, Rajesh K Badange, Ramkumar Subramanian, Surendra Petlu & Venkat Jasti. (2021) Histamine 3 receptor inverse agonist Samelisant (SUVN-G3031): Pharmacological characterization of an investigational agent for the treatment of cognitive disorders. Journal of Psychopharmacology 35:6, pages 713-729.
Crossref
Crossref
Katarzyna Szczepańska, Kamil J. Kuder & Katarzyna Kieć-Kononowicz. (2021) Dual-targeting Approach on Histamine H3 and Sigma-1 Receptor Ligands as Promising Pharmacological Tools in the Treatment of CNS-linked Disorders. Current Medicinal Chemistry 28:15, pages 2974-2995.
Crossref
Crossref
Kamil J. Kuder, Magdalena Kotańska, Katarzyna Szczepańska, Kamil Mika, David Reiner-Link, Holger Stark & Katarzyna Kieć-Kononowicz. (2021) Discovery of Potential, Dual-Active Histamine H3 Receptor Ligands with Combined Antioxidant Properties. Molecules 26:8, pages 2300.
Crossref
Crossref
Xiaoyuan Ma, Marta Arimont Segura, Barbara Zarzycka, Henry F. Vischer & Rob Leurs. (2021) Analysis of Missense Variants in the Human Histamine Receptor Family Reveals Increased Constitutive Activity of E4106.30×30K Variant in the Histamine H1 Receptor. International Journal of Molecular Sciences 22:7, pages 3702.
Crossref
Crossref
Katarzyna Szczepańska, Steffen Pockes, Sabina Podlewska, Carina Höring, Kamil Mika, Gniewomir Latacz, Marek Bednarski, Agata Siwek, Tadeusz Karcz, Martin Nagl, Merlin Bresinsky, Denise Mönnich, Ulla Seibel, Kamil J. Kuder, Magdalena Kotańska, Holger Stark, Sigurd Elz & Katarzyna Kieć-Kononowicz. (2021) Structural modifications in the distal, regulatory region of histamine H3 receptor antagonists leading to the identification of a potent anti-obesity agent. European Journal of Medicinal Chemistry 213, pages 113041.
Crossref
Crossref
Natalia C. Fernández & Federico Monczor. 2021. Encyclopedia of Molecular Pharmacology. Encyclopedia of Molecular Pharmacology
805
810
.
Natalia C. Fernández & Federico Monczor. 2020. Encyclopedia of Molecular Pharmacology. Encyclopedia of Molecular Pharmacology
1
6
.
Markus Falkenstein, Milica Elek & Holger Stark. 2022. The Functional Roles of Histamine Receptors. The Functional Roles of Histamine Receptors
29
76
.
Dorota Łażewska, Marek Bajda, Maria Kaleta, Paula Zaręba, Agata Doroz-Płonka, Agata Siwek, Alaa Alachkar, Szczepan Mogilski, Ali Saad, Kamil Kuder, Agnieszka Olejarz-Maciej, Justyna Godyń, Dorota Stary, Sylwia Sudoł, Małgorzata Więcek, Gniewomir Latacz, Maria Walczak, Jadwiga Handzlik, Bassem Sadek, Barbara Malawska & Katarzyna Kieć-Kononowicz. (2020) Rational design of new multitarget histamine H3 receptor ligands as potential candidates for treatment of Alzheimer’s disease. European Journal of Medicinal Chemistry 207, pages 112743.
Crossref
Crossref
Mizuki Watanabe, Takaaki Kobayashi, Yoshihiko Ito, Shizuo Yamada & Satoshi Shuto. (2020) Conformational Restriction of Histamine with a Rigid Bicyclo[3.1.0]hexane Scaffold Provided Selective H3 Receptor Ligands. Molecules 25:16, pages 3562.
