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Article

Regulation of ABCG2 Expression at the 3′ Untranslated Region of Its mRNA through Modulation of Transcript Stability and Protein Translation by a Putative MicroRNA in the S1 Colon Cancer Cell Line

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Pages 5147-5161 | Received 27 Feb 2008, Accepted 11 Jun 2008, Published online: 27 Mar 2023

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Crossref
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Crossref
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Crossref
Xin An, Cesar Sarmiento, Tao Tan & Hua Zhu. (2017) Regulation of multidrug resistance by microRNAs in anti-cancer therapy. Acta Pharmaceutica Sinica B 7:1, pages 38-51.
Crossref
Yuanzhang Fang, Lu Zhang, Zhenghu Li, Yujing Li, Cheng Huang & Xiongbin Lu. 2017. MiRNAs in Differentiation and Development. MiRNAs in Differentiation and Development 1 49 .
Dagmara Szkolnicka, Baltasar Lucendo-Villarin, Joanna K. Moore, Kenneth J. Simpson, Stuart J. Forbes & David C. Hay. (2016) Reducing Hepatocyte Injury and Necrosis in Response to Paracetamol Using Noncoding RNAs. Stem Cells Translational Medicine 5:6, pages 764-772.
Crossref
Kai Wu, Yang Yang, Jia Zhao & Song Zhao. (2016) BAG3-mediated miRNA let-7g and let-7i inhibit proliferation and enhance apoptosis of human esophageal carcinoma cells by targeting the drug transporter ABCC10. Cancer Letters 371:1, pages 125-133.
Crossref
A.-M. Yu, Y. Tian, M.-J. Tu, P. Y. Ho & J. L. Jilek. (2015) MicroRNA Pharmacoepigenetics: Posttranscriptional Regulation Mechanisms behind Variable Drug Disposition and Strategy to Develop More Effective Therapy. Drug Metabolism and Disposition 44:3, pages 308-319.
Crossref
HYUN-HYE MOON, SUNG-HEE KIM & JA-LOK KU. (2016) Correlation between the promoter methylation status of ATP-binding cassette sub-family G member 2 and drug sensitivity in colorectal cancer cell lines. Oncology Reports 35:1, pages 298-306.
Crossref
Kai-Xuan Sun, Jin-Wen Jiao, Shuo Chen, Bo-Liang Liu & Yang Zhao. (2015) MicroRNA-186 induces sensitivity of ovarian cancer cells to paclitaxel and cisplatin by targeting ABCB1. Journal of Ovarian Research 8:1.
Crossref
Yueping Zhan, Fenfen Xiang, Rong Wu, Jian Xu, Zhenhua Ni, Jiemin Jiang & Xiangdong Kang. (2015) MiRNA-149 modulates chemosensitivity of ovarian cancer A2780 cells to paclitaxel by targeting MyD88. Journal of Ovarian Research 8:1.
Crossref
Kenneth K.W. To, W.W. Leung & Simon S.M. Ng. (2015) Exploiting a novel miR-519c–HuR–ABCG2 regulatory pathway to overcome chemoresistance in colorectal cancer. Experimental Cell Research 338:2, pages 222-231.
Crossref
Jennifer Bolleyn, Joery De Kock, Robim Marcelino Rodrigues, Mathieu Vinken, Vera Rogiers & Tamara Vanhaecke. (2014) MicroRNAs as key regulators of xenobiotic biotransformation and drug response. Archives of Toxicology 89:9, pages 1523-1541.
Crossref
KS Burgess, S Philips, EA Benson, Z Desta, A Gaedigk, R Gaedigk, MW Segar, Y Liu & TC Skaar. (2015) Age-Related Changes in MicroRNA Expression and Pharmacogenes in Human Liver. Clinical Pharmacology & Therapeutics 98:2, pages 205-215.
