Advanced search
Publication Cover
Journal of Enzyme Inhibition and Medicinal Chemistry Volume 35, 2020 - Issue 1
Submit an article Journal homepage
1,618
Views
7
CrossRef citations to date
0
Altmetric
Research Paper

Imidazopyridine-fused [1,3]diazepinones: modulations of positions 2 to 4 and their impacts on the anti-melanoma activity

Paul Le Baccon-Solliera Institut des Biomolécules Max Mousseron, UMR 5247, CNRS, Universités Montpellier, UFR des Sciences Pharmaceutiques et Biologiques, Montpellier, FranceView further author information
,
Yohan Malkia Institut des Biomolécules Max Mousseron, UMR 5247, CNRS, Universités Montpellier, UFR des Sciences Pharmaceutiques et Biologiques, Montpellier, FranceView further author information
,
Morgane Mayea Institut des Biomolécules Max Mousseron, UMR 5247, CNRS, Universités Montpellier, UFR des Sciences Pharmaceutiques et Biologiques, Montpellier, FranceView further author information
,
Lamiaa M. A. Alia Institut des Biomolécules Max Mousseron, UMR 5247, CNRS, Universités Montpellier, UFR des Sciences Pharmaceutiques et Biologiques, Montpellier, France;b Department of Biochemistry, Medical Research Institute, University of Alexandria, Alexandria, EgyptORCID Iconhttps://orcid.org/0000-0003-1176-5335View further author information
ORCID Icon,
Laure Lichona Institut des Biomolécules Max Mousseron, UMR 5247, CNRS, Universités Montpellier, UFR des Sciences Pharmaceutiques et Biologiques, Montpellier, FranceView further author information
,
Pierre Cuqa Institut des Biomolécules Max Mousseron, UMR 5247, CNRS, Universités Montpellier, UFR des Sciences Pharmaceutiques et Biologiques, Montpellier, FranceORCID Iconhttps://orcid.org/0000-0002-5440-9165View further author information
ORCID Icon,
Laure-Anaïs Vincenta Institut des Biomolécules Max Mousseron, UMR 5247, CNRS, Universités Montpellier, UFR des Sciences Pharmaceutiques et Biologiques, Montpellier, FranceORCID Iconhttps://orcid.org/0000-0003-3613-859XView further author information
ORCID Icon &
Nicolas Masuriera Institut des Biomolécules Max Mousseron, UMR 5247, CNRS, Universités Montpellier, UFR des Sciences Pharmaceutiques et Biologiques, Montpellier, FranceCorrespondence[email protected]
ORCID Iconhttps://orcid.org/0000-0001-9169-8149View further author information
ORCID Icon show all
Pages 935-949 | Received 23 Dec 2019, Accepted 22 Mar 2020, Published online: 05 Apr 2020

Citations (7)

Keep up to date with the latest research on this topic with citation updates for this article.

Subscribe to citation updates

Read on this site (1)

Hesham Haffez, Nosaiba A. Elsayed, Marwa F. Ahmed, Samar S. Fatahala, Eman F. Khaleel, Rehab Mustafa Badi, Eslam B. Elkaeed, Mahmoud A. El Hassab, Sherif F. Hammad, Wagdy M. Eldehna, Nicolas Masurier & Radwan El-Haggar. (2023) Novel N-Arylmethyl-aniline/chalcone hybrids as potential VEGFR inhibitors: synthesis, biological evaluations, and molecular dynamic simulations. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1.
Read now

Articles from other publishers (6)

Marwa F. Ahmed, Radwan El‐Haggar, Atiah H. Almalki, Omeima Abdullah, Mahmoud A. El Hassab, Nicolas Masurier & Sherif F. Hammad. (2023) Novel hydrazone‐isatin derivatives as potential EGFR inhibitors: Synthesis and in vitro pharmacological profiling. Archiv der Pharmazie 356:9.
Crossref
Rajeswari Kannuri, Shireesha Manturthi, Venkanna Muripiti & Amar nath Velidandi. (2023) Tin Chloride Mediated Grinding Method for Preparation of 2,4-Disubstituted Benzodiazepine Scaffolds Their In Silico, and In Vitro Cell Viability Studies. Russian Journal of Bioorganic Chemistry 49:3, pages 682-688.
Crossref
Yohan Malki, Ludovic T. Maillard & Nicolas Masurier. (2021) 1,3‐Diazepine Derivatives: Strategies for Synthesis. European Journal of Organic Chemistry 2022:21.
Crossref
Yohan Malki, Jean Martinez & Nicolas Masurier. (2021) 1,3‐Diazepine: A privileged scaffold in medicinal chemistry. Medicinal Research Reviews 41:4, pages 2247-2315.
Crossref
Koceïla Doufène, Yohan Malki, Laure-Anaïs Vincent, Pierre Cuq, Jean-Marie Devoisselle, Nicolas Masurier & Anne Aubert-Pouëssel. (2021) Vegetable Oil-based Hybrid Submicron Particles Loaded with JMV5038: A Promising Formulation against Melanoma. Journal of Pharmaceutical Sciences 110:3, pages 1197-1205.
Crossref
Anthony Feral, Guillaume Laconde, Muriel Amblard & Nicolas Masurier. (2020) PROteolysis TArgetting Chimeras (PROTACs) Strategy Applied to Kinases: Recent Advances. Advanced Therapeutics 3:11.
Crossref

Related research

People also read lists articles that other readers of this article have read.

Recommended articles lists articles that we recommend and is powered by our AI driven recommendation engine.

Cited by lists all citing articles based on Crossref citations.
Articles with the Crossref icon will open in a new tab.