Crossref
Crossref
Hannes Schihada, Xiaoyuan Ma, Ulrike Zabel, Henry F. Vischer, Gunnar Schulte, Rob Leurs, Steffen Pockes & Martin J. Lohse. (2020)
Development of a Conformational Histamine H
3
Receptor Biosensor for the Synchronous Screening of Agonists and Inverse Agonists
. ACS Sensors 5:6, pages 1734-1742.
Crossref
Crossref
Gustavo Provensi, Maria Beatrice Passani, Alessia Costa, Ivan Izquierdo & Patrizio Blandina. (2018) Neuronal histamine and the memory of emotionally salient events. British Journal of Pharmacology 177:3, pages 557-569.
Crossref
Crossref
Cinzia Volonté, Savina Apolloni & Mario Sabatelli. (2019) Histamine beyond its effects on allergy: Potential therapeutic benefits for the treatment of Amyotrophic Lateral Sclerosis (ALS). Pharmacology & Therapeutics 202, pages 120-131.
Crossref
Crossref
Salim M. A. Bastaki, Naheed Amir, Małgorzata Więcek, Katarzyna Kieć-Kononowicz & Bassem Sadek. (2019) Influence of the Novel Histamine H3 Receptor Antagonist/Inverse Agonist M39 on Gastroprotection and PGE2 Production Induced by (R)-Alpha-Methylhistamine in C57BL/6 Mice. Frontiers in Pharmacology 10.
Crossref
Crossref
Sara Salimi & Esmaeal Tamaddonfard. (2019) Microinjection of histamine and its H3 receptor agonist and antagonist into the agranular insular cortex influence sensory and affective components of neuropathic pain in rats. European Journal of Pharmacology 857, pages 172450.
Crossref
Crossref
Younggi Choi & Brian K. Raymer. (2019) Sleep modulating agents. Bioorganic & Medicinal Chemistry Letters 29:16, pages 2025-2033.
Crossref
Crossref
Ajeet Kumar, Venkata Reddy Pasam, Ravi Kumar Thakur, Maninder Singh, Kartikey Singh, Mahendra Shukla, Anubhav Yadav, Shalini Dogra, Chandan Sona, Deepmala Umrao, Swati Jaiswal, Hafsa Ahmad, Mamunur Rashid, Sandeep K. Singh, Muhammad Wahajuddin, Anil Kumar Dwivedi, Mohammad Imran Siddiqi, Jawahar Lal, Rama Pati Tripathi & Prem N. Yadav. (2019) Novel Tetrahydroquinazolinamines as Selective Histamine 3 Receptor Antagonists for the Treatment of Obesity. Journal of Medicinal Chemistry 62:9, pages 4638-4655.
Crossref
Crossref
Darren M. Riddy, Anna E. Cook, David M. Shackleford, Tracie L. Pierce, Elisabeth Mocaer, Clotilde Mannoury la Cour, Aurore Sors, William N. Charman, Roger J. Summers, Patrick M. Sexton, Arthur Christopoulos & Christopher J. Langmead. (2019) Drug-receptor kinetics and sigma-1 receptor affinity differentiate clinically evaluated histamine H3 receptor antagonists. Neuropharmacology 144, pages 244-255.
Crossref
Crossref
Takehito Ito, Yasuyuki Kimura, Chie Seki, Masanori Ichise, Keita Yokokawa, Kazunori Kawamura, Hidehiko Takahashi, Makoto Higuchi, Ming-Rong Zhang, Tetsuya Suhara & Makiko Yamada. (2018) Histamine H3 receptor density is negatively correlated with neural activity related to working memory in humans. EJNMMI Research 8:1.
Crossref
Crossref
Mohammad A. Khanfar, David Reiner, Stefanie Hagenow & Holger Stark. (2018) Design, synthesis, and biological evaluation of novel oxadiazole- and thiazole-based histamine H3R ligands. Bioorganic & Medicinal Chemistry 26:14, pages 4034-4046.
Crossref
Crossref