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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 37, 2022 - Issue 1
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Research Paper

4-Anilinoquinazoline-based benzenesulfonamides as nanomolar inhibitors of carbonic anhydrase isoforms I, II, IX, and XII: design, synthesis, in-vitro, and in-silico biological studies

Hossam Nadaa BK21 FOUR Team and Integrated Research Institute for Drug Development, College of Pharmacy, Dongguk University-Seoul, Goyang, Republic of KoreaORCID Iconhttps://orcid.org/0000-0002-4882-5621View further author information
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Ahmed Elkamhawya BK21 FOUR Team and Integrated Research Institute for Drug Development, College of Pharmacy, Dongguk University-Seoul, Goyang, Republic of Korea;b Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura, EgyptORCID Iconhttps://orcid.org/0000-0001-7398-6155View further author information
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Magda H. Abdellattifc Department of Chemistry, College of Science, Taif University, Taif, Saudi ArabiaORCID Iconhttps://orcid.org/0000-0002-8562-4749View further author information
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Andrea Angelid NEUROFARBA Department, Sezione di Scienze Farmaceutiche, University of Florence, Sesto Fiorentino, Florence, ItalyORCID Iconhttps://orcid.org/0000-0002-1470-7192View further author information
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Chang Hoon Leea BK21 FOUR Team and Integrated Research Institute for Drug Development, College of Pharmacy, Dongguk University-Seoul, Goyang, Republic of KoreaView further author information
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Claudiu T. Supurand NEUROFARBA Department, Sezione di Scienze Farmaceutiche, University of Florence, Sesto Fiorentino, Florence, ItalyORCID Iconhttps://orcid.org/0000-0003-4262-0323View further author information
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Kyeong Leea BK21 FOUR Team and Integrated Research Institute for Drug Development, College of Pharmacy, Dongguk University-Seoul, Goyang, Republic of KoreaCorrespondence[email protected]
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Pages 994-1004 | Received 17 Nov 2021, Accepted 11 Mar 2022, Published online: 30 Mar 2022

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Zainab M. Elsayed, Hadia Almahli, Alessio Nocentini, Andrea Ammara, Claudiu T. Supuran, Wagdy M. Eldehna & Sahar M. Abou-Seri. (2023) Development of novel anilinoquinazoline-based carboxylic acids as non-classical carbonic anhydrase IX and XII inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1.
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Khulood H. Oudah, Walaa R. Mahmoud, Fadi M. Awadallah, Azza T. Taher, Safinaz E.-S Abbas, Heba Abdelrasheed Allam, Daniela Vullo & Claudiu T. Supuran. (2023) Design and synthesis of some new benzoylthioureido benzenesulfonamide derivatives and their analogues as carbonic anhydrase inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1, pages 12-23.
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H.E. Bostancı, U.A. Çevik, R. Kapavarapu, Y.C. Güldiken, Z.D.Ş. Inan, Ö.Ö. Güler, T.K. Uysal, A. Uytun, F.N. Çetin, Y. Özkay & Z.A. Kaplancıklı. (2023) Synthesis, biological evaluation and in silico studies of novel thiadiazole-hydrazone derivatives for carbonic anhydrase inhibitory and anticancer activities. SAR and QSAR in Environmental Research 34:7, pages 543-567.
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Articles from other publishers (5)

Sertan Aytac, Ozlem Gundogdu, Zeynebe Bingol & İlhami Gulcin. (2023) Synthesis of Schiff Bases Containing Phenol Rings and Investigation of Their Antioxidant Capacity, Anticholinesterase, Butyrylcholinesterase, and Carbonic Anhydrase Inhibition Properties. Pharmaceutics 15:3, pages 779.
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Zahid Hussain, Abid Mahmood, Qasim Shah, Aqeel Imran, Ehsan Ullah Mughal, Wajiha Khan, Ayesha Baig, Jamshed Iqbal & Amara Mumtaz. (2022) Synthesis and Evaluation of Amide and Thiourea Derivatives as Carbonic Anhydrase (CA) Inhibitors. ACS Omega 7:50, pages 47251-47264.
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Heba T. Abdel‐Mohsen, Mohamed A. Omar, Andrea Petreni & Claudiu T. Supuran. (2022) Novel 2‐substituted thioquinazoline‐benzenesulfonamide derivatives as carbonic anhydrase inhibitors with potential anticancer activity. Archiv der Pharmazie 355:12.
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Hossam Nada, Ahmed Elkamhawy & Kyeong Lee. (2022) Identification of 1H-purine-2,6-dione derivative as a potential SARS-CoV-2 main protease inhibitor: molecular docking, dynamic simulations, and energy calculations. PeerJ 10, pages e14120.
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Phuong Linh Nguyen, Ahmed Elkamhawy, Young Hee Choi, Chang Hoon Lee, Kyeong Lee & Jungsook Cho. (2022) Suppression of Tumor Growth and Cell Migration by Indole-Based Benzenesulfonamides and Their Synergistic Effects in Combination with Doxorubicin. International Journal of Molecular Sciences 23:17, pages 9903.
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