Crossref
Mei-Mei Li, Balasubrahmanyam Addepalli, Mei-Juan Tu, Qiu-Xia Chen, Wei-Peng Wang, Patrick A. Limbach, Janine M. LaSalle, Su Zeng, Min Huang & Ai-Ming Yu. (2015) Chimeric MicroRNA-1291 Biosynthesized Efficiently in Escherichia coli Is Effective to Reduce Target Gene Expression in Human Carcinoma Cells and Improve Chemosensitivity . Drug Metabolism and Disposition 43:7, pages 1129-1136.
Crossref
Y He, J R Chevillet, G Liu, T K Kim & K Wang. (2015) The effects of microRNA on the absorption, distribution, metabolism and excretion of drugs. British Journal of Pharmacology 172:11, pages 2733-2747.
Crossref
Nirmalya Dasgupta, Bhupesh Kumar Thakur, Atri Ta & Santasabuj Das. (2015) Caveolin-1 is transcribed from a hypermethylated promoter to mediate colonocyte differentiation and apoptosis. Experimental Cell Research 334:2, pages 323-336.
Crossref
Qingcheng Mao & Jashvant D. Unadkat. (2014) Role of the Breast Cancer Resistance Protein (BCRP/ABCG2) in Drug Transport—an Update. The AAPS Journal 17:1, pages 65-82.
Crossref
Shuo Chen, Xi Chen, Yin-Ling Xiu, Kai-Xuan Sun, Zhi-Hong Zong & Yang Zhao. (2014) microRNA 490-3P enhances the drug-resistance of human ovarian cancer cells. Journal of Ovarian Research 7:1.
Crossref
Can Zong, Jun Wang & Tie-Mei Shi. (2014) MicroRNA 130b enhances drug resistance in human ovarian cancer cells. Tumor Biology 35:12, pages 12151-12156.
Crossref
Mei-Mei Li, Wei-Peng Wang, Wen-Juan Wu, Min Huang & Ai-Ming Yu. (2014) Rapid Production of Novel Pre-MicroRNA Agent hsa-mir-27b in Escherichia coli Using Recombinant RNA Technology for Functional Studies in Mammalian Cells . Drug Metabolism and Disposition 42:11, pages 1791-1795.
Crossref
Xiaolan Zhu, Yuefeng Li, Chanjuan Xie, Xinming Yin, Yueqin Liu, Yuan Cao, Yue Fang, Xin Lin, Yao Xu, Wenlin Xu, Huiling Shen & Jian Wen. (2014) miR-145 sensitizes ovarian cancer cells to paclitaxel by targeting Sp1 and Cdk6. International Journal of Cancer 135:6, pages 1286-1296.
Crossref
Jenny Wong. (2014) Regulation of a TrkB Alternative Transcript by microRNAs. Dementia and Geriatric Cognitive Disorders Extra 4:3, pages 364-374.
Crossref
Agnes Basseville, Robert W. Robey, Julian C. Bahr & Susan E. Bates. 2014. Drug Transporters. Drug Transporters 187 221 .
Feng Li & Ram I. Mahato. (2014) MicroRNAs and Drug Resistance in Prostate Cancers. Molecular Pharmaceutics 11:8, pages 2539-2552.
Crossref
Ke Shen, Rurong Mao, Li Ma, Yueqi Li, Yanyan Qiu, Daling Cui, Vanminh Le, Peihao Yin, Lei Ni & Jianwen Liu. (2014) Post-transcriptional regulation of the tumor suppressor miR-139-5p and a network of miR-139-5p-mediated mRNA interactions in colorectal cancer. FEBS Journal 281:16, pages 3609-3624.
Crossref
Anneke N. Werk, Henrike Bruckmueller, Sierk Haenisch & Ingolf Cascorbi. (2014) Genetic variants may play an important role in mRNA–miRNA interaction. Pharmacogenetics and Genomics 24:6, pages 283-291.
Crossref
Andreas Gisel, Mirna Valvano, Imane El Idrissi, Patrizia Nardulli, Amalia Azzariti, Antonio Carrieri, Marialessandra Contino & Nicola Colabufo. (2014) miRNAs for the Detection of MultiDrug Resistance: Overview and Perspectives. Molecules 19:5, pages 5611-5623.
