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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 32, 2017 - Issue 1
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Research Paper

Design, synthesis and evaluation of 2-aryl benzoxazoles as promising hit for the A2A receptor

Romain DurouxINSERM, CHU Lille, UMR-S 1172 – JPArc – Centre de Recherche Jean-Pierre AUBERT Neurosciences et Cancer, Universite de Lille, Lille, France;
,
Nicolas RenaultINSERM, CHU Lille, U995 – LIRIC – Lille Inflammation Research International Center, Universite de Lille, Lille, France;
,
Joana Esteves CuelhoInstituto de Medecina Molecular, Lisbon, Portugal
,
Laurence AgouridasINSERM, CHU Lille, UMR-S 1172 – JPArc – Centre de Recherche Jean-Pierre AUBERT Neurosciences et Cancer, Universite de Lille, Lille, France;
,
David BlumINSERM, CHU Lille, UMR-S 1172 – JPArc – Centre de Recherche Jean-Pierre AUBERT Neurosciences et Cancer, Universite de Lille, Lille, France;
,
Luisa V. LopesInstituto de Medecina Molecular, Lisbon, Portugal
,
Patricia MelnykINSERM, CHU Lille, UMR-S 1172 – JPArc – Centre de Recherche Jean-Pierre AUBERT Neurosciences et Cancer, Universite de Lille, Lille, France;
&
Saïd YousINSERM, CHU Lille, UMR-S 1172 – JPArc – Centre de Recherche Jean-Pierre AUBERT Neurosciences et Cancer, Universite de Lille, Lille, France; Correspondence[email protected]
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Pages 850-864 | Received 24 Mar 2017, Accepted 18 May 2017, Published online: 29 Jun 2017

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Zhi Li, Lijuan Kou, Xinzhen Fu, Zeping Xie, Maolei Xu, Lin Guo, Tiantian Lin, Shizhou Gong, Shumin Zhang & Ming Liu. (2022) Design, synthesis, and biological evaluation of triazole-pyrimidine-methylbenzonitrile derivatives as dual A2A/A2B adenosine receptor antagonists. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 1514-1526.
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Anjali Saini, Rajiv Patel, Sobhi Gaba, Gurpreet Singh, G.D. Gupta & Vikramdeep Monga. (2022) Adenosine receptor antagonists: Recent advances and therapeutic perspective. European Journal of Medicinal Chemistry 227, pages 113907.
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Zhihai Ke & Ying-Yeung Yeung. 2022. Comprehensive Heterocyclic Chemistry IV. Comprehensive Heterocyclic Chemistry IV 412 449 .
Nicolae Baranov, Stefania Racovita, Silvia Vasiliu, Ana Maria Macsim, Catalina Lionte, Valeriu Sunel, Marcel Popa, Jacques Desbrieres & Corina Cheptea. (2021) Immobilization and Release Studies of Triazole Derivatives from Grafted Copolymer Based on Gellan-Carrying Betaine Units. Molecules 26:11, pages 3330.
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Niranjan Panda & Kanchanbala Sahoo. (2018) Synthesis of 4‐Alkenyl Benzoxazoles via Pd‐catalyzed ortho C−H Functionalization of 2‐Amidophenols . Advanced Synthesis & Catalysis 361:3, pages 617-627.
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Yun-Xin Yao, Nan-Nan Jia, Ya-Nan Cao, Xing-Xiu Chen, Feng Gao & Xiao-Xia Liang. (2018) Copper-Catalyzed Synthesis, Bio-Evaluation, and in Silico Studies of 2-Aryl-N-alkylbenzimidazoles as Neuroprotective Agents. Catalysts 8:10, pages 433.
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Rajaa Boulahjar, Angela Rincon Arias, Raphaël Bolteau, Nicolas Renault, Mathilde Coevoet, Amélie Barczyk, Romain Duroux, Saïd Yous, Patricia Melnyk & Laurence Agouridas. (2018) Design and synthesis of 2,6-disubstituted-8-amino imidazo[1,2a]pyridines, a promising privileged structure. Bioorganic & Medicinal Chemistry 26:12, pages 3296-3307.
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Romain Duroux, Laurence Agouridas, Nicolas Renault, Jamal El Bakali, Christophe Furman, Patricia Melnyk & Saïd Yous. (2018) Antagonists of the adenosine A 2A receptor based on a 2-arylbenzoxazole scaffold: Investigation of the C5- and C7-positions to enhance affinity. European Journal of Medicinal Chemistry 144, pages 151-163.
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