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Philosophical Magazine Volume 91, 2011 - Issue 13-15: Twelfth International Workshop on Complex Systems: Andalo (Trento) Italy. 15–18 March 2010
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Original Articles

Comprehensive studies on physical and chemical stability in liquid and glassy states of telmisartan (TEL): solubility advantages given by cryomilled and quenched material

K. Adrjanowicz Institute of Physics, University of Silesia, Uniwersytecka 4, 40-007 Katowice, PolandCorrespondence[email protected]
,
K. Grzybowska Institute of Physics, University of Silesia, Uniwersytecka 4, 40-007 Katowice, Poland
,
K. Kaminski Institute of Physics, University of Silesia, Uniwersytecka 4, 40-007 Katowice, Poland
,
L. Hawelek Institute of Physics, University of Silesia, Uniwersytecka 4, 40-007 Katowice, Poland
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M. Paluch Institute of Physics, University of Silesia, Uniwersytecka 4, 40-007 Katowice, Poland
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D. Zakowiecki Preformulation Department R&D, Pharmaceutical Works Polpharma SA, Pelplinska 19, 83-200 Starogard Gdanski, Poland
Pages 1926-1948 | Received 11 May 2010, Accepted 19 Oct 2010, Published online: 11 Jan 2011

Citations (26)

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Nirmal Kumar Katiyar, Krishanu Biswas & C. S. Tiwary. (2021) Cryomilling as environmentally friendly synthesis route to prepare nanomaterials. International Materials Reviews 66:7, pages 493-532.
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Articles from other publishers (25)