Crossref
Sierk Haenisch, Anneke Nina Werk & Ingolf Cascorbi. (2014) MicroRNAs and their relevance to ABC transporters. British Journal of Clinical Pharmacology 77:4, pages 587-596.
Crossref
Zhuo Dong, Zhiwei Zhong, Lihua Yang, Shaomin Wang & Zhaohui Gong. (2014) MicroRNA-31 inhibits cisplatin-induced apoptosis in non-small cell lung cancer cells by regulating the drug transporter ABCB9. Cancer Letters 343:2, pages 249-257.
Crossref
In-Wha Kim, Nayoung Han, Gilbert J. Burckart & Jung Mi Oh. (2014) Epigenetic Changes in Gene Expression for Drug-Metabolizing Enzymes and Transporters. Pharmacotherapy: The Journal of Human Pharmacology and Drug Therapy 34:2, pages 140-150.
Crossref
Sara Donzelli, Federica Mori, Francesca Biagioni, Teresa Bellissimo, Claudio Pulito, Paola Muti, Sabrina Strano & Giovanni Blandino. (2014) MicroRNAs: short non-coding players in cancer chemoresistance. Molecular and Cellular Therapies 2:1, pages 16.
Crossref
Zhaohui Gong, Zhuo Dong, Lihua Yang, Jie Yang, Jingqiu Li, Yanping Le, Shaomin Wang, Meng Ye & Hui-Kuan Lin. 2014. MicroRNA Targeted Cancer Therapy. MicroRNA Targeted Cancer Therapy 51 82 .
Çiğir Biray Avci & Yusuf Baran. 2014. miRNomics: MicroRNA Biology and Computational Analysis. miRNomics: MicroRNA Biology and Computational Analysis 311 325 .
Kenneth KW To. (2013) MicroRNA: a prognostic biomarker and a possible druggable target for circumventing multidrug resistance in cancer chemotherapy. Journal of Biomedical Science 20:1.
Crossref
Magnus Ingelman-Sundberg, Xiao-Bo Zhong, Oliver Hankinson, Sudheer Beedanagari, Ai-Ming Yu, Lai Peng & Yoichi Osawa. (2013) Potential Role of Epigenetic Mechanisms in the Regulation of Drug Metabolism and Transport. Drug Metabolism and Disposition 41:10, pages 1725-1731.
Crossref
Yu-Zhuo Pan, Amy Zhou, Zihua Hu & Ai-Ming Yu. (2013) Small Nucleolar RNA-Derived MicroRNA hsa-miR-1291 Modulates Cellular Drug Disposition through Direct Targeting of ABC Transporter ABCC1. Drug Metabolism and Disposition 41:10, pages 1744-1751.
Crossref
Meng-Tao Ma, Miao He, Yan Wang, Xu-Yang Jiao, Lin Zhao, Xue-Feng Bai, Zhao-Jin Yu, Hui-Zhe Wu, Ming-Li Sun, Zhi-Guo Song & Min-Jie Wei. (2013) MiR-487a resensitizes mitoxantrone (MX)-resistant breast cancer cells (MCF-7/MX) to MX by targeting breast cancer resistance protein (BCRP/ABCG2). Cancer Letters 339:1, pages 107-115.
Crossref
Michela Garofalo & Carlo M. Croce. (2013) MicroRNAs as therapeutic targets in chemoresistance. Drug Resistance Updates 16:3-5, pages 47-59.
Crossref
Xuyang Jiao, Lin Zhao, Mengtao Ma, Xuefeng Bai, Miao He, Yuanyuan Yan, Yan Wang, Qiuchen Chen, Xinnan Zhao, Mingyi Zhou, Zeshi Cui, Zhihong Zheng, Enhua Wang & Minjie Wei. (2013) MiR-181a enhances drug sensitivity in mitoxantone-resistant breast cancer cells by targeting breast cancer resistance protein (BCRP/ABCG2). Breast Cancer Research and Treatment 139:3, pages 717-730.
