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Xavier Khawaja, John Dunlop & Dianne Kowal. (2008) Scintillation proximity assay in lead discovery. Expert Opinion on Drug Discovery 3:11, pages 1267-1280.
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Liwen Hua, Danni Wang, Keran Wang, Yuxuan Wang, Jinying Gu, Qiuyue Zhang, Qidong You & Lei Wang. (2023) Design of Tracers in Fluorescence Polarization Assay for Extensive Application in Small Molecule Drug Discovery. Journal of Medicinal Chemistry.
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Jayeon Song, Hansol Kim, Chang Yeol Lee, Junhyeok Yoon, Won Sang Yoo & Hyun Gyu Park. (2021) Identification of thyroid hormone/thyroid hormone receptor interaction based on aptamer-assisted protein-induced fluorescence enhancement. Biosensors and Bioelectronics 191, pages 113444.
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David Reiner & Holger Stark. (2019) Ligand binding kinetics at histamine H3 receptors by fluorescence-polarization with real-time monitoring. European Journal of Pharmacology 848, pages 112-120.
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Asif Iqbal Zia & Subhas Chandra MukhopadhyayAsif Iqbal Zia & Subhas Chandra Mukhopadhyay. 2016. Electrochemical Sensing: Carcinogens in Beverages. Electrochemical Sensing: Carcinogens in Beverages
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Kari Kopra, Markus Kainulainen, Piia Mikkonen, Anita Rozwandowicz-Jansen, Pekka Hänninen & Harri Härmä. (2013) Multiparametric Homogeneous Method for Identification of Ligand Binding to G Protein-Coupled Receptors: Receptor–Ligand Binding and β-Arrestin Assay. Analytical Chemistry 85:4, pages 2276-2281.
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Kari Kopra, Shweta, Eija Martikkala, Pekka Hänninen, Ulla Petäjä-Repo & Harri Härmä. (2013) A homogeneous single-label quenching resonance energy transfer assay for a δ-opioid receptor–ligand using intact cells. The Analyst 138:17, pages 4907.
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David N. LangelaanPascaline NgweniformJan K. Rainey. (2011) Biophysical characterization of G-protein coupled receptor–peptide ligand bindingThis paper is one of a selection of papers published in a Special Issue entitled CSBMCB 53rd Annual Meeting — Membrane Proteins in Health and Disease, and has undergone the Journal’s usual peer review process.. Biochemistry and Cell Biology 89:2, pages 98-105.
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Sung-Hou Lee. (2011) Platform Technologies for Research on the G Protein Coupled Receptor: Applications to Drug Discovery Research. Biomolecules and Therapeutics 19:1, pages 1-8.
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Martin Cottet, Orestis Faklaris, Jurriaan M. Zwier, Eric Trinquet, Jean-Philippe Pin & Thierry Durroux. (2011) Original Fluorescent Ligand-Based Assays Open New Perspectives in G-Protein Coupled Receptor Drug Screening. Pharmaceuticals 4:1, pages 202-214.
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Jean-Philippe Leyris, Thomas Roux, Eric Trinquet, Pascal Verdié, Jean-Alain Fehrentz, Nadia Oueslati, Stéphanie Douzon, Emmanuel Bourrier, Laurent Lamarque, Didier Gagne, Jean-Claude Galleyrand, Céline M’kadmi, Jean Martinez, Sophie Mary, Jean-Louis Banères & Jacky Marie. (2011) Homogeneous time-resolved fluorescence-based assay to screen for ligands targeting the growth hormone secretagogue receptor type 1a. Analytical Biochemistry 408:2, pages 253-262.
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Miklós Kecskés, T. Santhosh Kumar, Lena Yoo, Zhan-Guo Gao & Kenneth A. Jacobson. (2010) Novel Alexa Fluor-488 labeled antagonist of the A2A adenosine receptor: Application to a fluorescence polarization-based receptor binding assay. Biochemical Pharmacology 80:4, pages 506-511.