Mustafa Bookwala & Peter L. D. Wildfong. (2023) Re-visitation of Two Models for Predicting Mechanically-Induced Disordering after Cryogenic Impact Milling. Pharmaceutical Research.
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Emeline Dudognon, Florence Danède & Mathieu Guerain. (2021) Milling-Induced Phase Transformations, Underlying Mechanisms, and Resulting Physical States in an Enantiotropic System: The Case of Bezafibrate. Crystal Growth & Design 22:1, pages 363-378.
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Julia L. Shamshina, Robin S. Stein & Noureddine Abidi. (2021) Choosing the right strategy: cryogrinding vs. ball milling – comparing apples to apples . Green Chemistry 23:23, pages 9646-9657.
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Justyna Knapik-Kowalczuk, Marzena Rams-Baron & Marian Paluch. (2021) Current research trends in dielectric relaxation studies of amorphous pharmaceuticals: Physical stability, tautomerism, and the role of hydrogen bonding. TrAC Trends in Analytical Chemistry 134, pages 116097.
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Katarzyna Grzybowska, Andrzej Grzybowski, Justyna Knapik-Kowalczuk, Krzysztof Chmiel, Krzysztof Woyna-Orlewicz, Joanna Szafraniec-Szczęsny, Agata Antosik-Rogóż, Renata Jachowicz, Katarzyna Kowalska-Szojda, Piotr Lodowski & Marian Paluch. (2020) Molecular Dynamics and Physical Stability of Ibuprofen in Binary Mixtures with an Acetylated Derivative of Maltose. Molecular Pharmaceutics 17:8, pages 3087-3105.
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A. Minecka, M. Tarnacka, K. Jurkiewicz, B. Hachuła, K. Kamiński, M. Paluch & E. Kamińska. (2020) Influence of the Internal Structure and Intermolecular Interactions on the Correlation between Structural (α) and Secondary (β-JG) Relaxation below the Glass Transition Temperature in Neat Probucol and Its Binary Mixtures with Modified Saccharides. The Journal of Physical Chemistry B 124:23, pages 4821-4834.
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Emeline Dudognon, Jeanne-Annick Bama & Frédéric Affouard. (2019) Molecular Mobility of Terfenadine: Investigation by Dielectric Relaxation Spectroscopy and Molecular Dynamics Simulation. Molecular Pharmaceutics 16:11, pages 4711-4724.
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Justyna Knapik-Kowalczuk, Zaneta Wojnarowska, Krzysztof Chmiel, Marzena Rams-Baron, Lidia Tajber & Marian Paluch. (2018) Can Storage Time Improve the Physical Stability of Amorphous Pharmaceuticals with Tautomerization Ability Exposed to Compression? The Case of a Chloramphenicol Drug. Molecular Pharmaceutics 15:5, pages 1928-1940.
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Dorota Haznar-Garbacz, Ewa Kaminska, Daniel Zakowiecki, Marek Lachmann, Kamil Kaminski, Grzegorz Garbacz, Przemysław Dorożyński & Piotr Kulinowski. (2017) Melts of Octaacetyl Sucrose as Oral-Modified Release Dosage Forms for Delivery of Poorly Soluble Compound in Stable Amorphous Form. AAPS PharmSciTech 19:2, pages 951-960.
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K. Grzybowska, K. Chmiel, J. Knapik-Kowalczuk, A. Grzybowski, K. Jurkiewicz & M. Paluch. (2017) Molecular Factors Governing the Liquid and Glassy States Recrystallization of Celecoxib in Binary Mixtures with Excipients of Different Molecular Weights. Molecular Pharmaceutics 14:4, pages 1154-1168.
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Justyna Szczurek, Marzena Rams-Baron, Justyna Knapik-Kowalczuk, Agata Antosik, Joanna Szafraniec, Witold Jamróz, Mateusz Dulski, Renata Jachowicz & Marian Paluch. (2017) Molecular Dynamics, Recrystallization Behavior, and Water Solubility of the Amorphous Anticancer Agent Bicalutamide and Its Polyvinylpyrrolidone Mixtures. Molecular Pharmaceutics 14:4, pages 1071-1081.
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Joaquim J. Moura Ramos & Hermínio P. Diogo. (2017) Thermal behavior and molecular mobility in the glassy state of three anti-hypertensive pharmaceutical ingredients. RSC Advances 7:18, pages 10831-10840.
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K. Wolnica, M. Dulski, E. Kaminska, A. Cecotka, M. Tarnacka, R. Wrzalik, K. Kaminski & M. Paluch. (2017) A study on the progress of mutarotation above and below the T g and the relationship between constant rates and structural relaxation times . Physical Chemistry Chemical Physics 19:31, pages 20949-20958.
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Grzegorz Szklarz, Karolina Adrjanowicz, Mateusz Dulski, Justyna Knapik & Marian Paluch. (2016) Dielectric Relaxation Study at Ambient and Elevated Pressure of the Modeled Lipophilic Drug Fenofibrate. The Journal of Physical Chemistry B 120:43, pages 11298-11306.
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Katarzyna Grzybowska, Simone Capaccioli & Marian Paluch. (2016) Recent developments in the experimental investigations of relaxations in pharmaceuticals by dielectric techniques at ambient and elevated pressure. Advanced Drug Delivery Reviews 100, pages 158-182.
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Daniel Zakowiecki, Krzysztof Cal, Kamil Kaminski, Karolina Adrjanowicz, Lech Swinder, Ewa Kaminska & Grzegorz Garbacz. (2015) The Improvement of the Dissolution Rate of Ziprasidone Free Base from Solid Oral Formulations. AAPS PharmSciTech 16:4, pages 922-933.
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Ahmed H.H. Bakheit, Ahmed A. Abd-Elgalil, Bakheit Mustafa, Anzarul Haque & Tanveer A. Wani. 2015. 371 429 .
J. Knapik, Z. Wojnarowska, K. Grzybowska, L. Hawelek, W. Sawicki, K. Wlodarski, J. Markowski & M. Paluch. (2014) Physical Stability of the Amorphous Anticholesterol Agent (Ezetimibe): The Role of Molecular Mobility. Molecular Pharmaceutics 11:11, pages 4280-4290.
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E. Kaminska, M. Tarnacka, K. Kolodziejczyk, M. Dulski, D. Zakowiecki, L. Hawelek, K. Adrjanowicz, M. Zych, G. Garbacz & K. Kaminski. (2014) Impact of low molecular weight excipient octaacetylmaltose on the liquid crystalline ordering and molecular dynamics in the supercooled liquid and glassy state of itraconazole. European Journal of Pharmaceutics and Biopharmaceutics 88:3, pages 1094-1104.
Crossref
E. Kaminska, K. Adrjanowicz, M. Tarnacka, K. Kolodziejczyk, M. Dulski, E. U. Mapesa, D. Zakowiecki, L. Hawelek, I. Kaczmarczyk-Sedlak & K. Kaminski. (2014) Impact of Inter- and Intramolecular Interactions on the Physical Stability of Indomethacin Dispersed in Acetylated Saccharides. Molecular Pharmaceutics 11:8, pages 2935-2947.
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K. Kolodziejczyk, M. Paluch, K. Grzybowska, A. Grzybowski, Z. Wojnarowska, L. Hawelek & J. D. Ziolo. (2013) Relaxation Dynamics and Crystallization Study of Sildenafil in the Liquid and Glassy States. Molecular Pharmaceutics 10:6, pages 2270-2282.
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E. Kaminska, K. Adrjanowicz, K. Kaminski, P. Wlodarczyk, L. Hawelek, K. Kolodziejczyk, M. Tarnacka, D. Zakowiecki, I. Kaczmarczyk-Sedlak, J. Pilch & M. Paluch. (2013) A New Way of Stabilization of Furosemide upon Cryogenic Grinding by Using Acylated Saccharides Matrices. The Role of Hydrogen Bonds in Decomposition Mechanism. Molecular Pharmaceutics 10:5, pages 1824-1835.
Crossref
K. Adrjanowicz, D. Zakowiecki, K. Kaminski, L. Hawelek, K. Grzybowska, M. Tarnacka, M. Paluch & K. Cal. (2012) Molecular Dynamics in Supercooled Liquid and Glassy States of Antibiotics: Azithromycin, Clarithromycin and Roxithromycin Studied by Dielectric Spectroscopy. Advantages Given by the Amorphous State. Molecular Pharmaceutics 9:6, pages 1748-1763.
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K. Grzybowska, M. Paluch, P. Wlodarczyk, A. Grzybowski, K. Kaminski, L. Hawelek, D. Zakowiecki, A. Kasprzycka & I. Jankowska-Sumara. (2012) Enhancement of Amorphous Celecoxib Stability by Mixing It with Octaacetylmaltose: The Molecular Dynamics Study. Molecular Pharmaceutics 9:4, pages 894-904.
Crossref
K. Adrjanowicz, Z. Wojnarowska, K. Grzybowska, L. Hawelek, K. Kaminski, M. Paluch, A. Kasprzycka & K. Walczak. (2011) Molecular dynamics and crystallization phenomenon of supercooled and glassy DNA and RNA nucleosides: -adenosine, -thymidine, and -uridine . Physical Review E 84:5.
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