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Journal of Enzyme Inhibition Volume 16, 2001 - Issue 2
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Original Article

Carbonic Anhydrase Inhibitors, Interaction of Boron Derivatives with Isozymes I and II: A New Binding Site for Hydrophobic Inhibitors at the Entrance of the Active Site as shown by Docking Studies

Celine Chazalette Université Paul Sabatier, Laboratoire d'Hétérochimie Fondamentale el Appliquée, UMR 5069 du CNRS, 118 route de Narbonne, 31062 Toulouse CedexFrance; Università degli Studi di Firenze, Laboratorio di Chimka Inorganica e Bioinorganica, Via Gino Capponi 7, 1-50121, Florence, Italy
,
Monique Riviere-Baudet Université Paul Sabatier, Laboratoire d'Hétérochimie Fondamentale el Appliquée, UMR 5069 du CNRS, 118 route de Narbonne, 31062 Toulouse CedexFrance
,
Andrea Scozzafava Università degli Studi di Firenze, Laboratorio di Chimka Inorganica e Bioinorganica, Via Gino Capponi 7, 1-50121, Florence, Italy
,
Francesco Abbate Università degli Studi di Firenze, Laboratorio di Chimka Inorganica e Bioinorganica, Via Gino Capponi 7, 1-50121, Florence, Italy
,
Zahra Ben Maarouf Université Ibnou Zohr, Laboratoire de Chintie Organique et Organométallique, BP28S, Agadir, Monaco
&
Claudiu T. Supuran Università degli Studi di Firenze, Laboratorio di Chimka Inorganica e Bioinorganica, Via Gino Capponi 7, 1-50121, Florence, ItalyCorrespondence[email protected]
Pages 125-133 | Received 29 Jun 2000, Published online: 02 Jul 2010

Citations (13)

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Claudiu T. Supuran. (2017) Advances in structure-based drug discovery of carbonic anhydrase inhibitors. Expert Opinion on Drug Discovery 12:1, pages 61-88.
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Silvia Pastorekova, Seppo Parkkila, Jaromir Pastorek & Claudiu T. Supuran. (2004) Review Article. Journal of Enzyme Inhibition and Medicinal Chemistry 19:3, pages 199-229.
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MILAN REMKO & VLADIMÍR GARAJ. (2003) Thermodynamics of binding of Zn2+ to carbonic anhydrase inhibitors. Molecular Physics 101:15, pages 2357-2368.
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Claudiu T Supuran & Andrea Scozzafava. (2002) Applications of carbonic anhydrase inhibitors and activators in therapy. Expert Opinion on Therapeutic Patents 12:2, pages 217-242.
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Articles from other publishers (9)

Simone Giovannuzzi, Anna Nikitjuka, Bruna Rafaela Pereira Resende, Michael Smietana, Alessio Nocentini, Claudiu T. Supuran & Jean-Yves Winum. (2024) Boron-containing carbonic anhydrases inhibitors. Bioorganic Chemistry 143, pages 106976.
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Marion Boyet, Laurent Chabaud & Mathieu Pucheault. (2023) Recent Advances in the Synthesis of Borinic Acid Derivatives. Molecules 28:6, pages 2660.
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Vaida Linkuvienė, Asta Zubrienė, Elena Manakova, Vytautas Petrauskas, Lina Baranauskienė, Audrius Zakšauskas, Alexey Smirnov, Saulius Gražulis, John E. Ladbury & Daumantas Matulis. (2018) Thermodynamic, kinetic, and structural parameterization of human carbonic anhydrase interactions toward enhanced inhibitor design. Quarterly Reviews of Biophysics 51.
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Diego Amado Torres, Malar A. Azagarsamy & S. Thayumanavan. (2012) Supramolecular Displacement-Mediated Activation of a Silent Fluorescence Probe for Label-Free Ligand Screening. Journal of the American Chemical Society 134:17, pages 7235-7237.
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Milan Remko. (2010) Molecular structure, pKa, lipophilicity, solubility and absorption of biologically active aromatic and heterocyclic sulfonamides. Journal of Molecular Structure: THEOCHEM 944:1-3, pages 34-42.
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Rohit Tiwari, Kiran Mahasenan, Ryan Pavlovicz, Chenglong Li & Werner Tjarks. (2009) Carborane Clusters in Computational Drug Design: A Comparative Docking Evaluation Using AutoDock, FlexX, Glide, and Surflex. Journal of Chemical Information and Modeling 49:6, pages 1581-1589.
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Laure C. Bouchez, Māris Turks, Srinivas Reddy Dubbaka, Freddy Fonquerne, Cotinica Craita, Sylvain Laclef & Pierre Vogel. (2005) Sulfur dioxide mediated one-pot, four-component synthesis of polyfunctional sulfones and sulfonamides, including medium-ring cyclic derivatives. Tetrahedron 61:48, pages 11473-11487.
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C. Chazalette, A. Khallaayoun, M. Rivière‐Baudet & F. El Baz. (2003) N ‐Germyl derivatives of sulfacetamide and ortho ‐(sulfonamido)phenylamines: characterization of N ‐[ o ‐( N ′, N ′‐dimethylsulfonamido)phenyl]‐ N ‐dimesitylgermaimine . Applied Organometallic Chemistry 17:3, pages 181-190.
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Milan Remko. (2003) Theoretical Study of Molecular Structure and Gas-Phase Acidity of Some Biologically Active Sulfonamides. The Journal of Physical Chemistry A 107:5, pages 720-725.
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