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Synthetic Communications
An International Journal for Rapid Communication of Synthetic Organic Chemistry
Volume 33, 2003 - Issue 3
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Original Articles

An Efficient One-Pot Procedure for Preparation of 2,4(1H,3H)-Quinazolinediones and 2-Thioxoquinazolinone Derivatives Under Microwave Irradiation

Javad Azizian Department of Chemistry, Faculty of Science, Shahid Beheshti University, Tehran, IranCorrespondence[email protected]
,
Ali A. Mohammadi Department of Chemistry, Faculty of Science, Shahid Beheshti University, Tehran, Iran
&
Ali R. Karimi Department of Chemistry, Faculty of Science, Shahid Beheshti University, Tehran, Iran
Pages 415-420 | Received 21 Jan 2002, Published online: 17 Aug 2006

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Ghasem Rezanejade Bardajee, Aseyeh Ghaedi, Shohreh Hekmat, Ghazale Abarashi, Mohammad Mahdavi & Tahmineh Akbarzadeh. (2017) A green and efficient synthesis of 2-thioxoquinazolinone derivatives in water using potassium thiocyanate. Journal of Sulfur Chemistry 38:5, pages 519-529.
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Samir Y. Abbas, Khairy A. M. El-Bayouki & Wahid M. Basyouni. (2016) Utilization of isatoic anhydride in the syntheses of various types of quinazoline and quinazolinone derivatives. Synthetic Communications 46:12, pages 993-1035.
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Gamal A. El-Hiti, Ajaz Hussain, Amany S. Hegazy & Mohammad H. Alotaibi. (2011) Thioxoquinazolines: synthesis, reactions and biological activities. Journal of Sulfur Chemistry 32:4, pages 361-395.
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Javad Azizian, Javad Hosseini, Mohammadkazem Mohammadi & Fatemeh Sheikholeslami. (2010) Efficient Route for the Synthesis of Highly Substituted Pyrroles. Synthetic Communications 40:23, pages 3472-3479.
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Javad Azizian, Mohammad R. Mohammadizadeh, Fatemeh Teimouri, Ali A. Mohammadi & Ali R. Karimi. (2006) Reactions of 6‐Aminouracils: The First Simple, Fast, and Highly Efficient Synthesis of bis(6‐Aminopyrimidonyl)methanes (BAPMs) Using Thermal or Microwave‐Assisted Solvent‐Free Methods. Synthetic Communications 36:23, pages 3631-3638.
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Sherin M. Elfeky, Tariq R. Sobahi, Magdy M. Gineinah & Nesreen S. Ahmed. (2019) Synthesis, biological screening, and molecular docking of quinazolinone and quinazolinethione as phosphodiesterase 7 inhibitors. Archiv der Pharmazie 353:1, pages 1900211.
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Ali A. Mohammadi, Salman Taheri & Saber Askari. (2017) One-Pot Pseudo Five-Component Synthesis of Some New bis(Quinazolinon-4(1 H )-one) Derivatives . Journal of Heterocyclic Chemistry 54:1, pages 484-488.
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Hossein Eshghi, Amir Khojastehnezhad, Farid Moeinpour, Mehdi Bakavoli, Nafiseh Zeinabi & Sadegh Allameh. (2014) Nanomagnetically modified polyphosphoric acid (NiFe2O4@SiO2–PPA): an efficient, fast, and reusable catalyst for the synthesis of 2-thioxoquinazolinones under solvent-free conditions. Research on Chemical Intermediates 41:10, pages 7915-7924.
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Weiwei Liu, Qiang Zhang, Feng Gong, Zhiling Cao & Yunfeng Huo. (2015) A Convenient and Efficient Synthesis of 2-Thioxoquinazolinone Derivatives via Microwave Irradiation. Journal of Heterocyclic Chemistry 52:2, pages 317-321.
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Mehdi Asadi, Shiva Masoomi, Seyed Mostafa Ebrahimi, Mohammad Mahdavi, Mina Saeedi, Abbas Shafiee & Alireza Foroumadi. (2013) Convenient and sequential one-pot route for synthesis of 2-thioxoquinazolinone and quinazolinobenzothiazinedione derivatives. Monatshefte für Chemie - Chemical Monthly 145:3, pages 497-504.
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Ali A. Mohammadi, Armin Hadadzahmatkesh & Mohammad R. Asghariganjeh. (2011) FeNH4(SO4)2·12H2O (alum)-catalyzed preparation of 1,4-dihydropyridines: improved conditions for the Hantzsch reaction. Monatshefte für Chemie - Chemical Monthly 143:6, pages 931-933.
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S. Allameh, M.M. Heravi, M.M. Hashemi & F.F. Bamoharram. (2011) Synthesis of 3-(aryl)-2-thioxo-2,3-dihydroquinazolin-4(1H)-one derivatives using heteropolyacids as green, heterogeneous and recyclable catalysts. Chinese Chemical Letters 22:2, pages 131-134.
