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Tarek S. Ibrahim, Amr H. Moustafa, Ahmad J. Almalki, Rasha M. Allam, Abdulhamid Althagafi, Shadab Md & Mamdouh F. A. Mohamed. (2021) Novel chalcone/aryl carboximidamide hybrids as potent anti-inflammatory via inhibition of prostaglandin E2 and inducible NO synthase activities: design, synthesis, molecular docking studies and ADMET prediction. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 1067-1078.
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Yang Li, Ying Sun, Yang Zhou, Xinyang Li, Huan Zhang & Guojun Zhang. (2021) Discovery of orally active chalcones as histone lysine specific demethylase 1 inhibitors for the treatment of leukaemia. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 207-217.
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Emilio Guillén-Mancina, María del Rosario García-Lozano, Estefanía Burgos-Morón, Sarah Mazzotta, Pablo Martínez-Aguado, José Manuel Calderón-Montaño, José Manuel Vega-Pérez, Miguel López-Lázaro, Fernando Iglesias-Guerra & Margarita Vega-Holm. (2023) Repurposing Study of 4-Acyl-1-phenylaminocarbonyl-2-substituted-piperazine Derivatives as Potential Anticancer Agents—In Vitro Evaluation against Breast Cancer Cells. International Journal of Molecular Sciences 24:23, pages 17041.
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Najla Altwaijry, Rehab Sabour, Mona H. Ibrahim, Omkulthom Al kamaly, Omeima Abdullah & Marwa F. Harras. (2023) Design, synthesis, and anti-hepatocellular carcinoma of thiopyrimidine/chalcone hybrids as dual STAT3/STAT5 inhibitors. RSC Medicinal Chemistry 14:10, pages 1981-1991.
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Jiahui Yang, Jianmei Lv, Shuxian Cheng, Tingyu Jing, Tenghao Meng, Dezhen Huo, Xin Ma & Ran Wen. (2023) Recent Progresses in Chalcone Derivatives as Potential Anticancer Agents. Anti-Cancer Agents in Medicinal Chemistry 23:11, pages 1265-1283.
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Jiatao Song, Jiawei Wang, Sheng Tian & Huanqiu Li. (2023) Discovery of STAT3 Inhibitors: Recent Advances and Future Perspectives. Current Medicinal Chemistry 30:16, pages 1824-1847.
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María del Rosario García-Lozano, Filippo Dragoni, Paloma Gallego, Sarah Mazzotta, Alejandro López-Gómez, Adele Boccuto, Carlos Martínez-Cortés, Alejandro Rodríguez-Martínez, Horacio Pérez-Sánchez, José Manuel Vega-Pérez, José Antonio Del Campo, Ilaria Vicenti, Margarita Vega-Holm & Fernando Iglesias-Guerra. (2023) Piperazine-derived small molecules as potential Flaviviridae NS3 protease inhibitors. In vitro antiviral activity evaluation against Zika and Dengue viruses. Bioorganic Chemistry 133, pages 106408.
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Nicole D. Bartolo, Niall Mortimer, Mariah A. Manter, Nicholas Sanchez, Misha Riley, Tiernan T. O’Malley & Jacob M. Hooker. (2022) Identification and Prioritization of PET Neuroimaging Targets for Microglial Phenotypes Associated with Microglial Activity in Alzheimer’s Disease. ACS Chemical Neuroscience 13:24, pages 3641-3660.
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Tung H. To, Dang B. Tran, Thang C. Pham & Phong D. Tran. (2022) A new approach to pyrimidine-type heterocycles based on Petrenko–Kritschenko synthesis. Chemistry of Heterocyclic Compounds 58:11, pages 608-614.
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Khaled R.A. Abdellatif, Eman K.A. Abdelall, Phoebe F. Lamie, Madlen B. Labib, Marwa M. Abdelhakeem, Maha M. Abdel-Fattah & El-Shaymaa El-Nahaas. (2022) Novel pyrazole-oxadiazole hybrids possessing methanesulphonyl pharmacophore with good gastric safety profile: Design, synthesis, cyclooxygenase inhibition, anti-inflammatory activity and histopathological studies. Journal of Molecular Structure 1266, pages 133529.