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Peter Cornelius, Eunsun Lee, Wen Lin, Ruduan Wang, Wendy Werner, Janice A. Brown, Frank Stuhmeier, James G. Boyd & Kim McClure. (2009) Design, Synthesis, and Pharmacology of Fluorescently Labeled Analogs of Serotonin: Application to Screening of the 5-HT2C Receptor. SLAS Discovery 14:4, pages 360-370.
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Peter Spies, Guo Jun Chen & Daniel Gygax. (2008) Establishment of a miniaturized enzyme-linked immunosorbent assay for human transferrin quantification using an intelligent multifunctional analytical plate. Analytical Biochemistry 382:1, pages 35-39.
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G.J. Dear, N. Patel, Alan Weightman, Hans Pirard & Miika Talvitie. (2008) Utilizing a −100°C microplate CCD Imager, yttrium silicate coated 384-microplates and ultra-performance liquid chromatography for improved profiling of radiolabeled drug metabolites in complex biological samples. Journal of Chromatography B 868:1-2, pages 49-57.
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Laura Albizu, Géraldine Teppaz, René Seyer, Hervé Bazin, Hervé Ansanay, Maurice Manning, Bernard Mouillac & Thierry Durroux. (2007) Toward Efficient Drug Screening by Homogeneous Assays Based on the Development of New Fluorescent Vasopressin and Oxytocin Receptor Ligands. Journal of Medicinal Chemistry 50:20, pages 4976-4985.
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Olivier Nosjean, Sophie Souchaud, Clarisse Deniau, Olivier Geneste, Nicolas Cauquil & Jean A. Boutin. (2006) A Simple Theoretical Model for Fluorescence Polarization Binding Assay Development. SLAS Discovery 11:8, pages 949-958.
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Ernest U. Do, Eun Bae Jo, Gyu Choi, Long Zhu Piao, Jaekyoon Shin, Min-Duk Seo, Su-Jin Kang, Bong-Jin Lee, Kang Ho Kim, Jae Bum Kim & Su-il Kim. (2006) Melanocortin 4 receptors interact with antimicrobial frog peptide analogues. Biochemical and Biophysical Research Communications 343:4, pages 1094-1100.
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Wayne R. Leifert, Amanda L. Aloia, Olgatina Bucco, Richard V. Glatz & Edward J. McMurchie. (2005) G-Protein-Coupled Receptors in Drug Discovery: Nanosizing Using Cell-Free Technologies and Molecular Biology Approaches. SLAS Discovery 10:8, pages 765-779.
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Lutea A.A. de Jong, Donald R.A. Uges, Jan Piet Franke & Rainer Bischoff. (2005) Receptor–ligand binding assays: Technologies and Applications. Journal of Chromatography B 829:1-2, pages 1-25.
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Leena Kokko, Nina Johansson, Timo Lövgren & Tero Soukka. (2005) Enzyme Inhibitor Screening Using a Homogeneous Proximity-Based Immunoassay for Estradiol. SLAS Discovery 10:4, pages 348-354.
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Peter J. Greasley & Frank P. Jansen. (2005) G-protein-coupled receptor screening technologies. Drug Discovery Today: Technologies 2:2, pages 163-170.
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Julia OosteromEls J.P. van DoornmalenSendy LobregtMarion BlomenröhrGuido J.R. Zaman. (2005) High-Throughput Screening Using β-Lactamase Reporter-Gene Technology for Identification of Low-Molecular-Weight Antagonists of the Human Gonadotropin Releasing Hormone Receptor. ASSAY and Drug Development Technologies 3:2, pages 143-154.
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Philip Gribbon & Andreas Sewing. (2003) Fluorescence readouts in HTS: no gain without pain?. Drug Discovery Today 8:22, pages 1035-1043.
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Ponnal Nambi & Nambi Aiyar. (2003) G Protein-Coupled Receptors in Drug Discovery. ASSAY and Drug Development Technologies 1:2, pages 305-310.
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