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Zhaoguang Li, He Huang, Hongbin Sun, Hualiang Jiang & Hong Liu. (2008) Microwave-Assisted Efficient and Convenient Synthesis of 2,4(1 H ,3 H )-Quinazolinediones and 2-Thioxoquinazolines . Journal of Combinatorial Chemistry 10:3, pages 484-486.
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Ali Asghar Mohammadi, Ali A. Mohammadi, Javad Azizian, Armin Hadadzahmatkesh & Mohammad R. Asghariganjeh. (2008) Green Protocol for the Friedländer Synthesis: KAl(SO4)2·12H2O-SiO2 (Alum- SiO2), a Highly Efficient Catalyst in the Synthesis of Quinolines. HETEROCYCLES 75:4, pages 947.
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G.W. Rewcastle. 2008. Comprehensive Heterocyclic Chemistry III. Comprehensive Heterocyclic Chemistry III 117 272 .
Yanling Huang, Cuifen Lu, Zuxing Chen & Guichun Yang. (2009) Traceless synthesis of quinazoline‐2,4‐diones by curtius rearrangement reaction using poly(ethylene glycol) as soluble polymeric support. Journal of Heterocyclic Chemistry 44:6, pages 1421-1424.
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Javad Azizian, Ali A. Mohammadi, M. Kohshari, Ali R. Karimi & Mohammad R. Mohammadizadeh. (2009) Biginelli‐like three component reaction: Synthesis of some new ethyl 6‐ethoxycarbonylmethyl‐4‐aryl‐2‐oxo‐1,2,3,4‐tetrahydropyrimidine‐5‐carboxylate derivatives. Journal of Heterocyclic Chemistry 44:2, pages 455-458.
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W. Russell Bowman, Mark R. J. Elsegood, Tobias Stein & George W. Weaver. (2007) Radical reactions with 3H-quinazolin-4-ones: synthesis of deoxyvasicinone, mackinazolinone, luotonin A, rutaecarpine and tryptanthrin. Org. Biomol. Chem. 5:1, pages 103-113.
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Onorato Campopiano & David J. St. JeanJr.Jr.. 2001. Encyclopedia of Reagents for Organic Synthesis. Encyclopedia of Reagents for Organic Synthesis.
Javad Azizian, Farhad Hatamjafari & Ali Reza Karimi. (2006) Four component and solvent-free synthesis of some new spiro-1,4-dihydropyridines on solid support montmorillonite K10. Journal of Heterocyclic Chemistry 43:5, pages 1349-1352.
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Yoshinao Tamaru & Paul J. Nichols. 2001. Encyclopedia of Reagents for Organic Synthesis. Encyclopedia of Reagents for Organic Synthesis.
Javad Azizian, Ali Reza Karimi, Ebrahim Soleimani, Ali A. Mohammadi & Mohammad R. Mohammadizadeh. (2006) Highly functionalized dihydrofuran derivatives: Synthesis by diastereoselective intramolecular Wittig reaction. Heteroatom Chemistry 17:4, pages 277-279.
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Javad Azizian, Ali A. Mohammadi, Ebrahim Soleimani, Ali R. Karimi & Mohammad R. Mohammadizadeh. (2009) A stereoselective three‐component reaction: One‐pot synthesis of cis ‐isoquinolonic acids catalyzed by silica sulfuric acid under mild and heterogeneous conditions . Journal of Heterocyclic Chemistry 43:1, pages 187-190.
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Javad Azizian, Ali Reza Karimi, Zahra Kazemizadeh, Ali A. Mohammadi & Mohammad R. Mohammadizadeh. (2005) A synthetic route to 11-(1H-pyrrol-1-yl)-11H-indeno[1,2-b]quinoxaline derivatives exploiting a three-component coupling strategy under microwave irradiation. Tetrahedron Letters 46:36, pages 6155-6157.
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Javad Azizian, Mohammad R. Mohammadizadeh, Narges Karimi, Ali A. Mohammadi & Ali R. Karimi. (2005) One-Pot Synthesis of Alkyl Indeno[1,2-b]quinoxalin-11-ylideneacetates under Solvent-free Conditions. HETEROCYCLES 65:1, pages 143.
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Minoo Dabiri, Peyman Salehi, Mohammad S. Khajavi & Ali A. Mohammadi. (2004) Microwave-assisted One-Pot Three Component Synthesis of Some New 4(3H)-Quinazolinone Derivatives. HETEROCYCLES 63:6, pages 1417.
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Javad Azizian, Ali A. Mohammadi, F. Ardakani, Ali R. Karimi & Mohammad R. Mohammadizadeh. (2004) A Simple and Efficient Synthesis of New 6-Arylimino-6H-indolo[2,1-b]quinazolin-12-ones under Microwave Irradiation. HETEROCYCLES 63:4, pages 791.
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Javad Azizian, Ali A. Mohammadi & Ali R. Karimi. (2003) An Efficient One‐Pot Procedure for Preparation of 2,4(1H,3H)‐Quinazolinediones and 2‐Thioxoquinazolinone Derivatives under Microwave Irradiation.. ChemInform 34:27.
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