Crossref
Y. Sun, Y. Fu, Y. Li & A. Xu. (2012) Genome-wide alternative polyadenylation in animals: insights from high-throughput technologies. Journal of Molecular Cell Biology 4:6, pages 352-361.
Crossref
Yi An, Alan Kiang, Jay Patrick Lopez, Selena Z. Kuo, Michael Andrew Yu, Eric L. Abhold, Jocelyn S. Chen, Jessica Wang-Rodriguez & Weg M. Ongkeko. (2012) Cigarette Smoke Promotes Drug Resistance and Expansion of Cancer Stem Cell-Like Side Population. PLoS ONE 7:11, pages e47919.
Crossref
Yun Chen, Ya-Hui Tsai, Yu Fang & Sheng-Hong Tseng. (2012) Micro-RNA-21 regulates the sensitivity to cisplatin in human neuroblastoma cells. Journal of Pediatric Surgery 47:10, pages 1797-1805.
Crossref
Raji Padmanabhan, Kevin G. Chen, Jean-Pierre Gillet, Misty Handley, Barbara S. Mallon, Rebecca S. Hamilton, Kyeyoon Park, Sudhir Varma, Michele G. Mehaffey, Pamela G. Robey, Ronald D. G. McKay & Michael M. Gottesman. (2012) Regulation and Expression of the ATP-Binding Cassette Transporter ABCG2 in Human Embryonic Stem Cells . Stem Cells 30:10, pages 2175-2187.
Crossref
Sierk Haenisch & Ingolf Cascorbi. (2012) miRNAs as mediators of drug resistance. Epigenomics 4:4, pages 369-381.
Crossref
Grace M. Y. Cheng & Kenneth K. W. To. (2012) Adverse Cell Culture Conditions Mimicking the Tumor Microenvironment Upregulate ABCG2 to Mediate Multidrug Resistance and a More Malignant Phenotype. ISRN Oncology 2012, pages 1-10.
Crossref
Benjamin Boyerinas, Sun-Mi Park, Andrea E. Murmann, Katja Gwin, Anton G. Montag, Marion Zillhardt, You-Jia Hua, Ernst Lengyel & Marcus E. Peter. (2012) Let-7 modulates acquired resistance of ovarian cancer to Taxanes via IMP-1-mediated stabilization of multidrug resistance 1. International Journal of Cancer 130:8, pages 1787-1797.
Crossref
Anuradha Ramamoorthy, Lang Li, Andrea Gaedigk, L. DiAnne Bradford, Eric A. Benson, David A. Flockhart & Todd C. Skaar. (2012) In Silico and In Vitro Identification of MicroRNAs That Regulate Hepatic Nuclear Factor 4α Expression. Drug Metabolism and Disposition 40:4, pages 726-733.
Crossref
Karthika Natarajan, Yi Xie, Maria R. Baer & Douglas D. Ross. (2012) Role of breast cancer resistance protein (BCRP/ABCG2) in cancer drug resistance. Biochemical Pharmacology 83:8, pages 1084-1103.
Crossref
Ai-Ming Yu & Yu-Zhuo Pan. (2012) Noncoding microRNAs: small RNAs play a big role in regulation of ADME?. Acta Pharmaceutica Sinica B 2:2, pages 93-101.
Crossref
Elisa Giovannetti, Ayse Erozenci, Jorn Smit, Romano Danesi & Godefridus J. Peters. (2012) Molecular mechanisms underlying the role of microRNAs (miRNAs) in anticancer drug resistance and implications for clinical practice. Critical Reviews in Oncology/Hematology 81:2, pages 103-122.
Crossref
Alice C. Rodrigues, Xin Li, Laura Radecki, Yu-Zhuo Pan, Jerrold C. Winter, Min Huang & Ai-Ming Yu. (2011) MicroRNA expression is differentially altered by xenobiotic drugs in different human cell lines. Biopharmaceutics & Drug Disposition 32:6, pages 355-367.
