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Drug Evaluation

Lomitapide for the treatment of hypertriglyceridemia

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Pages 1457-1463 | Received 08 Aug 2016, Accepted 25 Oct 2016, Published online: 09 Nov 2016

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Elad Shemesh & Barak Zafrir. (2019) Hypertriglyceridemia-Related Pancreatitis In Patients With Type 2 Diabetes: Links And Risks. Diabetes, Metabolic Syndrome and Obesity 12, pages 2041-2052.
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David Rhainds, Mathieu R. Brodeur & Jean-Claude Tardif. (2019) Investigational drugs in development for hypertriglyceridemia: a coming-of-age story. Expert Opinion on Investigational Drugs 28:12, pages 1059-1079.
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Etienne Khoury, Diane Brisson, Nathalie Roy, Gérald Tremblay & Daniel Gaudet. (2019) Review of the long-term safety of lomitapide: a microsomal triglycerides transfer protein inhibitor for treating homozygous familial hypercholesterolemia. Expert Opinion on Drug Safety 18:5, pages 403-414.
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Articles from other publishers (16)

Mingyu Zhang, Taoyuan Yin, Feng Xia, Suhong Xia, Wangdong Zhou, Yu Zhang, Xu Han, Kai Zhao, Lina Feng, Ruonan Dong, Dean Tian, Yan Yu & Jiazhi Liao. (2022) Hypertriglyceridemia may contribute to stroke and pancreatitis: A case report and review of the literature. Frontiers in Endocrinology 13.
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Yangmin Zheng, Yue Hu, Ziping Han, Feng Yan, Sijia Zhang, Zhenhong Yang, Fangfang Zhao, Lingzhi Li, Junfen Fan, Rongliang Wang & Yumin Luo. (2022) Lomitapide ameliorates middle cerebral artery occlusion‐induced cerebral ischemia/reperfusion injury by promoting neuronal autophagy and inhibiting microglial migration. CNS Neuroscience & Therapeutics 28:12, pages 2183-2194.
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Amanda J Berberich & Robert A Hegele. (2022) A Modern Approach to Dyslipidemia. Endocrine Reviews 43:4, pages 611-653.
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Isabel Shamsudeen & Robert A. Hegele. (2022) Advances in the care of lipodystrophies. Current Opinion in Endocrinology, Diabetes & Obesity 29:2, pages 152-160.
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Jun-Shang Huang, Bin-Bin Guo, Fei-Fei Lin, Li-Min Zeng, Ting Wang, Xiang-Yu Dang, Yang Yang, You-Hong Hu, Jia Liu & He-Yao Wang. (2021) A novel low systemic diacylglycerol acyltransferase 1 inhibitor, Yhhu2407, improves lipid metabolism. European Journal of Pharmaceutical Sciences 158, pages 105683.
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Angelo B. Cefalù, Antonina Giammanco, Davide Noto, Rossella Spina, Daniela Cabibi, Carlo M. Barbagallo & Maurizio Averna. (2020) Effectiveness and safety of lomitapide in a patient with familial chylomicronemia syndrome. Endocrine 71:2, pages 344-350.
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Alan S. Brown, Ehab G. Dababneh, Adib Chaus, Vadzim Chyzhyk, Victor Marinescu & Nataliya Pyslar. 2021. Therapeutic Lipidology. Therapeutic Lipidology 35 80 .
Antonio Gallo, Sophie Béliard, Laura D’Erasmo & Eric Bruckert. (2020) Familial Chylomicronemia Syndrome (FCS): Recent Data on Diagnosis and Treatment. Current Atherosclerosis Reports 22:11.
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Juan Pedro-Botet, Juan F. Ascaso, Mariano Blasco, Ángel Brea, Ángel Díaz, Antonio Hernández-Mijares, Xavier Pintó & Jesús Millán. (2020) Triglicéridos, colesterol HDL y dislipidemia aterogénica en la guía europea para el control de las dislipidemias 2019. Clínica e Investigación en Arteriosclerosis 32:5, pages 209-218.
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Juan Pedro-Botet, Juan F. Ascaso, Mariano Blasco, Ángel Brea, Ángel Díaz, Antonio Hernández-Mijares, Xavier Pintó & Jesús Millán. (2020) Triglycerides, HDL cholesterol and atherogenic dyslipidaemia in the 2019 European guidelines for the management of dyslipidaemias. Clínica e Investigación en Arteriosclerosis (English Edition) 32:5, pages 209-218.
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Antonina Giammanco, Angelo B. Cefalù, Davide Noto & Maurizio R. Averna. (2020) Therapeutic Options for Homozygous Familial Hypercholesterolemia: The Role of Lomitapide. Current Medicinal Chemistry 27:23, pages 3773-3783.
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Vadzim Chyzhyk & Alan S. Brown. (2020) Familial chylomicronemia syndrome: A rare but devastating autosomal recessive disorder characterized by refractory hypertriglyceridemia and recurrent pancreatitis. Trends in Cardiovascular Medicine 30:2, pages 80-85.
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Julieta Lazarte & Robert A. Hegele. (2020) Dyslipidemia Management in Adults With Diabetes. Canadian Journal of Diabetes 44:1, pages 53-60.
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Latifah Alothman & Jacques Genest. (2019) Chylomicrons: When you can't direct the wind, adjust the sail. Atherosclerosis 283, pages 121-123.
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Anthony C. Keech & Alicia J. Jenkins. (2017) Triglyceride-lowering trials. Current Opinion in Lipidology 28:6, pages 477-487.
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Xin Liu, Peng Men, Yuhui Wang, Suodi Zhai, Zhigang Zhao & George Liu. (2017) Efficacy and Safety of Lomitapide in Hypercholesterolemia. American Journal of Cardiovascular Drugs 17:4, pages 299-309.
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