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Research Article

A New Rapidly Absorbed Paracetamol Tablet Containing Sodium Bicarbonate. II. Dissolution Studies and In Vitro/In Vivo Correlation

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Pages 533-543 | Published online: 30 May 2002

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Claude Dubray, Philippe Maincent & Jean Yves Milon. (2021) From the pharmaceutical to the clinical: the case for effervescent paracetamol in pain management. A narrative review. Current Medical Research and Opinion 37:6, pages 1039-1048.
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Nathalie R. Wingert, Natália O. dos Santos, Sarah C. Campanharo, Elisa S. Simon, Nadia M. Volpato & Martin Steppe. (2018) In vitro dissolution method fitted to in vivo absorption profile of rivaroxaban immediate-release tablets applying in silico data. Drug Development and Industrial Pharmacy 44:5, pages 723-728.
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C.G. Wilson, Cyril P. Clarke, Yan Yan L. Starkey & Geoffrey D. Clarke. (2011) Comparison of a novel fast-dissolving acetaminophen tablet formulation (FD-APAP) and standard acetaminophen tablets using gamma scintigraphy and pharmacokinetic studies. Drug Development and Industrial Pharmacy 37:7, pages 747-753.
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Adrian Dunne, Clare Gaynor & John Davis. (2005) Deconvolution Based Approach for Level A In Vivo-In Vitro Correlation Modelling: Statistical Considerations. Clinical Research and Regulatory Affairs 22:1, pages 1-14.
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Yan Wu, D. O. Kildsig & E. S. Ghaly. (2004) Effect of Hydrodynamic Environment on Tablets Dissolution Rate. Pharmaceutical Development and Technology 9:1, pages 25-37.
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Freja Fredholt, Camilla Di Meo, Stine Sloth, Anette Müllertz & Ragna Berthelsen. (2022) Direct visualizing of paracetamol immediate release tablet disintegration in vivo and in vitro. European Journal of Pharmaceutics and Biopharmaceutics 180, pages 63-70.
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Alok Ranjan & Prateek K. Jha. (2021) Recent Advances in Dissolution Testing and Their Use to Improve In Vitro–In Vivo Correlations in Oral Drug Formulations. Journal of Pharmaceutical Innovation 17:3, pages 1011-1026.
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Kiyohiko Sugano. (2016) Theoretical Investigation of Dissolution Test Criteria for Waiver of Clinical Bioequivalence Study. Journal of Pharmaceutical Sciences 105:6, pages 1947-1951.
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David P. Elder, Martin Kuentz & René Holm. (2016) Pharmaceutical excipients — quality, regulatory and biopharmaceutical considerations. European Journal of Pharmaceutical Sciences 87, pages 88-99.
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Sarin Colón-Useche, Isabel González-Álvarez, Victor Mangas-Sanjuan, Marta González-Álvarez, Pilar Pastoriza, Irene Molina-Martínez, Marival Bermejo & Alfredo García-Arieta. (2015) Investigating the Discriminatory Power of BCS-Biowaiver in Vitro Methodology to Detect Bioavailability Differences between Immediate Release Products Containing a Class I Drug . Molecular Pharmaceutics 12:9, pages 3167-3174.
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H. Kortejärvi, J. Malkki, R. Shawahna, J.-M. Scherrmann, A. Urtti & M. Yliperttula. (2014) Pharmacokinetic simulations to explore dissolution criteria of BCS I and III biowaivers with and without MDR-1 efflux transporter. European Journal of Pharmaceutical Sciences 61, pages 18-26.
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Kiyohiko Sugano. 2012. Biopharmaceutics Modeling and Simulations. Biopharmaceutics Modeling and Simulations 160 205 .
Stephen Chandler. (2013) Estimation of Onset of Analgesia From Simulated Data: Authors' Response. The Journal of Clinical Pharmacology 52:5, pages 779-779.
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Deirdre M. D’Arcy, Anne Marie Healy & Owen I. Corrigan. (2009) Towards determining appropriate hydrodynamic conditions for in vitro in vivo correlations using computational fluid dynamics. European Journal of Pharmaceutical Sciences 37:3-4, pages 291-299.
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Bertold Renner, Geoff Clarke, Tim Grattan, Angelika Beisel, Christian Mueller, Ulrike Werner, Gerd Kobal & Kay Brune. (2007) Caffeine Accelerates Absorption and Enhances the Analgesic Effect of Acetaminophen. The Journal of Clinical Pharmacology 47:6, pages 715-726.
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Sabah Souliman, Stéphanie Blanquet, Eric Beyssac & Jean-Michel Cardot. (2006) A level A in vitro/in vivo correlation in fasted and fed states using different methods: Applied to solid immediate release oral dosage form. European Journal of Pharmaceutical Sciences 27:1, pages 72-79.
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L. Kalantzi, C. Reppas, J.B. Dressman, G.L. Amidon, H.E. Junginger, K.K. Midha, V.P. Shah, S.A. Stavchansky & Dirk M. Barends. (2006) Biowaiver monographs for immediate release solid oral dosage forms: Acetaminophen (paracetamol). Journal of Pharmaceutical Sciences 95:1, pages 4-14.
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A. A. Litvin, G. B. Kolyvanov, V. P. Zherdev & A. P. Arzamastsev. (2004) Relationship between physicochemical characteristics and pharmacokinetic parameters of 1,4-benzodiazepine derivatives. Pharmaceutical Chemistry Journal 38:11, pages 583-586.
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