Crossref
Sierk Haenisch, Sandra Laechelt, Henrike Bruckmueller, Anneke Werk, Andreas Noack, Oliver Bruhn, Cornelia Remmler & Ingolf Cascorbi. (2011) Down-Regulation of ATP-Binding Cassette C2 Protein Expression in HepG2 Cells after Rifampicin Treatment Is Mediated by MicroRNA-379. Molecular Pharmacology 80:2, pages 314-320.
Crossref
Cheng-Fen Chen, Xiaolong He, Ahmet Dirim Arslan, Yin-Yuan Mo, William C. Reinhold, Yves Pommier & William T. Beck. (2011) Novel Regulation of Nuclear Factor-YB by miR-485-3p Affects the Expression of DNA Topoisomerase IIα and Drug Responsiveness . Molecular Pharmacology 79:4, pages 735-741.
Crossref
K Moitra, H Lou & M Dean. (2011) Multidrug Efflux Pumps and Cancer Stem Cells: Insights Into Multidrug Resistance and Therapeutic Development. Clinical Pharmacology & Therapeutics 89:4, pages 491-502.
Crossref
Xin Li, Yu-Zhuo Pan, Gail M. Seigel, Zi-Hua Hu, Min Huang & Ai-Ming Yu. (2011) Breast cancer resistance protein BCRP/ABCG2 regulatory microRNAs (hsa-miR-328, -519c and -520h) and their differential expression in stem-like ABCG2+ cancer cells. Biochemical Pharmacology 81:6, pages 783-792.
Crossref
Rossella Rota, Roberta Ciarapica, Antonio Giordano, Lucio Miele & Franco Locatelli. (2011) MicroRNAs in rhabdomyosarcoma: pathogenetic implications and translational potentiality. Molecular Cancer 10:1, pages 120.
Crossref
Erik A.C. Wiemer. 2011. MicroRNAs in Cancer Translational Research. MicroRNAs in Cancer Translational Research 449 483 .
Henriette E. Meyer zu Schwabedissen & Heyo K. Kroemer. 2011. Drug Transporters. Drug Transporters 325 371 .
Paul Cao, Zhiyong Deng, Meimei Wan, Weiwei Huang, Scott D Cramer, Jianfeng Xu, Ming Lei & Guangchao Sui. (2010) MicroRNA-101 negatively regulates Ezh2 and its expression is modulated by androgen receptor and HIF-1α/HIF-1β. Molecular Cancer 9:1.
Crossref
F Wang, X Xue, J Wei, Y An, J Yao, H Cai, J Wu, C Dai, Z Qian, Z Xu & Y Miao. (2010) hsa-miR-520h downregulates ABCG2 in pancreatic cancer cells to inhibit migration, invasion, and side populations. British Journal of Cancer 103:4, pages 567-574.
Crossref
J Ma, C Dong & C Ji. (2010) MicroRNA and drug resistance. Cancer Gene Therapy 17:8, pages 523-531.
Crossref
Dominique Cheneval, Tania Kastelic, Peter Fuerst & Christian N. Parker. (2010) A Review of Methods to Monitor the Modulation of mRNA Stability: A Novel Approach to Drug Discovery and Therapeutic Intervention. SLAS Discovery 15:6, pages 609-622.
Crossref
Curtis Balch, Daniela E Matei, Tim H-M Huang & Kenneth P Nephew. (2010) Role of epigenomics in ovarian and endometrial cancers. Epigenomics 2:3, pages 419-447.
Crossref
Sook Wah Yee, Ligong Chen & Kathleen M Giacomini. (2010) Pharmacogenomics of membrane transporters: past, present and future. Pharmacogenomics 11:4, pages 475-479.
Crossref
Xi-wei Ding, Jun-hua Wu & Chun-ping Jiang. (2010) ABCG2: A potential marker of stem cells and novel target in stem cell and cancer therapy. Life Sciences 86:17-18, pages 631-637.
