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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 37, 2022 - Issue 1
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Research Papers

Novel 3-(6-methylpyridin-2-yl)coumarin-based chalcones as selective inhibitors of cancer-related carbonic anhydrases IX and XII endowed with anti-proliferative activity

Haytham O. Tawfika Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Tanta University, Tanta, EgyptORCID Iconhttps://orcid.org/0000-0001-6455-5716View further author information
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Moataz A. Shaldamb Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, EgyptORCID Iconhttps://orcid.org/0000-0002-0420-4364View further author information
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Alessio Nocentinic Section of Pharmaceutical and Nutraceutical Sciences, Department of NEUROFARBA, University of Florence, Polo Scientifico, Firenze, ItalyORCID Iconhttps://orcid.org/0000-0003-3342-702XView further author information
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Rofaida Salemb Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, EgyptView further author information
,
Hadia Almahlid Department of Chemistry, University of Cambridge, Cambridge, UKView further author information
,
Sara T. Al-Rashoode Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, Riyadh, Saudi ArabiaView further author information
,
Claudiu T. Supuranc Section of Pharmaceutical and Nutraceutical Sciences, Department of NEUROFARBA, University of Florence, Polo Scientifico, Firenze, ItalyCorrespondence[email protected]
ORCID Iconhttps://orcid.org/0000-0003-4262-0323View further author information
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Wagdy M. Eldehnab Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, EgyptCorrespondence[email protected]
ORCID Iconhttps://orcid.org/0000-0001-6996-4017View further author information
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Pages 1043-1052 | Received 22 Feb 2022, Accepted 18 Mar 2022, Published online: 19 Apr 2022

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Zainab M. Elsayed, Hadia Almahli, Alessio Nocentini, Andrea Ammara, Claudiu T. Supuran, Wagdy M. Eldehna & Sahar M. Abou-Seri. (2023) Development of novel anilinoquinazoline-based carboxylic acids as non-classical carbonic anhydrase IX and XII inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1.
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Shaik Mahammad Ghouse, Kavyaraj Bahatam, Andrea Angeli, Gaurav Pawar, Krishna Kartheek Chinchilli, Venkata Madhavi Yaddanapudi, Arifuddin Mohammed, Claudiu T. Supuran & Srinivas Nanduri. (2023) Synthesis and biological evaluation of new 3-substituted coumarin derivatives as selective inhibitors of human carbonic anhydrase IX and XII. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1.
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Jekaterīna Ivanova, Morteza Abdoli, Alessio Nocentini, Raivis Žalubovskis & Claudiu T. Supuran. (2023) Derivatives of 4-methyl-1,2,3-benzoxathiazine 2,2-dioxide as selective inhibitors of human carbonic anhydrases IX and XII over the cytosolic isoforms I and II. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1.
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Jekaterina Ivanova, Morteza Abdoli, Alessio Nocentini, Raivis Žalubovskis & Claudiu T. Supuran. (2023) 1,2,3-Benzoxathiazine-2,2-dioxides – effective inhibitors of human carbonic anhydrases. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1, pages 225-238.
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H.E. Bostancı, U.A. Çevik, R. Kapavarapu, Y.C. Güldiken, Z.D.Ş. Inan, Ö.Ö. Güler, T.K. Uysal, A. Uytun, F.N. Çetin, Y. Özkay & Z.A. Kaplancıklı. (2023) Synthesis, biological evaluation and in silico studies of novel thiadiazole-hydrazone derivatives for carbonic anhydrase inhibitory and anticancer activities. SAR and QSAR in Environmental Research 34:7, pages 543-567.
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Tarfah Al-Warhi, Mostafa M. Elbadawi, Alessandro Bonardi, Alessio Nocentini, Ahmed A. Al-Karmalawy, Nada Aljaeed, Ohoud J. Alotaibi, Hatem A. Abdel-Aziz, Claudiu T. Supuran & Wagdy M. Eldehna. (2022) Design and synthesis of benzothiazole-based SLC-0111 analogues as new inhibitors for the cancer-associated carbonic anhydrase isoforms IX and XII. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 2635-2643.
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Articles from other publishers (3)

Metin Yildirim, Samet Poyraz & Mehmet Ersatir. (2023) Recent advances on biologically active coumarin-based hybrid compounds. Medicinal Chemistry Research 32:4, pages 617-642.
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Monalisa Mahapatra, Suman K. Mekap, Suvadeep Mal, Jyotirmaya Sahoo, Sanjeeb K. Sahoo & Sudhir K. Paidesetty. (2023) Coumaryl‐sulfonamide moiety: Unraveling their synthetic strategy and specificity toward  h CA IX/XII, facilitating anticancer drug development . Archiv der Pharmazie 356:4.
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Rinshana Fathima Abdul Azeez, Susi Zara, Alessia Ricci, Sanal Dev, Ajeesh Vengamthodi, Fathima Sahla Kavully, Raihan Arikkattel Abdu, Kadeeja Thottungal Kalathil, Mohamed A. Abdelgawad, Bijo Mathew & Simone Carradori. (2022) Integrating N-alkyl amide in the chalcone framework: synthesis and evaluation of its anti-proliferative potential against AGS cancer cell line. Research on Chemical Intermediates 49:1, pages 203-220.
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