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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 31, 2016 - Issue sup1
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Research Article

1-(5-Carboxyindazol-1-yl)propan-2-ones as dual inhibitors of cytosolic phospholipase A2α and fatty acid amide hydrolase: bioisosteric replacement of the carboxylic acid moiety

Jan AlthausInstitute of Pharmaceutical and Medicinal Chemistry, University of Münster, Germany
,
Theresa HakeInstitute of Pharmaceutical and Medicinal Chemistry, University of Münster, Germany
,
Walburga HanekampInstitute of Pharmaceutical and Medicinal Chemistry, University of Münster, Germany
&
Matthias LehrInstitute of Pharmaceutical and Medicinal Chemistry, University of Münster, GermanyCorrespondence[email protected]
Pages 131-140 | Received 27 Jan 2016, Accepted 25 Mar 2016, Published online: 09 May 2016

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Domenico Fazio, Emanuele Criscuolo, Alessandra Piccoli, Barbara Barboni, Filomena Fezza & Mauro Maccarrone. (2020) Advances in the discovery of fatty acid amide hydrolase inhibitors: what does the future hold?. Expert Opinion on Drug Discovery 15:7, pages 765-778.
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Articles from other publishers (6)

Shakila Ghomashi, Reihane Ghomashi, Hamidreza Aghaei & Ahmad Reza Massah. (2023) Recent Advances in Biological Active Sulfonamide based Hybrid Compounds Part B: Two-Component Sulfonamide Hybrids. Current Medicinal Chemistry 30:5, pages 604-665.
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Karolina Dzedulionytė, Melita Veikšaitė, Vít Morávek, Vida Malinauskienė, Greta Račkauskienė, Algirdas Šačkus, Asta Žukauskaitė & Eglė Arbačiauskienė. (2022) Convenient Synthesis of N-Heterocycle-Fused Tetrahydro-1,4-Diazepinones. Molecules 27:24, pages 8666.
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Paweł Kozyra & Monika Pitucha. (2022) Terminal Phenoxy Group as a Privileged Moiety of the Drug Scaffold—A Short Review of Most Recent Studies 2013–2022. International Journal of Molecular Sciences 23:16, pages 8874.
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Rati Kailash Prasad Tripathi. (2020) A perspective review on fatty acid amide hydrolase (FAAH) inhibitors as potential therapeutic agents. European Journal of Medicinal Chemistry 188, pages 111953.
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Aikaterini Nikolaou, Maroula G. Kokotou, Sofia Vasilakaki & George Kokotos. (2019) Small-molecule inhibitors as potential therapeutics and as tools to understand the role of phospholipases A2. Biochimica et Biophysica Acta (BBA) - Molecular and Cell Biology of Lipids 1864:6, pages 941-956.
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Frederik Diness, Niels J Bjerrum & Mikael Begtrup. (2018) Synthesis and stability of strongly acidic benzamide derivatives. Beilstein Journal of Organic Chemistry 14, pages 523-530.
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