Crossref
Takeshi HIROTA, Ichiro IEIRI & Shun HIGUCHI. (2010) . Rinsho yakuri/Japanese Journal of Clinical Pharmacology and Therapeutics 41:3, pages 105S-106S.
Crossref
Anna Maria Calcagno & Suresh V. Ambudkar. 2010. Multi-Drug Resistance in Cancer. Multi-Drug Resistance in Cancer 77 93 .
Tongsen Zheng, Jiabei Wang, Xi Chen & Lianxin Liu. (2010) Role of microRNA in anticancer drug resistance. International Journal of Cancer 126:1, pages 2-10.
Crossref
Eran E. Bram, Michal Stark, Shachar Raz & Yehuda G. Assaraf. (2009) Chemotherapeutic Drug-Induced ABCG2 Promoter Demethylation as a Novel Mechanism of Acquired Multidrug Resistance. Neoplasia 11:12, pages 1359-IN11.
Crossref
Kenneth K.W. To, Robert W. Robey, Turid Knutsen, Zhirong Zhan, Thomas Ried & Susan E. Bates. (2009) Escape from hsa-miR-519c enables drug-resistant cells to maintain high expression of ABCG2. Molecular Cancer Therapeutics 8:10, pages 2959-2968.
Crossref
Yu-Zhuo Pan, Wenqing Gao & Ai-Ming Yu. (2009) MicroRNAs Regulate CYP3A4 Expression via Direct and Indirect Targeting. Drug Metabolism and Disposition 37:10, pages 2112-2117.
Crossref
XueMei Wu & HuaSheng Xiao. (2009) miRNAs modulate the drug response of tumor cells. Science in China Series C: Life Sciences 52:9, pages 797-801.
Crossref
Aoife J Lowery, Nicola Miller, Amanda Devaney, Roisin E McNeill, Pamela A Davoren, Christophe Lemetre, Vladimir Benes, Sabine Schmidt, Jonathon Blake, Graham Ball & Michael J Kerin. (2009) MicroRNA signatures predict oestrogen receptor, progesterone receptor and HER2/neureceptor status in breast cancer. Breast Cancer Research 11:3.
Crossref
Yu-Zhuo Pan, Marilyn E. Morris & Ai-Ming Yu. (2009) MicroRNA-328 Negatively Regulates the Expression of Breast Cancer Resistance Protein (BCRP/ABCG2) in Human Cancer Cells. Molecular Pharmacology 75:6, pages 1374-1379.
Crossref
A Gomez & M Ingelman-Sundberg. (2009) Pharmacoepigenetics: Its Role in Interindividual Differences in Drug Response. Clinical Pharmacology & Therapeutics 85:4, pages 426-430.
Crossref
Robert W. Robey, Kenneth K.K. To, Orsolya Polgar, Marius Dohse, Patricia Fetsch, Michael Dean & Susan E. Bates. (2009) ABCG2: A perspective. Advanced Drug Delivery Reviews 61:1, pages 3-13.
Crossref
Gergely Szakács, Kenneth Kin Wah, Orsolya Polgár, Robert W. Robey & Susan E. Bates. 2009. Drug Resistance in Cancer Cells. Drug Resistance in Cancer Cells 1 20 .
William Kong, Jian-Jun Zhao, Lili He & Jin Q. Cheng. (2009) Strategies for profiling MicroRNA expression. Journal of Cellular Physiology 218:1, pages 22-25.
Crossref
Ágota Apáti, Tamás I. Orbán, Nóra Varga, Andrea Németh, Anita Schamberger, Virág Krizsik, Boglárka Erdélyi-Belle, László Homolya, György Várady, Rita Padányi, Éva Karászi, Evelien W.M. Kemna, Katalin Német & Balázs Sarkadi. (2008) High level functional expression of the ABCG2 multidrug transporter in undifferentiated human embryonic stem cells. Biochimica et Biophysica Acta (BBA) - Biomembranes 1778:12, pages 2700-2709.
Crossref

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