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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 34, 2019 - Issue 1
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Short Communication

Computationally driven discovery of phenyl(piperazin-1-yl)methanone derivatives as reversible monoacylglycerol lipase (MAGL) inhibitors

Giulio PoliDepartment of Pharmacy, University of Pisa, Pisa, Italy; View further author information
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Margherita LapilloDepartment of Pharmacy, University of Pisa, Pisa, Italy; View further author information
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Vibhu JhaDepartment of Pharmacy, University of Pisa, Pisa, Italy; View further author information
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Nayla MouawadDepartment of Pharmacy, University of Pisa, Pisa, Italy; ;Pathology Unit, Department of Molecular Biology and Translational Research, National Cancer Institute and Center for Molecular Biomedicine, Aviano, Italy; View further author information
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Isabella CaligiuriPathology Unit, Department of Molecular Biology and Translational Research, National Cancer Institute and Center for Molecular Biomedicine, Aviano, Italy; View further author information
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Marco MacchiaDepartment of Pharmacy, University of Pisa, Pisa, Italy; View further author information
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Filippo MinutoloDepartment of Pharmacy, University of Pisa, Pisa, Italy; ORCID Iconhttp://orcid.org/0000-0002-3312-104XView further author information
ORCID Icon,
Flavio RizzolioPathology Unit, Department of Molecular Biology and Translational Research, National Cancer Institute and Center for Molecular Biomedicine, Aviano, Italy; ;Department of Molecular Science and Nanosystems, Ca' Foscari Università di Venezia, Venezia, Italy; ORCID Iconhttp://orcid.org/0000-0002-3400-4363View further author information
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Tiziano TuccinardiDepartment of Pharmacy, University of Pisa, Pisa, Italy; Correspondence[email protected]
ORCID Iconhttp://orcid.org/0000-0002-6205-4069View further author information
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Carlotta GranchiDepartment of Pharmacy, University of Pisa, Pisa, Italy; ;Sbarro Institute for Cancer Research and Molecular Medicine, Center for Biotechnology, College of Science and Technology, Temple University, Philadelphia, PA, USAORCID Iconhttp://orcid.org/0000-0002-5849-0722View further author information
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Pages 589-596 | Received 02 Nov 2018, Accepted 28 Dec 2018, Published online: 30 Jan 2019

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Giulia Bononi, Giulio Poli, Flavio Rizzolio, Tiziano Tuccinardi, Marco Macchia, Filippo Minutolo & Carlotta Granchi. (2021) An updated patent review of monoacylglycerol lipase (MAGL) inhibitors (2018-present). Expert Opinion on Therapeutic Patents 31:2, pages 153-168.
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