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S. M. Mohammed, A. H. Moustafa, H. A. El-Sayed, A. S. Amin, A. Haggar, E. S. Tantawy & R. A. Haggam. (2022) A New Approach for Synthesis of 2-Thioxocytosine-5-carbonitrile as Antimicrobial Agents. Russian Journal of General Chemistry 92:9, pages 1806-1813.
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Ekaterina V. Neborak, Altynay B. Kaldybayeva, Lylia Bey, Aigul Y. Malmakova, Anna S. Tveritinova, Abdullah Hilal, Valentina K. Yu, Maria V. Ploskonos, Marina V. Komarova, Enzo Agostinelli & Dmitry D. Zhdanov. (2022) Anticancer Cytotoxic Activity of Bispidine Derivatives Associated with the Increasing Catabolism of Polyamines. Molecules 27:12, pages 3872.
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Khaled R.A. Abdellatif, Eman K.A. Abdelall, Heba A.H. Elshemy, John N. Philoppes, Emad H.M. Hassanein & Nesma M. Kahk. (2022) Design, synthesis, and pharmacological evaluation of novel and selective COX-2 inhibitors based on celecoxib scaffold supported with in vivo anti-inflammatory activity, ulcerogenic liability, ADME profiling and docking study. Bioorganic Chemistry 120, pages 105627.
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Ghada M. Safwat, Kamel M. A. Hassanin, Eman T. Mohammed, Essam Kh. Ahmed, Mahmoud R. Abdel Rheim, Mohamed A. Ameen, Mohamed Abdel-Aziz, Ahmed M. Gouda, Ilaria Peluso, Rafa Almeer, Mohamed M. Abdel-Daim & Ahmed Abdel-Wahab. (2021) Synthesis, Anticancer Assessment, and Molecular Docking of Novel Chalcone-Thienopyrimidine Derivatives in HepG2 and MCF-7 Cell Lines. Oxidative Medicine and Cellular Longevity 2021, pages 1-27.
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Jeelan Basha N & Naganna M. Goudgaon. (2021) A comprehensive review on pyrimidine analogs-versatile scaffold with medicinal and biological potential. Journal of Molecular Structure 1246, pages 131168.
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Khaled R.A. Abdellatif, Eman K.A. Abdelall, Heba A.H. Elshemy, John N. Philoppes, Emad H.M. Hassanein & Nesma M. Kahk. (2021) Optimization of pyrazole-based compounds with 1,2,4-triazole-3-thiol moiety as selective COX-2 inhibitors cardioprotective drug candidates: Design, synthesis, cyclooxygenase inhibition, anti-inflammatory, ulcerogenicity, cardiovascular evaluation, and molecular modeling studies. Bioorganic Chemistry 114, pages 105122.
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Sarah Mazzotta, Judith Berastegui-Cabrera, Margarita Vega-Holm, María del Rosario García-Lozano, Marta Carretero-Ledesma, Francesca Aiello, José Manuel Vega-Pérez, Jerónimo Pachón, Fernando Iglesias-Guerra & Javier Sánchez-Céspedes. (2021) Design, synthesis and in vitro biological evaluation of a novel class of anti-adenovirus agents based on 3-amino-1,2-propanediol. Bioorganic Chemistry 114, pages 105095.
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Jinyun Dong, Xiang-Dong Cheng, Wei-Dong Zhang & Jiang-Jiang Qin. (2021) Recent Update on Development of Small-Molecule STAT3 Inhibitors for Cancer Therapy: From Phosphorylation Inhibition to Protein Degradation. Journal of Medicinal Chemistry 64:13, pages 8884-8915.
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Tarek S. Ibrahim, Ahmad J. Almalki, Amr H. Moustafa, Rasha M. Allam, Gamal El-Din A. Abuo-Rahma, Hussein I. El Subbagh & Mamdouh F.A. Mohamed. (2021) Novel 1,2,4-oxadiazole-chalcone/oxime hybrids as potential antibacterial DNA gyrase inhibitors: Design, synthesis, ADMET prediction and molecular docking study. Bioorganic Chemistry 111, pages 104885.
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Saba Farooq & Zainab Ngaini. (2021)
One‐pot
and
two‐pot
methods for chalcone derived pyrimidines synthesis and applications
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