Identification of sulphonamide-tethered N-((triazol-4-yl)methyl)isatin derivatives as inhibitors of SARS-CoV-2 main protease

Mai H. ElNaggara Department of Pharmacognosy, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, EgyptCorrespondence[email protected]

https://orcid.org/0000-0001-5481-2053 View further author information

Abdullah A. Elgazara Department of Pharmacognosy, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, Egypt

https://orcid.org/0000-0002-5851-3306 View further author information

Ghada Gamala Department of Pharmacognosy, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, EgyptView further author information

Shimaa M. Hamedb Scientific Research and Innovation Support Unit, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, EgyptView further author information

Zainab M. Elsayedb Scientific Research and Innovation Support Unit, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, EgyptView further author information

Mohamed K. El-Ashreyc Pharmaceutical Chemistry Department, Faculty of Pharmacy, Cairo University, Cairo, EgyptView further author information

Amira Aboodd Chemistry of Natural and microbial products, National Research center, Egypt;e Department of Bioscience, University of Kent, Canterbury, UKView further author information

Mahmoud A. El Hassabf Department of Medicinal Chemistry, Faculty of Pharmacy, King Salman International University (KSIU), EgyptView further author information

Ahmed M. Solimang Department of Microbiology and Immunology, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, EgyptView further author information

Ramadan A. El-Domanyg Department of Microbiology and Immunology, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, EgyptView further author information

Farid A. Badriah Department of Pharmacognosy, Faculty of Pharmacy, Mansoura University, Mansoura, EgyptView further author information

Claudiu T. Supurani Department of NEUROFARBA, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Firenze, Italy

https://orcid.org/0000-0003-4262-0323 View further author information

Wagdy M. Eldehnaj Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, Egypt;k School of Biotechnology, Badr University in Cairo, Badr City, EgyptCorrespondence[email protected]

https://orcid.org/0000-0001-6996-4017 View further author information

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Identification of sulphonamide-tethered N-((triazol-4-yl)methyl)isatin derivatives as inhibitors of SARS-CoV-2 main protease

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Identification of sulphonamide-tethered N-((triazol-4-yl)methyl)isatin derivatives as inhibitors of SARS-CoV-2 main protease

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