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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 37, 2022 - Issue 1
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Brief Report

First studies on tumor associated carbonic anhydrases IX and XII monoclonal antibodies conjugated to small molecule inhibitors

Chiara Testaa Interdepartmental Research Unit of Peptide and Protein Chemistry and Biology”, Department of Chemistry “Ugo Schiff”, University of Florence, Sesto Fiorentino, ItalyView further author information
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Anna Maria Papinia Interdepartmental Research Unit of Peptide and Protein Chemistry and Biology”, Department of Chemistry “Ugo Schiff”, University of Florence, Sesto Fiorentino, ItalyORCID Iconhttps://orcid.org/0000-0002-2947-7107View further author information
ORCID Icon,
Reinhard Zeidlerb Research Group Therapeutic Antibodies, Helmholtz Centre Munich German Research Centre for Environmental Health, Munich, Germany;c Department of Otorhinolaryngology, Klinikum der Universitaet, Munich, GermanyView further author information
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Daniela Vullod NEUROFARBA Dept., Sezione di Scienze Farmaceutiche e Nutraceutiche, University of Florence, via Ugo Schff 6, Sesto Fiorentino (Florence), 50019ItalyView further author information
,
Fabrizio Cartad NEUROFARBA Dept., Sezione di Scienze Farmaceutiche e Nutraceutiche, University of Florence, via Ugo Schff 6, Sesto Fiorentino (Florence), 50019ItalyCorrespondence[email protected]
ORCID Iconhttps://orcid.org/0000-0002-1141-6146View further author information
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Claudiu T. Supurand NEUROFARBA Dept., Sezione di Scienze Farmaceutiche e Nutraceutiche, University of Florence, via Ugo Schff 6, Sesto Fiorentino (Florence), 50019ItalyORCID Iconhttps://orcid.org/0000-0003-4262-0323View further author information
ORCID Icon &
Paolo Roveroa Interdepartmental Research Unit of Peptide and Protein Chemistry and Biology”, Department of Chemistry “Ugo Schiff”, University of Florence, Sesto Fiorentino, ItalyCorrespondence[email protected]
ORCID Iconhttps://orcid.org/0000-0001-9577-5228View further author information
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Pages 592-596 | Received 13 Oct 2021, Accepted 04 Nov 2021, Published online: 20 Jan 2022

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Claudiu T Supuran. (2023) Targeting carbonic anhydrases for the management of hypoxic metastatic tumors. Expert Opinion on Therapeutic Patents 0:0, pages 1-20.
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Alessandro Bonardi, Silvia Bua, Jacob Combs, Carrie Lomelino, Jacob Andring, Sameh Mohamed Osman, Alessandra Toti, Lorenzo Di Cesare Mannelli, Paola Gratteri, Carla Ghelardini, Robert McKenna, Alessio Nocentini & Claudiu T. Supuran. (2022) The three-tails approach as a new strategy to improve selectivity of action of sulphonamide inhibitors against tumour-associated carbonic anhydrase IX and XII. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 930-939.
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Mateusz Kciuk, Adrianna Gielecińska, Somdutt Mujwar, Mariusz Mojzych, Beata Marciniak, Rafał Drozda & Renata Kontek. (2022) Targeting carbonic anhydrase IX and XII isoforms with small molecule inhibitors and monoclonal antibodies. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 1278-1298.
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Alane Beatriz Vermelho, Giseli Capaci Rodrigues, Alessio Nocentini, Felipe R. P. Mansoldo & Claudiu T. Supuran. (2022) Discovery of novel drugs for Chagas disease: is carbonic anhydrase a target for antiprotozoal drugs?. Expert Opinion on Drug Discovery 17:10, pages 1147-1158.
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Sridhar Goud Nerella, Priti Singh, Mohammed Arifuddin & Claudiu T Supuran. (2022) Anticancer carbonic anhydrase inhibitors: a patent and literature update 2018-2022. Expert Opinion on Therapeutic Patents 32:8, pages 833-847.
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Articles from other publishers (7)

Toni C. Denner, Niels Heise, Julian Zacharias, Oliver Kraft, Sophie Hoenke & René Csuk. (2023) Small Structural Differences Govern the Carbonic Anhydrase II Inhibition Activity of Cytotoxic Triterpene Acetazolamide Conjugates. Molecules 28:3, pages 1009.
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Jacob Combs, Murat Bozdag, Lochlin D. Cravey, Anusha Kota, Robert McKenna, Andrea Angeli, Fabrizio Carta & Claudiu T. Supuran. (2023) New Insights into Conformationally Restricted Carbonic Anhydrase Inhibitors. Molecules 28:2, pages 890.
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Laura Braconi, Elisabetta Teodori, Chiara Riganti, Marcella Coronnello, Alessio Nocentini, Gianluca Bartolucci, Marco Pallecchi, Marialessandra Contino, Dina Manetti, Maria Novella Romanelli, Claudiu T. Supuran & Silvia Dei. (2022) New Dual P-Glycoprotein (P-gp) and Human Carbonic Anhydrase XII (hCA XII) Inhibitors as Multidrug Resistance (MDR) Reversers in Cancer Cells. Journal of Medicinal Chemistry 65:21, pages 14655-14672.
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Lisa Hiepp, Doris Mayr, Kathrin Gärtner, Elisa Schmoeckel, Frederick Klauschen, Alexander Burges, Sven Mahner, Reinhard Zeidler & Bastian Czogalla. (2022) Carbonic anhydrase XII as biomarker and therapeutic target in ovarian carcinomas. PLOS ONE 17:7, pages e0271630.
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Paul C. McDonald, Shawn C. Chafe, Claudiu T. Supuran & Shoukat Dedhar. (2022) Cancer Therapeutic Targeting of Hypoxia Induced Carbonic Anhydrase IX: From Bench to Bedside. Cancers 14:14, pages 3297.
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Murat Bozdag, Lochlin Cravey, Jacob Combs, Anusha Kota, Robert McKenna, Andrea Angeli, Silvia Selleri, Fabrizio Carta & Claudiu T. Supuran. (2022) Small Molecule Alkoxy Oriented Selectiveness on Human Carbonic Anhydrase II and IX Inhibition. ChemMedChem 17:11.
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Dimitrios Tsikas. (2022) Editorial. Amino Acids 54:4, pages 481-484.
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